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知网期刊论文(231)
在“
Elsevier电子期刊
”中,
命中:
209
条,耗时:0.0319766 秒
在所有数据库中总计命中:
883
条
1.
Polysubstituted and ring-fused pyridazine systems from tetrafluoropyridazine
作者:
Graham Pattison
a
;
Graham Sandford
a
;
graham.sandford@durham.ac.uk
;
Ian Wilson
a
;
Dmitrii S. Yufit
a
;
Judith A.K. Howard
a
;
John A. Christopher
b
;
David D. Miller
b
关键词:
Heterocyclic
scaffold
;
Perfluoroheterocycle
;
Multi-functional pyridazine
;
Nucleophilic aromatic substitution
刊名:Tetrahedron
出版年:2017
2.
Synthetic approach and functionalization of novel 4-anilinoquinolino-quinazoline
heterocyclic
scaffold
s
作者:
Chamseddine Derabli
a
;
Raouf Boulcina
a
;
b
;
r.boulcina@univ-batna2.dz
;
Gilbert Kirsch
c
;
Abdelmadjid Debache
a
关键词:
Quinazoline derivatives
;
4-Anilinoquinazolines
;
Quinolino-quinazoline hybrids
;
SNAr reaction
刊名:Tetrahedron
出版年:2017
3.
Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole
scaffold
s as potent tumor associated human carbonic anhydrase IX and XII inhibitors
作者:
Rajiv Kumar
a
;
Silvia Bua
b
;
Sita Ram
a
;
Sonia Del Prete
b
;
c
;
Clemente Capasso
c
;
Claudiu T. Supuran
b
;
claudiu.supuran@unifi.it
;
Pawan K. Sharma
a
;
pksharma@kuk.ac.in
关键词:
Imidazothiadiazoles
;
Thiazolotriazoles
;
Benzenesulfonamide
;
Carbonic anhydrase isoforms I
;
II
;
IX
;
XII
;
Acetazolamide
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
4.
Synthesis and evaluation of the anti-proliferative activity of diaryl-3-pyrrolin-2-ones and fused analogs
作者:
Patricia Mowery
a
;
mowery@hws.edu
;
Fernando Banales Mejia
b
;
Courtney L. Franceschi
b
;
Maeve H. Kean
b
;
Deborah O. Kwansare
b
;
Megan M. Lafferty
b
;
Namita D. Neerukonda
a
;
Carly E. Rolph
a
;
b
;
Nathanyal J. Truax
b
;
Erin T. Pelkey
b
;
pelkey@hws.edu
关键词:
Indoles
;
Lactams
;
Anti-cancer
;
MTT
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
5.
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT
7
and 5-HT
1A
receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
作者:
Sebastiano Intagliata
a
;
1
;
s.intagliata@studium.unict.it
;
Maria N. Modica
a
;
1
;
Valeria Pittalà
;
a
;
Loredana Salerno
a
;
Maria A. Siracusa
a
;
Alfredo Cagnotto
b
;
Mario Salmona
b
;
Rafał Kurczab
c
;
Giuseppe Romeo
a
关键词:
5-HT7 receptor ligands
;
5-HT1A receptor ligands
;
Long-chain arylpiperazines
;
Molecular modeling
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
6.
Differential characterization using readily accessible NMR experiments of novel N- and O-alkylated quinolin-4-ol, 1,5-naphthyridin-4-ol and quinazolin-4-ol derivatives with antimycobacterial activity
作者:
Eleni Pitta
a
;
Olga Balabon
a
;
Maciej K. Rogacki
a
;
Jesú
;
s Gó
;
mez
b
;
Fraser Cunningham
b
;
Jurgen Joosens
a
;
Koen Augustyns
a
;
Pieter van der Veken
a
;
pieter.vanderveken@uantwerpen.be
;
Robert Bates
b
;
robert.h.bates@gsk.com
关键词:
Quinolinol
;
Naphthyridinol
;
Quinazolinol
;
Tuberculosis
;
Alkylation
;
Regioselectivity
;
NMR
刊名:European Journal of Medicinal Chemistry
出版年:2017
7.
DABCO functionalized dicationic ionic liquid (DDIL): A novel green benchmark in multicomponent synthesis of
heterocyclic
scaffold
s under sustainable reaction conditions
作者:
Trushant Lohar
;
Arjun Kumbhar
;
Madhuri Barge
;
Rajshri Salunkhe
;
rsschem1@gmail.com
关键词:
DABCO functionalized ionic liquids
;
Grinding
;
Ultrasound
;
Multicomponent reactions
刊名:Journal of Molecular Liquids
出版年:2016
8.
Multifunctional
heterocyclic
scaffold
s for hybrid Lewis acid/Lewis base catalysis of carbon-carbon bond formation
作者:
Dennis Wiedenhoeft
;
Adam R. Benoit
;
Yibiao Wu
;
Jacob D. Porter
;
Elisia Meyle
;
Teresa H.W. Yeung
;
Raechel Huff
;
Sergey V. Lindeman
;
Chris Dockendorff
;
christopher.dockendorff@mu.edu" class="auth_mail" title="E-mail the corresponding author
关键词:
Hybrid catalyst
;
Organocatalyst
;
Lewis acid
;
Heterocycle
;
Aldol reaction
刊名:Tetrahedron
出版年:2016
9.
Design and synthesis of thiourea derivatives with sulfur-containing
heterocyclic
scaffold
s as potential tyrosinase inhibitors
作者:
Pingping Liu
;
Chen Shu
;
Lujie Liu
;
Qingchun Huang
;
Yanqing Peng
;
yqpeng@ecust.edu.cn" class="auth_mail" title="E-mail the corresponding author
关键词:
Tyrosinase
;
Inhibition
;
Thiourea derivatives
;
Thiadiazol
;
Thiophene
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
10.
Novel fluorinated benzimidazole-based
scaffold
s and their anticancer activity in vitro
作者:
Avninder S. Bhambra
a
;
;
Mark Edgar
b
;
Mark R.J. Elsegood
b
;
;
Lynne Horsburgh
b
;
Vladimí
;
r Kry&scaron
;
tof
c
;
Paul D. Lucas
b
;
Mariam Mojally
b
;
Simon J. Teat
d
;
Thomas G. Warwick
b
;
George W. Weaver
b
;
g.w.weaver@lboro.ac.uk" class="auth_mail" title="E-mail the corresponding author
;
Fatemeh Zeinali
b
关键词:
Anticancer activity
;
Benzimidazole
;
C-F activation
;
Fluorinated drug
scaffold
s
;
SNAr substitution
刊名:Journal of Fluorine Chemistry
出版年:2016
1
2
3
4
5
6
7
8
9
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