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在“Elsevier电子期刊”中，命中：184条，耗时：小于0.01 秒

在所有数据库中总计命中：281条

1.2,4-Disubstituted quinazolines as amyloid-β aggregation inhibitors with dual cholinesterase inhibition and antioxidant properties: Development and structure-activity relationship (SAR) studies

作者：Tarek Mohamed^a ; ^b ; Praveen P.N. Rao^a ; ^{praopera@uwaterloo.ca}

关键词：Alzheimer's disease ; Amyloid-beta ; Cholinesterase ; Quinazoline ; Molecular modeling

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.2-Guanidino-quinazolines as a novel class of translation inhibitors

作者：E.S. Komarova (Andreyanova)^a ; I.A. Osterman^b ; ^c ; ^d ; P.I. Pletnev^b ; ^c ; ^d ; Y.A. Ivanenkov^d ; ^e ; ^f ; A.G. Majouga^d ; ^f ; A.A. Bogdanov^b ; ^d ; P.V. Sergiev^b ; ^c ; ^d ; ^{petya@genebee.msu.ru}

关键词：Protein synthesis ; Bacteria ; Antibacterial ; Translation ; Reporter strain ; Screening ; Quinazoline

刊名：Biochimie

出版年：2017

3.Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity

作者：Murat Bozdag^a ; ^e ; Ahmed Mahmoud Alafeefy^b ; ^e ; Abdul Malik Altamimi^c ; Daniela Vullo^a ; Fabrizio Carta^d ; ^{fabrizio.carta@unifi.it} ; Claudiu T. Supuran^d ; ^{claudiu.supuran@unifi.it}

关键词：Carbonic anhydrase inhibitors (CAIs) ; Quinazolines ; Coumarins ; 2H-Benzo[e][12 ; 4]thiadiazine 1 ; 1-dioxides ; Hypoxic tumors

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

4.Quinazoline derivatives as cathepsins B, H and L inhibitors and cell proliferating agents

作者：Neera Raghav^a ; ^{nraghav.chem@gmail.com} ; Suman Jangra^a ; Ajay Kumar^b ; Shalmoli Bhattacharyya^b

关键词：Cathepsin B ; Cathepsin H ; Cathepsin L ; Kinetics studies ; Microwave assisted synthesis

刊名：International Journal of Biological Macromolecules

出版年：2017

5.Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold

作者：Justine Desroches^a ; ¹ ; Charline Kieffer^a ; ¹ ; Nicolas Primas^a ; Sé ; bastien Hutter^b ; Armand Gellis^a ; Hussein El-Kashef^c ; Pascal Rathelot^a ; Pierre Verhaeghe^d ; ^{pierre.verhaeghe@univ-tlse3.fr} ; Nadine Azas^b ; Patrice Vanelle^a ; ^{patrice.vanelle@univ-amu.fr}

关键词：Quinazoline ; Quinoline ; Quinoxaline ; Thienopyrimidine ; Trichloromethyl goup ; Plasmodium falciparum ; In vitro antiplasmodial activity ; In vitro HepG2 cytotoxicity ; Structure-activity relationships

刊名：European Journal of Medicinal Chemistry

出版年：2017

6.Synthesis, photophysical properties and DFT study of novel polycarbo-substituted quinazolines derived from the 2-aryl-6-bromo-4-chloro-8-iodoquinazolines

作者：Hugues K. Paumo^a ; Malose J. Mphahlele^a ; ^{mphahmj@unisa.ac.za" class="auth_mail" title="E-mail the corresponding author} ; Lydia Rhyman^b ; Ponnadurai Ramasami^b

关键词：2-Aryl-6-bromo-4-chloro-8-iodoquinazolines ; Cross-coupling reactions ; Polycarbo-substituted quinazolines ; Photophysical properties ; DFT

刊名：Tetrahedron

出版年：2016

7.Synthesis and biological evaluation of novel tricyclic oxazine and oxazepine fused quinazolines. Part 2: Gefitinib analogs

作者：Min Sun ; ^{sunmin@ask-pharm.com" class="auth_mail" title="E-mail the corresponding author} ; Jun Zhao ; Xiangfeng Chen ; Zaiwei Zong ; Jiyong Han ; Youguo Du ; Huanliang Sun ; Feidong Wang

关键词：Tricyclic fused quinazolines ; Antitumor activity ; EGFR ; HER2

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

8.Synthesis, biological evaluation and molecular docking studies of 2-piperazin-1-yl-quinazolines as platelet aggregation inhibitors and ligands of integrin α_IIbβ₃

作者：Andrei A. Krysko^a ; ^{peptides@physchem.od.ua" class="auth_mail" title="E-mail the corresponding author} ; Alexander Yu. Kornylov^a ; Pavel G. Polishchuk^b ; Georgiy V. Samoylenko^a ; Olga L. Krysko^a ; Tatyana A. Kabanova^a ; Victor Ch. Kravtsov^c ; Vladimir M. Kabanov^a ; Barbara Wicher^d ; Sergei A. Andronati^a

关键词：Fibrinogen receptor antagonists ; αIIbβ3 ; 2-Piperazin-1-yl-quinazoline ; Platelet aggregation

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

9.Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum

作者：Armand Gellis^a ; Nicolas Primas^a ; Sé ; bastien Hutter^b ; Gilles Lanzada^a ; Vincent Remusat^a ; Pierre Verhaeghe^c ; ^{pierre.verhaeghe@univ-tlse3.fr" class="auth_mail" title="E-mail the corresponding author} ; Patrice Vanelle^a ; ^{patrice.vanelle@univ-amu.fr" class="auth_mail" title="E-mail the corresponding author} ; Nadine Azas^b

关键词：2-trichloromethylquinazoline ; 4-benzyloxyquinazoline ; 4-phenoxyquinazoline ; DMAP-catalysis ; SNAr reaction ; Microwave-assisted chemistry ; Plasmodium falciparum ; Antiplasmodial activity ; HepG2 cytotoxicity ; SARs

刊名：European Journal of Medicinal Chemistry

出版年：2016

10.Cyclometallated PT^II complexes of 2-(2-thienyl)-4-(cycloalkylimino)-substituted quinazolines

作者：Emiliya V. Nosova^a ; ^b ; ^{emily74@rambler.ru" class="auth_mail" title="E-mail the corresponding author} ; Tatyana N. Moshkina^a ; Dmitry S. Kopchuk^a ; ^b ; Galina N. Lipunova^b ; Pavel A. Slepukhin^a ; ^b ; Valery N. Charushin^a ; ^b

刊名：Mendeleev Communications

出版年：2016

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