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CNKI学位论文(1)
在“
Elsevier电子期刊
”中,
命中:
18
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Evaluation of dipeptide nitriles as inhibitors of rhodesain, a major cysteine protease of Trypanosoma brucei
作者:
Tanja
Schirmeister
a
;
schirmei@uni-mainz.de
;
Janina Schmitz
b
;
Sascha Jung
a
;
Torsten Schmenger
c
;
R. Luise Krauth-Siegel
c
;
Michael Gü
;
tschow
b
关键词:
Dipeptide nitrile
;
Cysteine protease
;
Rhodesain
;
Inhibitor
;
Trypanosoma
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
2.
Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents
作者:
Roberta Ettari
a
;
Santo Previti
a
;
Sandro Cosconati
b
;
Santina Maiorana
a
;
Tanja
Schirmeister
c
;
Silvana Grasso
a
;
Maria Zappalà
;
a
;
mzappala@unime.it" class="auth_mail" title="E-mail the corresponding author
关键词:
Trypanosoma
;
Peptidomimetics
;
Michael acceptors
;
Microwave irradiation
;
Pharmacokinetic parameters
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
3.
Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening
作者:
Carmen Di Giovanni
a
;
Roberta Ettari
b
;
Serena Sarno
a
;
Archimede Rotondo
c
;
Alessandra Bitto
d
;
Francesco Squadrito
d
;
Domenica Altavilla
c
;
Tanja
Schirmeister
e
;
Ettore Novellino
a
;
Silvana Grasso
b
;
Maria Zappalà
;
b
;
Antonio Lavecchia
a
;
antonio.lavecchia@unina.it" class="auth_mail" title="E-mail the corresponding author
关键词:
Proteasome inhibitors
;
Non-covalent
;
Peptide scaffold
;
Docking studies
;
Virtual screening
刊名:European Journal of Medicinal Chemistry
出版年:2016
4.
Bistacrine derivatives as new potent antimalarials
作者:
Ines Schmidt
a
;
Gabriele Pradel
b
;
Ludmilla Sologub
b
;
Alexandra Golzmann
b
;
Che J. Ngwa
b
;
Anna Kucharski
a
;
Tanja
Schirmeister
c
;
Ulrike Holzgrabe
a
;
ulrike.holzgrabe@uni-wuerzburg.de" class="auth_mail" title="E-mail the corresponding author
关键词:
Bistacrines
;
Antimalarials
;
Falcipain-2 inhibitors
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
5.
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
作者:
Roberta Ettari
a
;
rettari@unime.it" class="auth_mail" title="E-mail the corresponding author
;
Andrea Pinto
b
;
Santo Previti
a
;
Lucia Tamborini
b
;
Ilenia C. Angelo
a
;
Valeria La Pietra
c
;
Luciana Marinelli
c
;
Ettore Novellino
c
;
Tanja
Schirmeister
d
;
Maria Zappalà
;
a
;
Silvana Grasso
e
;
Carlo De Micheli
b
;
Paola Conti
b
关键词:
Rhodesain
;
Dipeptide-like
;
3-Bromo isoxazoline
;
Inhibitor
;
Molecular modeling
刊名:Bioorganic & Medicinal Chemistry
出版年:2015
6.
Identification of a new series of amides as non-covalent proteasome inhibitors
作者:
Kety Scarbaci
a
;
Valeria Troiano
a
;
Nicola Micale
a
;
Roberta Ettari
b
;
roberta.ettari@unimi.it" class="auth_mail
;
Lucia Tamborini
b
;
Carmen Di Giovanni
c
;
Carmen Cerchia
c
;
Silvana Grasso
a
;
Ettore Novellino
c
;
Tanja
Schirmeister
d
;
Antonio Lavecchia
c
;
Maria Zappalà
;
a
关键词:
Amides
;
Proteasome inhibitors
;
Non-covalent inhibitors
;
Docking studies
刊名:European Journal of Medicinal Chemistry
出版年:9 April, 2014
7.
Development of peptidomimetic boronates as proteasome inhibitors
作者:
Nicola Micale
a
;
nmicale@unime.it
;
Roberta Ettari
b
;
Antonio Lavecchia
c
;
Carmen Di Giovanni
c
;
Kety Scarbaci
a
;
Valeria Troiano
a
;
Silvana Grasso
a
;
Ettore Novellino
c
;
Tanja
Schirmeister
d
;
Maria Zappalà
;
a
关键词:
Peptidomimetic boronates
;
Proteasome inhibitors
;
Docking studies
刊名:European Journal of Medicinal Chemistry
出版年:2013
8.
Selected gold compounds cause pronounced inhibition of Falcipain 2 and effectively block P. falciparum growth in vitro
作者:
Nicola
;
Micale
a
;
;
nmicale@unime.it
;
Maria Agostina
;
Cinellu
b
;
Laura
;
Maiore
b
;
Anna Rosa
;
Sannella
c
;
Carlo
;
Severini
c
;
Tanja
;
Schirmeister
d
;
Chiara
;
Gabbiani
e
;
Luigi
;
Messori
e
;
;
luigi.messori@unifi.it
关键词:
Gold compounds
;
Metallodrugs
;
Malaria
;
Falcipain 2
刊名:Journal of Inorganic Biochemistry
出版年:2011
9.
Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors
作者:
Roberta Ettari
;
Maria Zappalà
;
Nicola Micale
;
Giovanni Grazioso
;
Salvatore Giofrè
;
Tanja
Schirmeister
;
Silvana Grasso
关键词:
Peptidomimetics
;
Falcipain-2 inhibitors
;
Cysteine proteases
;
Docking studies
刊名:European Journal of Medicinal Chemistry
出版年:2011
10.
Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain
作者:
Roberta Ettari
;
Maria Zappalà
;
Nicola Micale
;
Tanja
Schirmeister
;
Christoph Gelhaus
;
Matthias Leippe
;
Astrid Evers
;
Silvana Grasso
关键词:
Peptidomimetics
;
Falcipain-2 inhibitors
;
Rhodesain inhibitors
;
Cysteine proteases
刊名:European Journal of Medicinal Chemistry
出版年:2010
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