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CNKI期刊论文0611(1)
知网期刊论文(37)
在“
Elsevier电子期刊
”中,
命中:
26
条,耗时:小于0.01 秒
在所有数据库中总计命中:
84
条
1.
Structure-activity relationship study and discovery of
indazole
3
-
carboxamide
s as calcium-release activated calcium channel blockers
作者:
Sha Bai
a
;
Masazumi Nagai
a
;
Steffi K. Koerner
a
;
Aristidis Veves
b
;
Lijun Sun
a
;
lsun1@bidmc.harvard.edu
关键词:
Mast cell
;
Inflammation
;
Calcium channel blockers
;
Indazole
-
3
-
carboxamide
s
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
2.
Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted
indazole
-5-
carboxamide
s as subnanomolar, selective monoamine oxidase B and dual MAO-A/B inhibitors
作者:
Nikolay T. Tzvetkov
a
;
ntzvetkov@ntzlab.com
;
Hans-Georg Stammler
b
;
Beate Neumann
b
;
Silvia Hristova
c
;
Liudmil Antonov
c
;
Marcus Gastreich
d
关键词:
ADME
;
MAO inhibitors
;
Molecular modeling
;
Indazole
-5-
carboxamide
s
;
Parkinson's disease
;
X-ray
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Enantioseparation of the
carboxamide
-type synthetic cannabinoids N-(1-amino-
3
-methyl-1-oxobutan-2-yl)-1-(5-fluoropentyl)-1H-
indazole
-
3
-
carboxamide
and methyl [1-(5-fluoropentyl)-1H-
indazole
-
3
-carbonyl]-valinate in illicit herbal products
作者:
Takahiro Doi
a
;
tdoi@iph.pref.osaka.jp" class="auth_mail" title="E-mail the corresponding author
;
Akiko Asada
a
;
Akihiro Takeda
a
;
Takaomi Tagami
a
;
Munehiro Katagi
b
;
Hiroe Kamata
b
;
Yoshiyuki Sawabe
a
关键词:
Carboxamide
-type synthetic cannabinoids
;
Enantiomer separation
;
5F-AB-PINACA
;
5F-AMB
刊名:Journal of Chromatography A
出版年:2016
4.
Linear propargylic alcohol functionality attached to the
indazole
-7-
carboxamide
as a JAK1-specific linear probe group
作者:
Mi Kyoung Kim
;
Heerim Shin
;
Seo Young Cho
;
Youhoon Chong
关键词:
Janus kinase (JAK)
;
Isozyme-specificity
;
Propargylic alcohol
;
Probe group
刊名:Bioorganic and Medicinal Chemistry
出版年:1 February, 2014
5.
Synthesis of substituted
3
-amino-N-phenyl-1H-
indazole
-1-
carboxamide
s endowed with antiproliferative activity
作者:
Benedetta Maggio
;
Maria Valeria Raimondi
;
Demetrio Raffa
;
Fabiana Plescia
;
Stella Cascioferro
;
Salvatore Plescia
;
Manlio Tolomeo
;
Antonietta Di Cristina
;
Rosaria Maria Pipitone
;
Stefania Grimaudo
;
Giuseppe Daidone
关键词:
3
-amino-N-phenyl-1H-
indazole
-1-
carboxamide
s
;
G0ȁ
3
;
G1 arrest
;
pRb
;
Antiproliferative agents
刊名:European Journal of Medicinal Chemistry
出版年:2011
6.
Synthesis and biological evaluation of substituted 2-phenyl-2H-
indazole
-7-
carboxamide
s as potent poly(ADP-ribose) polymerase (PARP) inhibitors
作者:
Rita Scarpelli
;
Julia K. Boueres
;
Mauro Cerretani
;
Federica Ferrigno
;
Jesus M. Ontoria
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Carlo Toniatti
;
Philip Jones
关键词:
Poly(ADP-ribose) polymerase
;
PARP inhibitor
;
2-Phenyl-2
H
-
indazole
-7-
carboxamide
s
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
7.
Fragment-based discovery of hydroxy-
indazole
-
carboxamide
s as novel small molecule inhibitors of Hsp90
作者:
Hans-Peter Buchstaller
;
hans-peter.buchstaller@merckgroup.com
;
Hans-Michael Eggenweiler
;
Christian Sirrenberg
;
Ulrich Grä
;
dler
;
Djordje Musil
;
Edmund Hoppe
;
Astrid Zimmermann
;
Harry Schwartz
;
Joachim Mä
;
rz
;
Jö
;
rg Bomke
;
Ansgar Wegener
;
Michael Wolf
关键词:
Hsp90
;
Heat shock protein 90
;
Anti-cancer drug
;
Fragments
;
Indazole
s
;
Docking
;
X-ray structure
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
8.
Synthesis and antiproliferative activity of
3
-amino-N-phenyl-1H-
indazole
-1-
carboxamide
s
作者:
Demetrio Raffa
;
Benedetta Maggio
;
Stella Cascioferro
;
Maria Valeria Raimondi
;
Domenico Schillaci
;
Giorgio Gallo
;
Giuseppe Daidone
;
Salvatore Plescia
;
Fiorella Meneghetti
;
Gabriella Bombieri
;
Antonietta Di Cristina
;
Rosaria M. Pipitone
;
Stefania Grimaudo
;
Manlio Tolomeo
关键词:
1
H
-
Indazole
-1-
carboxamide
s
;
Crystallographic study
;
G0ȁ
3
;
G1 arrest
;
pRb
刊名:European Journal of Medicinal Chemistry
出版年:2009
9.
The design and synthesis of
indazole
and pyrazolopyridine based glucokinase activators for the treatment of Type 2 diabetes mellitus
作者:
Jeffrey A. Pfefferkorn
a
;
jeffrey.a.pfefferkorn@pfizer.com
;
Meihua Tu
a
;
Kevin J. Filipski
a
;
Angel Guzman-Perez
b
;
Jianwei Bian
b
;
Gary E. Aspnes
b
;
Matthew F. Sammons
a
;
Wei Song
b
;
Jian-Cheng Li
b
;
Christopher S. Jones
b
;
Leena Patel
b
;
Tim Rasmusson
b
;
Dongxiang Zeng
b
;
Kapil Karki
b
;
Michael Hamilton
b
;
Richard Hank
b
;
Karen Atkinson
b
;
John Litchfield
b
;
Robert Aiello
b
;
Levenia Baker
b
;
Nicole Barucci
b
;
Patricia Bourassa
b
;
Francis Bourbounais
b
;
Theresa D’
;
Aquila
b
;
David R. Derksen
b
;
Margit MacDougall
b
;
Alan Robertson
b
关键词:
Glucokinase activator
;
Type 2 diabetes mellitus
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
10.
Inhibitory effects of a series of 7-substituted-
indazole
s toward nitric oxide synthases: Particular potency of 1H-
indazole
-7-carbonitrile
作者:
Betty Cottyn
;
Francine Acher
;
Booma Ramassamy
;
Luke Alvey
;
Michel Lepoivre
;
Yves Frapart
;
Dennis Stuehr
;
Daniel Mansuy
;
Jean-Luc Boucher
;
Dominique Vichard
关键词:
7-Nitro
indazole
;
Substituted
indazole
s
;
Nitric oxide synthase
;
Inhibitors
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
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