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ACS电子期刊(30)
在“
ACS电子期刊
”中,
命中:
30
条,耗时:小于0.01 秒
在所有数据库中总计命中:
137
条
1.
Design and Synthesis of a Series of l-trans-4-Substituted Prolines as Selective Antagonists for the Ionotropic Glutamate Receptors Including Functional and X-ray Crystallographic Studies of New Subtype Selective Kainic Acid Receptor Subtype 1 (GluK1) Antagonist (2S,4R)-4-(2-Carboxyphenoxy)pyrrolidin
作者:
Niels Krogsgaard-Larsen
;
Claudia G. Delgar
;
Karina Koch
;
Patricia M. G. E. Brown
;
Charlotte Møller
;
Liwei Han
;
Tri H. V. Huynh
;
Stinne W. Hansen
;
Birgitte
Nielsen
;
Derek Bowie
;
Darryl S. Pickering
;
Jette Sandholm Kastrup
;
Karla Frydenvang
;
Lennart Bunch
刊名:Journal of Medicinal Chemistry
出版年:2017
2.
Tweaking Subtype Selectivity and Agonist Efficacy at (S)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) Receptors in a Small Series of BnTetAMPA Analogues
作者:
Shuang-Yan Wang
;
Younes Larsen
;
Cristina Vara Navarrete
;
Anders A. Jensen
;
Birgitte
Nielsen
;
Ali Al-Musaed
;
Karla Frydenvang
;
Jette Sandholm Kastrup
;
Darryl S. Pickering
;
Rasmus Prætorius Clausen
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
New 4-Functionalized Glutamate Analogues Are Selective Agonists at Metabotropic Glutamate Receptor Subtype 2 or Selective Agonists at Metabotropic Glutamate Receptor Group III
作者:
Tri H. V. Huynh
;
Mette N. Erichsen
;
Amélie S. Tora
;
Cyril Goudet
;
Emmanuelle Sagot
;
Zeinab Assaf
;
Christian Thomsen
;
Robb Brodbeck
;
Tine B. Stensb?l
;
Walden E. Bj?rn-Yoshimoto
;
Birgitte
Nielsen
;
Jean-Philippe Pin
;
Thierry Gefflaut
;
Lennart Bunch
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors
作者:
Ewa Szymanska
;
Karla Frydenvang
;
Darryl S. Pickering
;
Christian Krintel
;
Birgitte
Nielsen
;
Ayesheh Kooshki
;
Linda G. Zachariassen
;
Lars Olsen
;
Jette S. Kastrup
;
Tommy N. Johansen
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
β-Sulfonamido Functionalized Aspartate Analogues as Excitatory Amino Acid Transporter Inhibitors: Distinct Subtype Selectivity Profiles Arising from Subtle Structural Differences
作者:
Jacob C. Hansen
;
Walden E. Bjørn-Yoshimoto
;
Niels Bisballe
;
Birgitte
Nielsen
;
Anders A. Jensen
;
Lennart Bunch
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Binding Mode of an 伪-Amino Acid-Linked Quinoxaline-2,3-dione Analogue at Glutamate Receptor Subtype GluK1
作者:
Charles S. Demmer
;
Charlotte M酶ller
;
Patricia M. G. E. Brown
;
Liwei Han
;
Darryl S. Pickering
;
Birgitte
Nielsen
;
Derek Bowie
;
Karla Frydenvang
;
Jette S. Kastrup
;
Lennart Bunch
刊名:ACS Chemical Neuroscience
出版年:2015
7.
Structure鈥揂ctivity Relationship Study of Ionotropic Glutamate Receptor Antagonist (2S,3R)-3-(3-Carboxyphenyl)pyrrolidine-2-carboxylic Acid
作者:
Niels Krogsgaard-Larsen
;
Morten Storgaard
;
Charlotte M酶ller
;
Charles S. Demmer
;
Jeanette Hansen
;
Liwei Han
;
Rune N. Monrad
;
Birgitte
Nielsen
;
Daniel Tapken
;
Darryl S. Pickering
;
Jette S. Kastrup
;
Karla Frydenvang
;
Lennart Bunch
刊名:Journal of Medicinal Chemistry
出版年:2015
8.
Development of 2鈥?Substituted (2S,1鈥?i>R,2鈥?i>S)-2-(Carboxycyclopropyl)glycine Analogues as Potent N-Methyl-d-aspartic Acid Receptor Agonists
作者:
Rune Risgaard
;
Simon D.
Nielsen
;
Kasper B. Hansen
;
Christina M. Jensen
;
Birgitte
Nielsen
;
Stephen F. Traynelis
;
Rasmus P. Clausen
刊名:Journal of Medicinal Chemistry
出版年:2013
9.
Chemoenzymatic Synthesis of New 2,4-syn-Functionalized (S)-Glutamate Analogues and Structure鈥揂ctivity Relationship Studies at Ionotropic Glutamate Receptors and Excitatory Amino Acid Tra
作者:
Zeinab Assaf
;
Anja P. Larsen
;
Raminta Venskutonyt臈
;
Liwei Han
;
Bjarke Abrahamsen
;
Birgitte
Nielsen
;
Michael Gajhede
;
Jette S. Kastrup
;
Anders A. Jensen
;
Darryl S. Pickering
;
Karla Frydenvang
;
Thierry Gefflaut
;
Lennart Bunch
刊名:Journal of Medicinal Chemistry
出版年:2013
10.
Exploring the Orthosteric Binding Site of the 纬-Aminobutyric Acid Type A Receptor Using 4-(Piperidin-4-yl)-1-hydroxypyrazoles 3- or 5-Imidazolyl Substituted: Design, Synthesis, and Pharmacological Eva
作者:
Jacob Krall
;
Claus H. Jensen
;
Troels E. S酶rensen
;
Birgitte
Nielsen
;
Anders A. Jensen
;
Tommy Sander
;
Thomas Balle
;
Bente Fr酶lund
刊名:Journal of Medicinal Chemistry
出版年:2013
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