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Wiley电子期刊(2)
Elsevier电子期刊(22)
ACS电子期刊(16)
在“
ACS电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
40
条
1.
Rapid and Reliable Binding Affinity Prediction of Bromodomain Inhibitors: A Computational Study
作者:
Shunzhou Wan
;
Agastya P. Bhati
;
Stefan J. Zasada
;
Ian Wall
;
Darren Green
;
Paul
Bamborough
;
Peter V. Coveney
刊名:Journal of Chemical Theory and Computation
出版年:2017
2.
GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain
作者:
Paul
Bamborough
;
Heather A. Barnett
;
Isabelle Becher
;
Mark J. Bird
;
Chun-wa Chung
;
Peter D. Craggs
;
Emmanuel H. Demont
;
Hawa Diallo
;
David J. Fallon
;
Laurie J. Gordon
;
Paola Grandi
;
Clare I. Hobbs
;
Edward Hooper-Greenhill
;
Emma J. Jones
;
Robert P. Law
;
Armelle Le Gall
;
David Lugo
;
Anne-Marie Michon
;
Darren J. Mitchell
;
Rab K. Prinjha
;
Robert J. Sheppard
;
Allan J. B. Watson
;
Robert J. Watson
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B
作者:
Peiling Chen
;
Apirat Chaikuad
;
Paul
Bamborough
;
Marcus Bantscheff
;
Chas Bountra
;
Chun-wa Chung
;
Oleg Fedorov
;
Paola Grandi
;
David Jung
;
Robert Lesniak
;
Matthew Lindon
;
Susanne Müller
;
Martin Philpott
;
Rab Prinjha
;
Catherine Rogers
;
Carolyn Selenski
;
Cynthia Tallant
;
Thilo Werner
;
Timothy M. Willson
;
Stefan Knapp
;
David H. Drewry
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition
作者:
Natalie H. Theodoulou
;
Paul
Bamborough
;
Andrew J. Bannister
;
Isabelle Becher
;
Rino A. Bit
;
Ka Hing Che
;
Chun-wa Chung
;
Antje Dittmann
;
Gerard Drewes
;
David H. Drewry
;
Laurie Gordon
;
Paola Grandi
;
Melanie Leveridge
;
Matthew Lindon
;
Anne-Marie Michon
;
Judit Molnar
;
Samuel C. Robson
;
Nicholas C. O. Tomkinson
;
Tony Kouzarides
;
Rab K. Prinjha
;
Philip G. Humphreys
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Fragment-Based Discovery of Low-Micromolar ATAD2 Bromodomain Inhibitors
作者:
Emmanuel H. Demont
;
Chun-wa Chung
;
Rebecca C. Furze
;
Paola Grandi
;
Anne-Marie Michon
;
Chris Wellaway
;
Nathalie Barrett
;
Angela M. Bridges
;
Peter D. Craggs
;
Hawa Diallo
;
David P. Dixon
;
Clement Douault
;
Amanda J. Emmons
;
Emma J. Jones
;
Bhumika V. Karamshi
;
Kelly Locke
;
Darren J. Mitchell
;
Bernadette H. Mouzon
;
Rab K. Prinjha
;
Andy D. Roberts
;
Robert J. Sheppard
;
Robert J. Watson
;
Paul
Bamborough
刊名:Journal of Medicinal Chemistry
出版年:2015
6.
Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors
作者:
Paul
Bamborough
;
Chun-wa Chung
;
Rebecca C. Furze
;
Paola Grandi
;
Anne-Marie Michon
;
Robert J. Sheppard
;
Heather Barnett
;
Hawa Diallo
;
David P. Dixon
;
Clement Douault
;
Emma J. Jones
;
Bhumika Karamshi
;
Darren J. Mitchell
;
Rab K. Prinjha
;
Christina Rau
;
Robert J. Watson
;
Thilo Werner
;
Emmanuel H. Demont
刊名:Journal of Medicinal Chemistry
出版年:2015
7.
1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain
作者:
Emmanuel H. Demont
;
Paul
Bamborough
;
Chun-wa Chung
;
Peter D. Craggs
;
David Fallon
;
Laurie J. Gordon
;
Paola Grandi
;
Clare I. Hobbs
;
Jameed Hussain
;
Emma J. Jones
;
Armelle Le Gall
;
Anne-Marie Michon
;
Darren J. Mitchell
;
Rab K. Prinjha
;
Andy D. Roberts
;
Robert J. Sheppard
;
Robert J. Watson
刊名:ACS Medicinal Chemistry Letters
出版年:2014
8.
The Discovery of I-BET726 (GSK1324726A), a Potent Tetrahydroquinoline ApoA1 Up-Regulator and Selective BET Bromodomain Inhibitor
作者:
Romain Gosmini
;
Van Loc Nguyen
;
J茅r么me Toum
;
Christophe Simon
;
Jean-Marie G. Brusq
;
Gael Krysa
;
Olivier Mirguet
;
Alizon M. Riou-Eymard
;
Eric V. Boursier
;
Lionel Trottet
;
Paul
Bamborough
;
Hugh Clark
;
Chun-wa Chung
;
Leanne Cutler
;
Emmanuel H. Demont
;
Rejbinder Kaur
;
Antonia J. Lewis
;
Mark B. Schilling
;
Peter E. Soden
;
Simon Taylor
;
Ann L. Walker
;
Matthew D. Walker
;
Rab K. Prinjha
;
Edwige Nicod猫me
刊名:Journal of Medicinal Chemistry
出版年:2014
9.
Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains
作者:
Olivier Mirguet
;
Romain Gosmini
;
J茅r么me Toum
;
Catherine A. Cl茅ment
;
M茅lanie Barnathan
;
Jean-Marie Brusq
;
Jacqueline E. Mordaunt
;
Richard M. Grimes
;
Miriam Crowe
;
Olivier Pineau
;
Myriam Ajakane
;
Alain Daugan
;
Phillip Jeffrey
;
Leanne Cutler
;
Andrea C. Haynes
;
Nicholas N. Smithers
;
Chun-wa Chung
;
Paul
Bamborough
;
Iain J. Uings
;
Antonia Lewis
;
Jason Witherington
;
Nigel Parr
;
Rab K. Prinjha
;
Edwige Nicod猫me
刊名:Journal of Medicinal Chemistry
出版年:2013
10.
Fragment-Based Discovery of Bromodomain Inhibitors Part 2: Optimization of Phenylisoxazole Sulfonamides
作者:
Paul
Bamborough
;
Hawa Diallo
;
Jonathan D. Goodacre
;
Laurie Gordon
;
Antonia Lewis
;
Jonathan T. Seal
;
David M. Wilson
;
Michael D. Woodrow
;
Chun-wa Chung
刊名:Journal of Medicinal Chemistry
出版年:2012
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