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Wiley电子期刊(1)
NATURE电子期刊(2)
ACS电子期刊(18)
SpringerLink电子期刊(3)
Elsevier电子期刊(64)
在“
ACS电子期刊
”中,
命中:
18
条,耗时:0.0199918 秒
在所有数据库中总计命中:
88
条
1.
High-Throughput Screening and Hit Validation of Extracellular-Related Kinase 5 (ERK5) Inhibitors
作者:
Stephanie M. Myers
;
Ruth H. Bawn
;
Louise C. Bisset
;
Timothy
J
. Blackburn
;
Betty Cottyn
;
Lauren Molyneux
;
Ai-Ching Wong
;
Celine Cano
;
William Clegg
;
Ross. W. Harrington
;
Hing Leung
;
Laurent Rigoreau
;
Sandrine Vidot
;
Bernard T. Golding
;
Roger
J
.
Griffin
;
Tim Hammonds
;
David R. Newell
;
Ian R. Hardcastle
刊名:ACS Combinatorial Science
出版年:2016
2.
8-Substituted O6-Cyclohexylmethylguanine CDK2 Inhibitors: Using Structure-Based Inhibitor Design to Optimize an Alternative Binding Mode
作者:
Benoit Carbain
;
David
J
. Paterson
;
Elizabeth Anscombe
;
Allyson
J
. Campbell
;
Celine Cano
;
Aude Echalier
;
J
ane A. Endicott
;
Bernard T. Golding
;
Karen Haggerty
;
Ian R. Hardcastle
;
Philip
J
. Jewsbury
;
David R. Newell
;
Martin E. M. Noble
;
Celine Roche
;
Lan Z. Wang
;
Roger
J
.
Griffin
刊名:
J
ournal of Medicinal Chemistry
出版年:2014
3.
1-Substituted (Dibenzo[b,d]thiophen-4-yl)-2-morpholino-4H-chromen-4-ones Endowed with Dual DNA-PK/PI3-K Inhibitory Activity
作者:
C茅line Cano
;
Kappusamy Saravanan
;
Chris Bailey
;
J
ulia Bardos
;
Nicola
J
. Curtin
;
Mark Frigerio
;
Bernard T. Golding
;
Ian R. Hardcastle
;
Marc G. Hummersone
;
Keith A. Menear
;
David R. Newell
;
Caroline
J
. Richardson
;
K. Shea
;
Graeme C. M. Smith
;
Pia Thommes
;
Attilla Ting
;
Roger
J
.
Griffin
刊名:
J
ournal of Medicinal Chemistry
出版年:2013
4.
Nucleoside Transport Inhibitors: Structure鈭扐ctivity Relationships for Pyrimido[5,4-d]pyrimidine Derivatives That Potentiate Pemetrexed Cytotoxicity in the Presence of 伪1-Acid Glycopr
作者:
Kappusamy Saravanan
;
Hannah C. Barlow
;
Marion Barton
;
A. Hilary Calvert
;
Bernard T. Golding
;
David R. Newell
;
J
ulian S. Northen
;
Nicola
J
. Curtin
;
Huw D. Thomas
;
Roger
J
.
Griffin
刊名:
J
ournal of Medicinal Chemistry
出版年:2011
5.
Isoindolinone Inhibitors of the Murine Double Minute 2 (MDM2)-p53 Protein鈭扨rotein Interaction: Structure鈭扐ctivity Studies Leading to Improved Potency
作者:
Ian R. Hardcastle
;
J
unfeng Liu
;
Eric Valeur
;
Anna Watson
;
Shafiq U. Ahmed
;
Timothy
J
. Blackburn
;
Karim Bennaceur
;
William Clegg
;
Catherine Drummond
;
J
ane A. Endicott
;
Bernard T. Golding
;
Roger
J
.
Griffin
;
J
an Gruber
;
Karen Haggerty
;
Ross W. Harrington
;
Claire Hutton
;
Stuart Kemp
;
Xiaohong Lu
;
J
ames M. McDonnell
;
David R. Newell
;
Martin E. M. Noble
;
Sara L. Payne
;
Charlotte H. Revill
;
Christiane Riedinger
;
Qing Xu
;
J
ohn Lunec
刊名:
J
ournal of Medicinal Chemistry
出版年:2011
6.
Antagonists of the Human A2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-d]pyrimidines
作者:
Roger
J
. Gillespie
;
Samantha
J
. Bamford
;
Ruth Botting
;
Mike Comer
;
Sarah Denny
;
Suneel Gaur
;
Michael
Griffin
;
Allan M.
J
ordan
;
Anthony R. Knight
;
J
oanne Lerpiniere
;
Stefania Leonardi
;
Sean Lightowler
刊名:
J
ournal of Medicinal Chemistry
出版年:2009
7.
Analysis of Chemical Shift Changes Reveals the Binding Modes of Isoindolinone Inhibitors of the MDM2-p53 Interaction
作者:
Christiane Riedinger
;
J
ane A. Endicott
;
Stuart
J
. Kemp
;
Lynette A. Smyth
;
Anna Watson
;
Eric Valeur
;
Bernard T. Golding
;
Roger
J
.
Griffin
;
Ian R. Hardcastle
;
Martin E. Noble
;
J
ames M. McDonnell
刊名:
J
ournal of the American Chemical Society
出版年:2008
8.
Interactions of 1-Methylimidazole with UO2(CH3CO2)2 and UO2(NO3)2: Structural, Spectroscopic, and Theoretical Evidence for
作者:
Keith E. Gutowski
;
Violina A. Cocalia
;
Scott T.
Griffin
;
Nicholas
J
. Bridges
;
David A. Dixon
;
Robin D.
Roger
s
刊名:
J
ournal of the American Chemical Society
出版年:2007
9.
J
udicious Application of Allyl Protecting Groups for the Synthesis of 2-Morpholin-4-yl-4-oxo-4H-chromen-8-yl Triflate, a Key Precursor of DNA-Dependent Protein Kinase Inhibitors
作者:
Sonsoles Rodriguez Aristegui
;
Marine Desage El-Murr
;
Bernard T. Golding
;
Roger
J
.
Griffin
;
Ian R. Hardcastle
刊名:Organic Letters
出版年:2006
10.
Small-Molecule Inhibitors of the MDM2-p53 Protein-Protein Interaction Based on an Isoindolinone Scaffold
作者:
Ian R. Hardcastle
;
Shafiq U. Ahmed
;
Helen Atkins
;
Gillian Farnie
;
Bernard T. Golding
;
Roger
J
.
Griffin
;
Sabrina Guyenne
;
Claire Hutton
;
Per Kä
;
llblad
;
Stuart
J
. Kemp
;
Martin S. Kitching
;
David R.
刊名:
J
ournal of Medicinal Chemistry
出版年:2006
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