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Elsevier电子期刊(3)
ACS电子期刊(9)
在“
ACS电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
12
条
1.
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
作者:
Essa Hu
;
Ning Chen
;
Roxanne
K.
Kunz
;
Dah-Ren Hwang
;
Klaus Michelsen
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Randall Hungate
;
James Treanor
;
Hang Chen
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 3. Structure鈥揂ctivity Relationships within the Aryl Carbinol Region of the N-Arylsulfonamido-N鈥?a
作者:
Nobuko Nishimura
;
Mark H. Norman
;
Longbin Liu
;
Kevin C. Yang
;
Kate S. Ashton
;
Michael D. Bartberger
;
Samer Chmait
;
Jie Chen
;
Rod Cupples
;
Christopher Fotsch
;
Joan Helmering
;
Steven R. Jordan
;
Roxanne
K.
Kunz
;
Lewis D. Pennington
;
Steve F. Poon
;
Aaron Siegmund
;
Glenn Sivits
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
3.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 2. Leveraging Structure-Based Drug Design to Identify Analogues with Improved Pharmacokinetic Profiles
作者:
David J. St. Jean
;
Jr.
;
Kate S. Ashton
;
Michael D. Bartberger
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Elizabeth Galbreath
;
Joan Helmering
;
Fang-Tsao Hong
;
Steven R. Jordan
;
Longbin Liu
;
Roxanne
K.
Kunz
;
Klaus Michelsen
;
Nobuko Nishimura
;
Lewis D. Pennington
;
Steve F. Poon
;
Darren Reid
;
Glenn Sivits
;
Markian M. Stec
;
Seifu Tadesse
;
Nuria Tamayo
;
Gwyneth Van
;
Kevin C. Yang
;
Jiandong Zhang
;
Mark H. Norman
;
Christopher Fotsch
;
David J. Lloyd
;
Clarence Hale
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phos
作者:
Essa Hu
;
Ning Chen
;
Matthew P. Bourbeau
;
Paul E. Harrington
;
Kaustav Biswas
;
Roxanne
K.
Kunz
;
Kristin L. Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Jean Danao
;
Jessica Able
;
Madelyn Cueva
;
Santosh Talreja
;
Thomas Kornecook
;
Hang Chen
;
Amy Porter
;
Randall Hungate
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
作者:
Essa Hu
;
Roxanne
K.
Kunz
;
Ning Chen
;
Shannon Rumfelt
;
Aaron Siegmund
;
Kristin Andrews
;
Samer Chmait
;
Sharon Zhao
;
Carl Davis
;
Hang Chen
;
Dianna Lester-Zeiner
;
Ji Ma
;
Christopher Biorn
;
Jianxia Shi
;
Amy Porter
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Rapid Identification of a Novel Small Molecule Phosphodiesterase 10A (PDE10A) Tracer
作者:
Essa Hu
;
Ji Ma
;
Christopher Biorn
;
Dianna Lester-Zeiner
;
Robert Cho
;
Shannon Rumfelt
;
Roxanne
K.
Kunz
;
Thomas Nixey
;
Klaus Michelsen
;
Silke Miller
;
Jianxia Shi
;
Jamie Wong
;
Geraldine Hill Della Puppa
;
Jessica Able
;
Santosh Talreja
;
Dah-Ren Hwang
;
Stephen A. Hitchcock
;
Amy Porter
;
David Immke
;
Jennifer R. Allen
;
James Treanor
;
Hang Chen
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
Discovery of Aryl Aminoquinazoline Pyridones as Potent, Selective, and Orally Efficacious Inhibitors of Receptor Tyrosine Kinase c-Kit
作者:
Essa Hu
;
Andrew Tasker
;
Ryan D. White
;
Roxanne
K.
Kunz
;
Jason Human
;
Ning Chen
;
Roland Bü
;
rli
;
Randall Hungate
;
Perry Novak
;
Andrea Itano
;
Xuxia Zhang
;
Violeta Yu
;
Yen Nguyen
;
Yanyan Tudor
;
Matthe
刊名:Journal of Medicinal Chemistry
出版年:2008
8.
Enantioselective Organocatalytic Cyclopropanations. The Identification of a New Class of Iminium Catalyst Based upon Directed Electrostatic Activation
作者:
Roxanne
K.
Kunz
and David W. C. MacMillan
刊名:Journal of the American Chemical Society
出版年:2005
9.
Chemoenzymatic Synthesis of 11-cis-Retinal Photoaffinity Analog by Use of Squid Retinochrome
作者:
Babak Borhan
;
Roxanne
Kunz
;
Andrew Y. Wang
;
Koji Nakanishi
;
Nina Bojkova
;
and Kazuo Yoshihara
刊名:Journal of the American Chemical Society
出版年:1997
1
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