设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
NATURE电子期刊(3)
Elsevier电子期刊(8)
ACS电子期刊(8)
在“
ACS电子期刊
”中,
命中:
8
条,耗时:小于0.01 秒
在所有数据库中总计命中:
19
条
1.
Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
作者:
Brian S. Gerstenberger
;
John D. Trzupek
;
Cynthia Tallant
;
Oleg Fedorov
;
Panagis Filippakopoulos
;
Paul E. Brennan
;
Vita Fedele
;
Sarah
Martin
;
Sarah
Picaud
;
Catherine Rogers
;
Mihir Parikh
;
Alexandria Taylor
;
Brian Samas
;
Alison O’Mahony
;
Ellen Berg
;
Gabriel Pallares
;
Adam D. Torrey
;
Daniel K. Treiber
;
Ivan J. Samardjiev
;
Brian T. Nasipak
;
Teresita Padilla-Benavides
;
Qiong Wu
;
Anthony N. Imbalzano
;
Jeffrey A. Nickerson
;
Mark E. Bunnage
;
Susanne Müller
;
Stefan Knapp
;
Dafydd R. Owen
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of New Bromodomain Scaffolds by Biosensor Fragment Screening
作者:
Iva Navratilova
;
Tonia Aristotelous
;
Sarah
Picaud
;
Apirat Chaikuad
;
Stefan Knapp
;
Panagis Filappakopoulos
;
Andrew L. Hopkins
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains
作者:
Duncan A. Hay
;
Oleg Fedorov
;
Sarah
Martin
;
Dean C. Singleton
;
Cynthia Tallant
;
Christopher Wells
;
Sarah
Picaud
;
Martin Philpott
;
Octovia P. Monteiro
;
Catherine M. Rogers
;
Stuart J. Conway
;
Timothy P. C. Rooney
;
Anthony Tumber
;
Clarence Yapp
;
Panagis Filippakopoulos
;
Mark E. Bunnage
;
Susanne M眉ller
;
Stefan Knapp
;
Christopher J. Schofield
;
Paul E. Brennan
刊名:Journal of the American Chemical Society
出版年:2014
4.
[1,2,4]Triazolo[4,3-a]phthalazines: Inhibitors of Diverse Bromodomains
作者:
Oleg Fedorov
;
Hannah Lingard
;
Chris Wells
;
Octovia P. Monteiro
;
Sarah
Picaud
;
Tracy Keates
;
Clarence Yapp
;
Martin Philpott
;
Sarah
J. Martin
;
Ildiko Felletar
;
Brian D. Marsden
;
Panagis Filippakopoulos
;
Susanne Müller
;
Stefan Knapp
;
Paul E. Brennan
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Optimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain Ligands
作者:
David S. Hewings
;
Oleg Fedorov
;
Panagis Filippakopoulos
;
Sarah
Martin
;
Sarah
Picaud
;
Anthony Tumber
;
Christopher Wells
;
Monica M. Olcina
;
Katherine Freeman
;
Andrew Gill
;
Alison J. Ritchie
;
David W. Sheppard
;
Angela J. Russell
;
Ester M. Hammond
;
Stefan Knapp
;
Paul E. Brennan
;
Stuart J. Conway
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Discovery of Novel Small-Molecule Inhibitors of BRD4 Using Structure-Based Virtual Screening
作者:
Lewis R. Vidler
;
Panagis Filippakopoulos
;
Oleg Fedorov
;
Sarah
Picaud
;
Sarah
Martin
;
Michael Tomsett
;
Hannah Woodward
;
Nathan Brown
;
Stefan Knapp
;
Swen Hoelder
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Identification of a Chemical Probe for Bromo and Extra C-Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit
作者:
Paul V. Fish
;
Panagis Filippakopoulos
;
Gerwyn Bish
;
Paul E. Brennan
;
Mark E. Bunnage
;
Andrew S. Cook
;
Oleg Federov
;
Brian S. Gerstenberger
;
Hannah Jones
;
Stefan Knapp
;
Brian Marsden
;
Karl Nocka
;
Dafydd R. Owen
;
Martin Philpott
;
Sarah
Picaud
;
Michael J. Primiano
;
Michael J. Ralph
;
Nunzio Sciammetta
;
John D. Trzupek
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
3,5-Dimethylisoxazoles Act As Acetyl-lysine-mimetic Bromodomain Ligands
作者:
David S. Hewings
;
Minghua Wang
;
Martin Philpott
;
Oleg Fedorov
;
Sagar Uttarkar
;
Panagis Filippakopoulos
;
Sarah
Picaud
;
Chaitanya Vuppusetty
;
Brian Marsden
;
Stefan Knapp
;
Stuart J. Conway
;
Tom D. Heightman
刊名:Journal of Medicinal Chemistry
出版年:2011
1
按检索点细分(8)
题名(8)
按出版年细分(8)
2016年(2)
2014年(2)
2013年(2)
2012年(1)
2011年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.