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Elsevier电子期刊(7)
ACS电子期刊(13)
在“
ACS电子期刊
”中,
命中:
13
条,耗时:0.0199913 秒
在所有数据库中总计命中:
20
条
1.
Regioselective Epoxide Ring Opening for the Stereospecific Scale-Up Synthesis of BMS-960, A Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
作者:
Xiaoping HouHuiping Zhang
;
Bang-Chi Chen
;
Zhiwei Guo
;
Amar
j
it Singh
;
Animesh Goswami
;
J
ohn L. Gilmore
;
J
ames E. Sheppeck
;
Alaric
J
.
Dyckman
;
Percy H. CarterArvind Mathur
刊名:Organic Process Research & Development
出版年:2017
2.
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials
作者:
T. G. Murali Dhar
;
Hai-Yun Xiao
;
J
enny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurng Wu
;
Marta Dabros
;
Xiaoxia Yang
;
Tracy L. Taylor
;
Xia D. Zhou
;
Elizabeth M. Heimrich
;
Rochelle Thomas
;
Kim W. McIntyre
;
Bethanne Warrack
;
Hong Shi
;
Paul C. Levesque
;
J
ia L. Zhu
;
J
ames Hennan
;
Praveen Balimane
;
Zheng Yang
;
Anthony M. Marino
;
Georgia Cornelius
;
Celia
J
. D’Arienzo
;
Arvind Mathur
;
Ding Ren Shen
;
Mary Ellen Cvi
j
ic
;
Luisa Salter-Cid
;
J
oel C. Barrish
;
Percy H. Carter
;
Alaric
J
.
Dyckman
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery and Structure–Activity Relationship (SAR) of a Series of Ethanolamine-Based Direct-Acting Agonists of Sphingosine-1-phosphate (S1P1)
作者:
J
ohn L. Gilmore
;
J
ames E. Sheppeck II
;
Scott H. Watterson
;
Lauren Haque
;
Parag Mukhopadhyay
;
Andrew
J
. Tebben
;
Michael A. Galella
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvi
j
ic
;
Virna Borowski
;
Kathleen Gillooly
;
Tracy Taylor
;
Kim W. McIntyre
;
Bethanne Warrack
;
Paul C. Levesque
;
J
ulia P. Li
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Luisa Salter-Cid
;
J
oel C. Barrish
;
William
J
. Pitts
;
Percy H. Carter
;
J
enny Xie
;
Alaric
J
.
Dyckman
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
4.
An Efficient Scale-Up Synthesis of BMS-520, a Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
作者:
Xiaoping Hou
;
J
uliang Zhu
;
Bang-Chi Chen
;
Scott H. Watterson
;
William
J
. Pitts
;
Alaric
J
.
Dyckman
;
Percy H. Carter
;
Arvind Mathur
;
Huiping Zhang
刊名:Organic Process Research & Development
出版年:2016
5.
Potent and Selective Agonists of Sphingosine 1-Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series
作者:
Scott H. Watterson
;
J
unqing Guo
;
Steve H. Spergel
;
Charles M. Langevine
;
Robert V. Moquin
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvi
j
ic
;
Dana Banas
;
Richard Liu
;
Suzanne
J
. Suchard
;
Kathleen Gillooly
;
Tracy Taylor
;
Sandra Rex-Rabe
;
David
J
. Shuster
;
Kim W. McIntyre
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Bethanne Warrack
;
Luisa Salter-Cid
;
Murray McKinnon
;
J
oel C. Barrish
;
Percy H. Carter
;
William
J
. Pitts
;
J
enny Xie
;
Alaric
J
.
Dyckman
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
6.
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
作者:
Hai-Yun Xiao
;
Scott H. Watterson
;
Charles M. Langevine
;
Anurag S. Srivastava
;
Soo S. Ko
;
Yanlei Zhang
;
Robert
J
. Cherney
;
Wei-Wei Guo
;
J
ohn L. Gilmore
;
J
ames E. Sheppeck II
;
Dauh-Rurng Wu
;
Peng Li
;
Duraisamy Ramasamy
;
Piramanayagam Arunachalam
;
Arvind Mathur
;
Tracy L. Taylor
;
David
J
. Shuster
;
Kim W. McIntyre
;
Ding-Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvi
j
ic
;
Anthony M. Marino
;
Praveen V. Balimane
;
Zheng Yang
;
Dana M. Banas
;
Georgia Cornelius
;
Celia
J
. D’Arienzo
;
Bethanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Salter-Cid
;
J
enny Xie
;
J
oel C. Barrish
;
Percy H. Carter
;
Alaric
J
.
Dyckman
;
T. G. Murali Dhar
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
7.
Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator
作者:
Michael G. YangZili Xiao
;
T. G. Murali Dhar
;
Hai-Yun Xiao
;
J
ohn L. Gilmore
;
David Marcoux
;
J
enny H. Xie
;
Kim W. McIntyre
;
Tracy L. Taylor
;
Virna Borowski
;
Elizabeth Heimrich
;
Yu-Wen Li
;
J
ianlin Feng
;
Alda Fernandes
;
Zheng Yang
;
Praveen Balimane
;
Anthony M. Marino
;
Georgia Cornelius
;
Bethanne M. Warrack
;
Arvind Mathur
;
Dauh-Rurng Wu
;
Peng Li
;
Anuradha Gupta
;
Bala Pragalathan
;
Ding Ren Shen
;
Mary Ellen Cvi
j
ic
;
Lois D. Lehman-McKeeman
;
Luisa Salter-Cid
;
J
oel C. Barrish
;
Percy H. Carter
;
Alaric
J
.
Dyckman
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
8.
Development of a Practical Synthesis of a p38 Kinase Inhibitor via a Safe and Robust Amination
作者:
Zhongping Shi
;
Susanne Kiau
;
Paul Lobben
;
J
ohn Hynes
;
J
r.
;
Hong Wu
;
Luca Parlanti
;
Robert Discordia
;
Wendel W. Doubleday
;
Katerina Leftheris
;
Alaric
J
.
Dyckman
;
Stephen T. Wrobleski
;
Konstantinos Dambalas
;
Srinivas Tummala
;
Simon Leung
;
Ehrlic Lo
刊名:Organic Process Research & Development
出版年:2012
9.
Discovery of 4-(5-(Cyclopropylcarbamoyl)-2-methylphenylamino)-5-methyl-N-propylpyrrolo[1,2-f][1,2,4]triazine-6-carboxamide (BMS-582949), a Clinical p38α MAP Kinase Inhibitor for the
作者:
Chun
j
ian Liu
;
J
ames Lin
;
Stephen T. Wrobleski
;
Shuqun Lin
;
J
ohn Hynes
;
J
r.
;
Hong Wu
;
Alaric
J
.
Dyckman
;
Tianle Li
;
J
ohn Wityak
;
Kathleen M. Gillooly
;
Sidney Pitt
;
Ding Ren Shen
;
Rosemary F. Zhang
;
Kim
刊名:
J
ournal of Medicinal Chemistry
出版年:2010
10.
Design, Synthesis, and Anti-inflammatory Properties of Orally Active 4-(Phenylamino)-pyrrolo[2,1-f][1,2,4]triazine p38α Mitogen-Activated Protein Kinase Inhibitors
作者:
J
ohn Hynes Jr.
;
Alaric
J
.
Dyckman
;
Shuqun Lin
;
Stephen T. Wrobleski
;
Hong Wu
;
Kathleen M. Gillooly
;
Steven B. Kanner
;
Herinder Lonial
;
Derek Loo
;
Kim W. McIntyre
;
Sidney Pitt
;
Ding Ren Shen
;
David
J
.
刊名:
J
ournal of Medicinal Chemistry
出版年:2008
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