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Wiley电子期刊(5)
SpringerLink电子期刊(3)
NATURE电子期刊(3)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
21
条
1.
Discovery of New Bromodomain Scaffolds by Biosensor Fragment Screening
作者:
Iva Navratilova
;
Tonia Aristotelous
;
Sarah Picaud
;
Apirat
Chaikuad
;
Stefan Knapp
;
Panagis Filappakopoulos
;
Andrew L. Hopkins
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B
作者:
Peiling Chen
;
Apirat
Chaikuad
;
Paul Bamborough
;
Marcus Bantscheff
;
Chas Bountra
;
Chun-wa Chung
;
Oleg Fedorov
;
Paola Grandi
;
David Jung
;
Robert Lesniak
;
Matthew Lindon
;
Susanne Müller
;
Martin Philpott
;
Rab Prinjha
;
Catherine Rogers
;
Carolyn Selenski
;
Cynthia Tallant
;
Thilo Werner
;
Timothy M. Willson
;
Stefan Knapp
;
David H. Drewry
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Structure-Based Identification of Inhibitory Fragments Targeting the p300/CBP-Associated Factor Bromodomain
作者:
Apirat
Chaikuad
;
Steffen Lang
;
Paul E. Brennan
;
Claudia Temperini
;
Oleg Fedorov
;
Johan Hollander
;
Ruta Nachane
;
Chris Abell
;
Susanne Müller
;
Gregg Siegal
;
Stefan Knapp
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases
作者:
Apirat
Chaikuad
;
Julien Diharce
;
Martin Schröder
;
Alicia Foucourt
;
Bertrand Leblond
;
Anne-Sophie Casagrande
;
Laurent Désiré
;
Pascal Bonnet
;
Stefan Knapp
;
Thierry Besson
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Bisubstrate Inhibitor Approach for Targeting Mitotic Kinase Haspin
作者:
Katrin Kestav
;
Darja Lavogina
;
Gerda Raidaru
;
Apirat
Chaikuad
;
Stefan Knapp
;
Asko Uri
刊名:Bioconjugate Chemistry
出版年:2015
6.
Structure Enabled Design of BAZ2-ICR, A Chemical Probe Targeting the Bromodomains of BAZ2A and BAZ2B
作者:
Ludovic Drouin
;
Sally McGrath
;
Lewis R. Vidler
;
Apirat
Chaikuad
;
Octovia Monteiro
;
Cynthia Tallant
;
Martin Philpott
;
Catherine Rogers
;
Oleg Fedorov
;
Manjuan Liu
;
Wasim Akhtar
;
Angela Hayes
;
Florence Raynaud
;
Susanne M眉ller
;
Stefan Knapp
;
Swen Hoelder
刊名:Journal of Medicinal Chemistry
出版年:2015
7.
10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A
作者:
Hannes Falke
;
Apirat
Chaikuad
;
Anja Becker
;
Nad猫ge Loa毛c
;
Olivier Lozach
;
Samira Abu Jhaisha
;
Walter Becker
;
Peter G. Jones
;
Lutz Preu
;
Knut Baumann
;
Stefan Knapp
;
Laurent Meijer
;
Conrad Kunick
刊名:Journal of Medicinal Chemistry
出版年:2015
8.
Selective Inhibitors of Cyclin G Associated Kinase (GAK) as Anti-Hepatitis C Agents
作者:
Sona Kovackova
;
Lei Chang
;
Elena Bekerman
;
Gregory Neveu
;
Rina Barouch-Bentov
;
Apirat
Chaikuad
;
Christina Heroven
;
Michal 艩谩la
;
Steven De Jonghe
;
Stefan Knapp
;
Shirit Einav
;
Piet Herdewijn
刊名:Journal of Medicinal Chemistry
出版年:2015
9.
Targeting Low-Druggability Bromodomains: Fragment Based Screening and Inhibitor Design against the BAZ2B Bromodomain
作者:
Fleur M. Ferguson
;
Oleg Fedorov
;
Apirat
Chaikuad
;
Martin Philpott
;
Joao R. C. Muniz
;
Ildiko Felletar
;
Frank von Delft
;
Tom Heightman
;
Stefan Knapp
;
Chris Abell
;
Alessio Ciulli
刊名:Journal of Medicinal Chemistry
出版年:2013
10.
Structure of Lactate Dehydrogenase from Plasmodium vivax: Complexes with NADH and APADH
作者:
Apirat
Chaikuad
;
Victoria Fairweather
;
Rebecca Conners
;
Tim Joseph-Horne
;
Dilek Turgut-Balik
;
and R. Leo Brady
刊名:Biochemistry
出版年:2005
1
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