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在“
ACS电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
285
条
1.
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
作者:
Essa
Hu
;
Ning Chen
;
Roxanne K. Kunz
;
Dah-Ren Hwang
;
Klaus Michelsen
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Randall
Hu
ngate
;
James Treanor
;
Hang Chen
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors
作者:
Ryan P. Wurz
;
Liping H. Pettus
;
Kate Ashton
;
James Brown
;
Jian Jeffrey Chen
;
Brad Herberich
;
Fang-Tsao Hong
;
Essa
Hu
-Harrington
;
Tom Nguyen
;
David J. St. Jean
;
Jr.
;
Seifu Tadesse
;
David Bauer
;
Michele Kubryk
;
Jing
hu
i Zhan
;
Keegan Cooke
;
Petia Mitchell
;
Kristin L. Andrews
;
Faye Hsieh
;
Dean Hickman
;
Nataraj Kalyanaraman
;
Tian Wu
;
Darren L. Reid
;
Edward K. Lobenhofer
;
Dina A. Andrews
;
Nancy Everds
;
Roberto Guzman
;
Andrew T. Parsons
;
Simon J. Hedley
;
Jason Tedrow
;
Oliver R. Thiel
;
Matthew Potter
;
Robert Radinsky
;
Pedro J. Beltran
;
Andrew S. Tasker
刊名:ACS Medicinal Chemistry Letters
出版年:2015
3.
Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
作者:
Essa
Hu
;
Kristin Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Silke Miller
;
Geraldine Hill Della Puppa
;
Mary Dovlatyan
;
Hang Chen
;
Dianna Lester-Zeiner
;
Jessica Able
;
Christopher Biorn
;
Ji Ma
;
Jianxia Shi
;
James Treanor
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2014
4.
Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phos
作者:
Essa
Hu
;
Ning Chen
;
Matthew P. Bourbeau
;
Paul E. Harrington
;
Kaustav Biswas
;
Roxanne K. Kunz
;
Kristin L. Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Jean Danao
;
Jessica Able
;
Madelyn Cueva
;
Santosh Talreja
;
Thomas Kornecook
;
Hang Chen
;
Amy Porter
;
Randall
Hu
ngate
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
作者:
Essa
Hu
;
Roxanne K. Kunz
;
Ning Chen
;
Shannon Rumfelt
;
Aaron Siegmund
;
Kristin Andrews
;
Samer Chmait
;
Sharon Zhao
;
Carl Davis
;
Hang Chen
;
Dianna Lester-Zeiner
;
Ji Ma
;
Christopher Biorn
;
Jianxia Shi
;
Amy Porter
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Rapid Identification of a Novel Small Molecule Phosphodiesterase 10A (PDE10A) Tracer
作者:
Essa
Hu
;
Ji Ma
;
Christopher Biorn
;
Dianna Lester-Zeiner
;
Robert Cho
;
Shannon Rumfelt
;
Roxanne K. Kunz
;
Thomas Nixey
;
Klaus Michelsen
;
Silke Miller
;
Jianxia Shi
;
Jamie Wong
;
Geraldine Hill Della Puppa
;
Jessica Able
;
Santosh Talreja
;
Dah-Ren Hwang
;
Stephen A. Hitchcock
;
Amy Porter
;
David Immke
;
Jennifer R. Allen
;
James Treanor
;
Hang Chen
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
Discovery of Aryl Aminoquinazoline Pyridones as Potent, Selective, and Orally Efficacious Inhibitors of Receptor Tyrosine Kinase c-Kit
作者:
Essa
Hu
;
Andrew Tasker
;
Ryan D. White
;
Roxanne K. Kunz
;
Jason
Hu
man
;
Ning Chen
;
Roland Bü
;
rli
;
Randall
Hu
ngate
;
Perry Novak
;
Andrea Itano
;
Xuxia Zhang
;
Violeta Yu
;
Yen Nguyen
;
Yanyan Tudor
;
Matthe
刊名:Journal of Medicinal Chemistry
出版年:2008
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