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Elsevier电子期刊(6)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
16
条
1.
Discovery and Biological Characterization of (2R,4S)-1鈥?Acetyl-N-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl}-2-(4-fluoro-2-methylphenyl)-N-methyl-4,4鈥?bipiperidin
作者:
Romano Di Fabio
;
Giuseppe Alvaro
;
Cristiana Griffante
;
Domenica A. Pizzi
;
Daniele Donati
;
Mario Mattioli
;
Zadeo Cimarosti
;
Giuseppe Guercio
;
Carla Marchioro
;
Stefano
Provera
;
Laura Zonzini
;
Dino Montanari
;
Sergio Melotto
;
Philip A. Gerrard
;
David G. Trist
;
Emiliangelo Ratti
;
Mauro Corsi
刊名:Journal of Medicinal Chemistry
出版年:2011
2.
Overall Synthesis of GSK356278: Quick Delivery of a PDE4 Inhibitor Using a Fit-for-Purpose Approach
作者:
Giuseppe Guercio
;
Damiano Castoldi
;
Nicola Giubellina
;
Alessandro Lamonica
;
Arianna Ribecai
;
Paolo Stabile
;
Pieter Westerduin
;
Riet Dams
;
Anna Nicoletti
;
Sara Rossi
;
Claudio Bismara
;
Stefano
Provera
L
刊名:Organic Process Research & Development
出版年:2010
3.
An Efficient Scalable Route for the Synthesis of Enantiomerically Pure tert-Butyl-(1R,4S,6R)-4-(hydroxymethyl)-3-azabicyclo[4.1.0]heptane-3-carboxylate
作者:
William M. Maton
;
Federica Stazi
;
Angelo Maria Manzo
;
Roberta Pachera
;
Arianna Ribecai
;
Paolo Stabile
;
Alcide Perboni
;
Nicola Giubellina
;
Fernando Bravo
;
Damiano Castoldi
;
Stefano
Provera
;
Lucilla Tur
刊名:Organic Process Research & Development
出版年:2010
4.
Development of a Dynamic Kinetic Resolution for the Isolation of an Intermediate in the Synthesis of Casopitant Mesylate: Application of QbD Principles in the Definition of the Parameter Ranges, Issue
作者:
Fernando Bravo
;
Zadeo Cimarosti
;
Francesco Tinazzi
;
Gillian E. Smith
;
Damiano Castoldi
;
Stefano
Provera
;
Pieter Westerduin
刊名:Organic Process Research & Development
出版年:2010
5.
The Synthesis of GV143253A: A Case Study for the Use of Analytical and Statistical Tools to Elucidate the Reaction Mechanism and to Optimize the Process
作者:
Giuseppe Guercio
;
Alcide Perboni
;
Francesco Tinazzi
;
Luca Rovatti
;
Stefano
Provera
刊名:Organic Process Research & Development
出版年:2010
6.
Identification of a Manufacturing Route of Novel CRF-1 Antagonists Containing a 2,3-Dihydro-1H-pyrrolo[2,3-b]pyridine Moiety
作者:
Arianna Ribecai
;
Sergio Bacchi
;
Monica Delpogetto
;
Simone Guelfi
;
Angelo Maria Manzo
;
Alcide Perboni
;
Paolo Stabile
;
Pieter Westerduin
;
Marie Hourdin
;
Sara Rossi
;
Stefano
Provera
;
Lucilla Turco
刊名:Organic Process Research & Development
出版年:2010
7.
Application of the QbD Principles in the Development of the Casopitant Mesylate Manufacturing Process. Process Research Studies for the Definition of the Control Strategy of some Drug Substance-CQAs f
作者:
Zadeo Cimarosti
;
Fernando Bravo
;
Damiano Castoldi
;
Francesco Tinazzi
;
Stefano
Provera
;
Alcide Perboni
;
Damiano Papini
;
Pieter Westerduin
刊名:Organic Process Research & Development
出版年:2010
8.
Synthesis of the NK1 Receptor Antagonist GW597599. Part 2: Development of a Scalable Route to a Key Chirally Pure Arylpiperazine
作者:
Giuseppe Guercio
;
Angelo Maria Manzo
;
Michael Goodyear
;
Sergio Bacchi
;
Stefano
Curti
;
Stefano
Provera
刊名:Organic Process Research & Development
出版年:2009
9.
Synthesis of the NK1 Receptor Antagonist GW597599. Part 3: Development of a Scalable Route to a Key Chirally Pure Arylpiperazine Urea, A Happy End
作者:
Giuseppe Guercio
;
Sergio Bacchi
;
Alcide Perboni
;
Corinne Leroi
;
Francesco Tinazzi
;
Ilaria Bientinesi
;
Marie Hourdin
;
Michael Goodyear
;
Stefano
Curti
;
Stefano
Provera
;
Zadeo Cimarosti
刊名:Organic Process Research & Development
出版年:2009
10.
Design, Synthesis, and Biological Evaluation of Novel Aminobisphosphonates Possessing an in Vivo Antitumor Activity Through a γδ-T Lymphocytes-Mediated Activation Mechanism
作者:
Daniele Simoni
;
Nicola Gebbia
;
Francesco Paolo Invidiata
;
Marco Eleopra
;
Paolo Marchetti
;
Riccardo Rondanin
;
Riccardo Baruchello
;
Stefano
Provera
;
Carla Marchioro
;
Manlio Tolomeo
;
Luciana Marinelli
;
V
刊名:Journal of Medicinal Chemistry
出版年:2008
1
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