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内部出版物
在“
ACS电子期刊
”中,
命中:
8
条,耗时:小于0.01 秒
1.
Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARα Selective Agonist
作者:
Yan Shi
;
Jun Li
;
Lawrence J. Kennedy
;
Shiwei Tao
;
Andrés S. Hernández
;
Zhi Lai
;
Sean Chen
;
Henry Wong
;
Juliang Zhu
;
Ashok Trehan
;
Ngiap-Kie Lim
;
Huiping Zhang
;
Bang-Chi Chen
;
Kenneth T. Locke
;
Kevin M. O’Malley
;
Litao Zhang
;
Rai Ajit Srivastava
;
Bowman Miao
;
Daniel S. Meyers
;
Hossain Monshizadegan
;
Debra Search
;
Denise Grimm
;
Rongan Zhang
;
Thomas Harrity
;
Lori K. Kunselman
;
Michael Cap
;
Jodi Muckelbauer
;
Chiehying
Chang
;
Stanley R. Krystek
;
Yi-Xin Li
;
Vinayak Hosagrahara
;
Lisa Zhang
;
Pathanjali Kadiyala
;
Carrie Xu
;
Michael A. Blanar
;
Robert Zahler
;
Ranjan Mukherjee
;
Peter T. W. Cheng
;
Joseph A. Tino
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Targeting the BACE1 Active Site Flap Leads to a Potent Inhibitor That Elicits Robust Brain Aβ Reduction in Rodents
作者:
Yong-Jin Wu
;
Jason Guernon
;
Fukang Yang
;
Lawrence Snyder
;
Jianliang Shi
;
Andrea Mcclure
;
Ramkumar Rajamani
;
Hyunsoo Park
;
Alicia Ng
;
Hal Lewis
;
ChiehYing
Chang
;
Dan Camac
;
Jeremy H. Toyn
;
Michael K. Ahlijanian
;
Charles F. Albright
;
John E. Macor
;
Lorin A. Thompson
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery of S3-Truncated, C-6 Heteroaryl Substituted Aminothiazine β-Site APP Cleaving Enzyme-1 (BACE1) Inhibitors
作者:
Yong-Jin Wu
;
Jason Guernon
;
Jianliang Shi
;
Lawrence Marcin
;
Mendi Higgins
;
Ramkumar Rajamani
;
Jodi Muckelbauer
;
Hal Lewis
;
ChiehYing
Chang
;
Dan Camac
;
Jeremy H. Toyn
;
Michael K. Ahlijanian
;
Charles F. Albright
;
John E. Macor
;
Lorin A. Thompson
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Small Molecule Reversible Inhibitors of Bruton’s Tyrosine Kinase (BTK): Structure–Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177)
作者:
George V. De Lucca
;
Qing Shi
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Rick Rampulla
;
Arvind Mathur
;
Lorell Discenza
;
Celia D’Arienzo
;
Jun Dai
;
Mary Obermeier
;
Rodney Vickery
;
Yingru Zhang
;
Zheng Yang
;
Punit Marathe
;
Andrew J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing
J.
Chang
;
Huiping Zhang
;
Kathleen Gillooly
;
Tracy Taylor
;
Mark A. Pattoli
;
Stacey Skala
;
Daniel W. Kukral
;
Kim W. McIntyre
;
Luisa Salter-Cid
;
Aberra Fura
;
James R. Burke
;
Joel C. Barrish
;
Percy H. Carter
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked
作者:
Scott H. Watterson
;
George V. De Lucca
;
Qing Shi
;
Charles M. Langevine
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Hua Gong
;
Jun Dai
;
Shiuhang Yip
;
Peng Li
;
Dawn Sun
;
Dauh-Rurng Wu
;
Chunlei Wang
;
Yingru Zhang
;
Sarah C. Traeger
;
Mark A. Pattoli
;
Stacey Skala
;
Lihong Cheng
;
Mary T. Obermeier
;
Rodney Vickery
;
Lorell N. Discenza
;
Celia J. D’Arienzo
;
Yifan Zhang
;
Elizabeth Heimrich
;
Kathleen M. Gillooly
;
Tracy L. Taylor
;
Claudine Pulicicchio
;
Kim W. McIntyre
;
Michael A. Galella
;
Andy J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing
Chang
;
Richard Rampulla
;
Arvind Mathur
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Aberra Fura
;
James R. Burke
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Image Annotation and Database Mining to Create a Novel Screen for the Chemotype-Dependent Crystallization of HCV NS3 Protease
作者:
Herbert E. Klei
;
Kevin Kish
;
Mark F. Russo
;
Steve J. Michalczyk
;
Matthew H. Cahn
;
Jeffrey Tredup
;
ChiehYing
Chang
;
Javed Khan
;
Eric T. Baldwin
刊名:Crystal Growth & Design
出版年:2011
7.
Discovery of a 2,4-Disubstituted Pyrrolo[1,2-f][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development
作者:
Mark D. Wittman
;
Joan M. Carboni
;
Zheng Yang
;
Francis Y. Lee
;
Melissa Antman
;
Ricardo Attar
;
Praveen Balimane
;
Chiehying
Chang
;
Cliff Chen
;
Lorell Discenza
;
David Frennesson
;
Marco M. Gottardis
;
Ann G
刊名:Journal of Medicinal Chemistry
出版年:2009
8.
Molecular, Biological, and Preliminary Structural Analysis of Recombinant Bryodin 1, a Ribosome-Inactivating Protein from the Plant Bryonia dioica
作者:
Susan L. Gawlak
;
Michael Neubauer
;
Herbert E. Klei
;
ChiehYing
Y.
Chang
;
Howard M. Einspahr
;
and Clay B. Siegall
刊名:Biochemistry
出版年:1997
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