设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
CNKI学位论文(1)
在“
ACS电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent
作者:
Paola Vianello
;
Oronza A. Botrugno
;
Anna Cappa
;
Roberto Dal Zuffo
;
Paola Dessanti
;
Antonello Mai
;
Biagina Marrocco
;
Andrea Mattevi
;
Giuseppe Meroni
;
Saverio Minucci
;
Giulia Stazi
;
Florian Thaler
;
Paolo Trifiró
;
Sergio Valente
;
Manuela Villa
;
Mario Varasi
;
Ciro
Mercurio
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Pure Diastereomers of a Tranylcypromine-Based LSD1 Inhibitor: Enzyme Selectivity and In-Cell Studies
作者:
Sergio Valente
;
Veronica Rodriguez
;
Ciro
Mercurio
;
Paola Vianello
;
Bruna Saponara
;
Roberto Cirilli
;
Giuseppe Ciossani
;
Donatella Labella
;
Biagina Marrocco
;
Giovanni Ruoppolo
;
Oronza A. Botrugno
;
Paola Dessanti
;
Saverio Minucci
;
Andrea Mattevi
;
Mario Varasi
;
Antonello Mai
刊名:ACS Medicinal Chemistry Letters
出版年:2015
3.
New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer
作者:
Giuseppe La Regina
;
Ruoli Bai
;
Antonio Coluccia
;
Valeria Famiglini
;
Sveva Pelliccia
;
Sara Passacantilli
;
Carmela Mazzoccoli
;
Vitalba Ruggieri
;
Annalisa Verrico
;
Andrea Miele
;
Ludovica Monti
;
Marianna Nalli
;
Romina Alfonsi
;
Lucia Di Marcotullio
;
Alberto Gulino
;
Biancamaria Ricci
;
Alessandra Soriani
;
Angela Santoni
;
Michele Caraglia
;
Stefania Porto
;
Eleonora Da Pozzo
;
Claudia Martini
;
Andrea Brancale
;
Luciana Marinelli
;
Ettore Novellino
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro
Mercurio
;
Chiara Bigogno
;
Giulio Dondio
;
Ernest Hamel
;
Patrizia Lavia
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
New Pyrrole Derivatives with Potent Tubulin Polymerization Inhibiting Activity As Anticancer Agents Including Hedgehog-Dependent Cancer
作者:
Giuseppe La Regina
;
Ruoli Bai
;
Antonio Coluccia
;
Valeria Famiglini
;
Sveva Pelliccia
;
Sara Passacantilli
;
Carmela Mazzoccoli
;
Vitalba Ruggieri
;
Lorenza Sisinni
;
Alessio Bolognesi
;
Whilelmina Maria Rensen
;
Andrea Miele
;
Marianna Nalli
;
Romina Alfonsi
;
Lucia Di Marcotullio
;
Alberto Gulino
;
Andrea Brancale
;
Ettore Novellino
;
Giulio Dondio
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro
Mercurio
;
Ernest Hamel
;
Patrizia Lavia
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors
作者:
Giuseppe La Regina
;
Ruoli Bai
;
Whilelmina Maria Rensen
;
Erica Di Cesare
;
Antonio Coluccia
;
Francesco Piscitelli
;
Valeria Famiglini
;
Alessia Reggio
;
Marianna Nalli
;
Sveva Pelliccia
;
Eleonora Da Pozzo
;
Barbara Costa
;
Ilaria Granata
;
Amalia Porta
;
Bruno Maresca
;
Alessandra Soriani
;
Maria Luisa Iannitto
;
Angela Santoni
;
Junjie Li
;
Marlein Miranda Cona
;
Feng Chen
;
Yicheng Ni
;
Andrea Brancale
;
Giulio Dondio
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro
Mercurio
;
Claudia Martini
;
Ernest Hamel
;
Patrizia Lavia
;
Ettore Novellino
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Design and Synthesis of 2-Heterocyclyl-3-arylthio-1H-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability
作者:
Giuseppe La Regina
;
Ruoli Bai
;
Willeke Rensen
;
Antonio Coluccia
;
Francesco Piscitelli
;
Valerio Gatti
;
Alessio Bolognesi
;
Antonio Lavecchia
;
Ilaria Granata
;
Amalia Porta
;
Bruno Maresca
;
Alessandra Soriani
;
Maria Luisa Iannitto
;
Marisa Mariani
;
Angela Santoni
;
Andrea Brancale
;
Cristiano Ferlini
;
Giulio Dondio
;
Mario Varasi
;
Ciro
Mercurio
;
Ernest Hamel
;
Patrizia Lavia
;
Ettore Novellino
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2011
7.
Discovery, Synthesis, and Pharmacological Evaluation of Spiropiperidine Hydroxamic Acid Based Derivatives as Structurally Novel Histone Deacetylase (HDAC) Inhibitors
作者:
Mario Varasi
;
Florian Thaler
;
Agnese Abate
;
Chiara Bigogno
;
Roberto Boggio
;
Giacomo Carenzi
;
Tiziana Cataudella
;
Roberto Dal Zuffo
;
Maria Carmela Fulco
;
Marco Giulio Rozio
;
Antonello Mai
;
Giulio Dondio
;
Saverio Minucci
;
Ciro
Mercurio
刊名:Journal of Medicinal Chemistry
出版年:2011
8.
Identification of Potent Pyrazolo[4,3-h]quinazoline-3-carboxamides as Multi-Cyclin-Dependent Kinase Inhibitors
作者:
Gabriella Traquandi
;
Marina Ciomei
;
Dario Ballinari
;
Elena Casale
;
Nicoletta Colombo
;
Valter Croci
;
Francesco Fiorentini
;
Antonella Isacchi
;
Antonio Longo
;
Ciro
Mercurio
;
Achille Panzeri
;
Wilma Pastor
刊名:Journal of Medicinal Chemistry
出版年:2010
9.
Triazole-Modified Histone Deacetylase Inhibitors As a Rapid Route to Drug Discovery
作者:
Tracey Pirali
;
Francesca Pagliai
;
Ciro
Mercurio
;
Roberto Boggio
;
Pier Luigi Canonico
;
Giovanni Sorba
;
Gian Cesare Tron
;
Armando A. Genazzani
刊名:Journal of Combinatorial Chemistry
出版年:2008
1
按检索点细分(9)
题名(9)
按出版年细分(9)
2016年(1)
2015年(2)
2014年(1)
2013年(1)
2011年(2)
2010年(1)
2008年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.