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内部出版物
在“
ACS电子期刊
”中,
命中:
5
条,耗时:小于0.01 秒
1.
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
作者:
Essa Hu
;
Ning Chen
;
Roxanne K. Kunz
;
Dah-Ren Hwang
;
Klaus Michelsen
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna
Lester
-
Zeiner
;
Randall Hungate
;
James Treanor
;
Hang Chen
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
作者:
Essa Hu
;
Kristin Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Silke Miller
;
Geraldine Hill Della Puppa
;
Mary Dovlatyan
;
Hang Chen
;
Dianna
Lester
-
Zeiner
;
Jessica Able
;
Christopher Biorn
;
Ji Ma
;
Jianxia Shi
;
James Treanor
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2014
3.
Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phos
作者:
Essa Hu
;
Ning Chen
;
Matthew P. Bourbeau
;
Paul E. Harrington
;
Kaustav Biswas
;
Roxanne K. Kunz
;
Kristin L. Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna
Lester
-
Zeiner
;
Jean Danao
;
Jessica Able
;
Madelyn Cueva
;
Santosh Talreja
;
Thomas Kornecook
;
Hang Chen
;
Amy Porter
;
Randall Hungate
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
作者:
Essa Hu
;
Roxanne K. Kunz
;
Ning Chen
;
Shannon Rumfelt
;
Aaron Siegmund
;
Kristin Andrews
;
Samer Chmait
;
Sharon Zhao
;
Carl Davis
;
Hang Chen
;
Dianna
Lester
-
Zeiner
;
Ji Ma
;
Christopher Biorn
;
Jianxia Shi
;
Amy Porter
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2013
5.
Rapid Identification of a Novel Small Molecule Phosphodiesterase 10A (PDE10A) Tracer
作者:
Essa Hu
;
Ji Ma
;
Christopher Biorn
;
Dianna
Lester
-
Zeiner
;
Robert Cho
;
Shannon Rumfelt
;
Roxanne K. Kunz
;
Thomas Nixey
;
Klaus Michelsen
;
Silke Miller
;
Jianxia Shi
;
Jamie Wong
;
Geraldine Hill Della Puppa
;
Jessica Able
;
Santosh Talreja
;
Dah-Ren Hwang
;
Stephen A. Hitchcock
;
Amy Porter
;
David Immke
;
Jennifer R. Allen
;
James Treanor
;
Hang Chen
刊名:Journal of Medicinal Chemistry
出版年:2012
1
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