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CNKI学位论文(77)
知网期刊论文(16)
在“
ACS电子期刊
”中,
命中:
12
条,耗时:小于0.01 秒
在所有数据库中总计命中:
93
条
1.
Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement
作者:
Isaac E. Marx
;
Thomas A. Dineen
;
Jessica Able
;
Christiane Bode
;
Howard
Bregman
;
Margaret Chu-Moyer
;
Erin F. DiMauro
;
Bingfan Du
;
Robert S. Foti
;
Robert T. Fremeau Jr.
;
Hua Gao
;
Hakan Gunaydin
;
Brian E. Hall
;
Liyue Huang
;
Thomas Kornecook
;
Charles R. Kreiman
;
Daniel S. La
;
Joseph Ligutti
;
Min-Hwa Jasmine Lin
;
Dong Liu
;
Jeff S. McDermott
;
Bryan D. Moyer
;
Emily A. Peterson
;
Jonathan T. Roberts
;
Paul Rose
;
Jean Wang
;
Beth D. Youngblood
;
Violeta Yu
;
Matthew M. Weiss
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors
作者:
Erin F. DiMauro
;
Stephen Altmann
;
Loren M. Berry
;
Howard
Bregman
;
Nagasree Chakka
;
Margaret Chu-Moyer
;
Elma Feric Bojic
;
Robert S. Foti
;
Robert Fremeau
;
Hua Gao
;
Hakan Gunaydin
;
Angel Guzman-Perez
;
Brian E. Hall
;
Hongbing Huang
;
Michael Jarosh
;
Thomas Kornecook
;
Josie Lee
;
Joseph Ligutti
;
Dong Liu
;
Bryan D. Moyer
;
Daniel Ortuno
;
Paul E. Rose
;
Laurie B. Schenkel
;
Kristin Taborn
;
Jean Wang
;
Yan Wang
;
Violeta Yu
;
Matthew M. Weiss
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Structure-Based Design of 2-Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors
作者:
Hongbing Huang
;
Angel Guzman-Perez
;
Lisa Acquaviva
;
Virginia Berry
;
Howard
Bregman
;
Jennifer Dovey
;
Hakan Gunaydin
;
Xin Huang
;
Liyue Huang
;
Doug Saffran
;
Randy Serafino
;
Steve Schneider
;
Cindy Wilson
;
Erin F. DiMauro
刊名:ACS Medicinal Chemistry Letters
出版年:2013
4.
Discovery of a Class of Novel Tankyrase Inhibitors that Bind to Both the Nicotinamide Pocket and the Induced Pocket
作者:
Howard
Bregman
;
Hakan Gunaydin
;
Yan Gu
;
Steve Schneider
;
Cindy Wilson
;
Erin F. DiMauro
;
Xin Huang
刊名:Journal of Medicinal Chemistry
出版年:2013
5.
Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Howard
Bregman
;
Nagasree Chakka
;
Angel Guzman-Perez
;
Hakan Gunaydin
;
Yan Gu
;
Xin Huang
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue Huang
;
Bryan Egge
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Ankita Mishra
;
John Newcomb
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Zihao Hua
;
Howard
Bregman
;
John L. Buchanan
;
Nagasree Chakka
;
Angel Guzman-Perez
;
Hakan Gunaydin
;
Xin Huang
;
Yan Gu
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue Huang
;
Bryan Egge
;
Renee Emkey
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Lisa Acquaviva
;
Jennifer Dovey
;
Ankita Mishra
;
John Newcomb
;
Douglas Saffran
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Mary Stanton
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Structure-Based Design of Potent and Selective CK1纬 Inhibitors
作者:
Hongbing Huang
;
Lisa Acquaviva
;
Virginia Berry
;
Howard
Bregman
;
Nagasree Chakka
;
Anne O鈥機onnor
;
Erin F. DiMauro
;
Jennifer Dovey
;
Oleg Epstein
;
Barbara Grubinska
;
Jon Goldstein
;
Hakan Gunaydin
;
Zihao Hua
;
Xin Huang
;
Liyue Huang
;
Jason Human
;
Alex Long
;
John Newcomb
;
Vinod F. Patel
;
Doug Saffran
;
Randy Serafino
;
Steve Schneider
;
Craig Strathdee
;
Jin Tang
;
Susan Turci
;
Ryan White
;
Violeta Yu
;
Huilin Zhao
;
Cindy Wilson
;
Matthew W. Martin
刊名:ACS Medicinal Chemistry Letters
出版年:2012
8.
Identification of a Potent, State-Dependent Inhibitor of Nav1.7 with Oral Efficacy in the Formalin Model of Persistent Pain
作者:
Howard
Bregman
;
Loren Berry
;
John L. Buchanan
;
April Chen
;
Bingfan Du
;
Elma Feric
;
Markus Hierl
;
Liyue Huang
;
David Immke
;
Brett Janosky
;
Danielle Johnson
;
Xingwen Li
;
Joseph Ligutti
;
Dong Liu
;
Annika Malmberg
;
David Matson
;
Jeff McDermott
;
Peter Miu
;
Hanh Nho Nguyen
;
Vinod F. Patel
;
Daniel Waldon
;
Ben Wilenkin
;
Xiao Mei Zheng
;
Anruo Zou
;
Stefan I. McDonough
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2011
9.
From Imide to Lactam Metallo-pyridocarbazoles: Distinct Scaffolds for the Design of Selective Protein Kinase Inhibitors
作者:
Nicholas Pagano
;
Eric Y. Wong
;
Tom Breiding
;
Haidong Liu
;
Alexander Wilbuer
;
Howard
Bregman
;
Qi Shen
;
Scott L. Diamond
;
Eric Meggers
刊名:Journal of Organic Chemistry
出版年:2009
10.
The Crystal Structure of BRAF in Complex with an Organoruthenium Inhibitor Reveals a Mechanism for Inhibition of an Active Form of BRAF Kinase
作者:
Peng Xie
;
Craig Streu
;
Jie Qin
;
Howard
Bregman
;
Nicholas Pagano
;
Eric Meggers
;
Ronen Marmorstein
刊名:Biochemistry
出版年:2009
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