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在“
ACS电子期刊
”中,
命中:
14
条,耗时:小于0.01 秒
在所有数据库中总计命中:
10
条
1.
Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer Agent
作者:
Yong Liu
;
Radoslaw Laufer
;
Narendra Kumar Patel
;
Grace Ng
;
Peter B. Sampson
;
Sze-Wan Li
;
Yunhui Lang
;
Miklos
Feher
;
Richard Brokx
;
Irina Beletskaya
;
Richard Hodgson
;
Olga Plotnikova
;
Donald E. Awrey
;
Wei Qiu
;
Nickolay Y. Chirgadze
;
Jacqueline M. Mason
;
Xin Wei
;
Dan Chi-Chia Lin
;
Yi Che
;
Reza Kiarash
;
Graham C. Fletcher
;
Tak W. Mak
;
Mark R. Bray
;
Henry W. Pauls
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
The Discovery of Polo-Like Kinase 4 Inhibitors: Identification of (1R,2S)-2-(3-((E)-4-(((cis)-2,6-Dimethylmorpholino)methyl)styryl)-1H-indazol-6-yl)-5鈥?methoxyspiro[
作者:
Peter B. Sampson
;
Yong Liu
;
Bryan Forrest
;
Graham Cumming
;
Sze-Wan Li
;
Narendra Kumar Patel
;
Louise Edwards
;
Radoslaw Laufer
;
Miklos
Feher
;
Fuqiang Ban
;
Donald E. Awrey
;
Guodong Mao
;
Olga Plotnikova
;
Richard Hodgson
;
Irina Beletskaya
;
Jacqueline M. Mason
;
Xunyi Luo
;
Vincent Nadeem
;
Xin Wei
;
Reza Kiarash
;
Brian Madeira
;
Ping Huang
;
Tak W. Mak
;
Guohua Pan
;
Henry W. Pauls
刊名:Journal of Medicinal Chemistry
出版年:2015
3.
The Discovery of Polo-Like Kinase 4 Inhibitors: Design and Optimization of Spiro[cyclopropane-1,3鈥瞇3H]indol]-2鈥?1鈥?i>H)-ones as Orally Bioavailable Antitumor Agents
作者:
Peter B. Sampson
;
Yong Liu
;
Narendra Kumar Patel
;
Miklos
Feher
;
Bryan Forrest
;
Sze-Wan Li
;
Louise Edwards
;
Radoslaw Laufer
;
Yunhui Lang
;
Fuqiang Ban
;
Donald E. Awrey
;
Guodong Mao
;
Olga Plotnikova
;
Genie Leung
;
Richard Hodgson
;
Jacqueline Mason
;
Xin Wei
;
Reza Kiarash
;
Erin Green
;
Wei Qiu
;
Nickolay Y. Chirgadze
;
Tak W. Mak
;
Guohua Pan
;
Henry W. Pauls
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
The Discovery of Orally Bioavailable Tyrosine Threonine Kinase (TTK) Inhibitors: 3-(4-(heterocyclyl)phenyl)-1H-indazole-5-carboxamides as Anticancer Agents
作者:
Yong Liu
;
Yunhui Lang
;
Narendra Kumar Patel
;
Grace Ng
;
Radoslaw Laufer
;
Sze-Wan Li
;
Louise Edwards
;
Bryan Forrest
;
Peter B. Sampson
;
Miklos
Feher
;
Fuqiang Ban
;
Donald E. Awrey
;
Irina Beletskaya
;
Guodong Mao
;
Richard Hodgson
;
Olga Plotnikova
;
Wei Qiu
;
Nickolay Y. Chirgadze
;
Jacqueline M. Mason
;
Xin Wei
;
Dan Chi-Chia Lin
;
Yi Che
;
Reza Kiarash
;
Brian Madeira
;
Graham C. Fletcher
;
Tak W. Mak
;
Mark R. Bray
;
Henry W. Pauls
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
The Discovery of PLK4 Inhibitors: (E)-3-((1H-Indazol-6-yl)methylene)indolin-2-ones as Novel Antiproliferative Agents
作者:
Radoslaw Laufer
;
Bryan Forrest
;
Sze-Wan Li
;
Yong Liu
;
Peter Sampson
;
Louise Edwards
;
Yunhui Lang
;
Donald E. Awrey
;
Guodong Mao
;
Olga Plotnikova
;
Genie Leung
;
Richard Hodgson
;
Irina Beletskaya
;
Jacqueline M. Mason
;
Xunyi Luo
;
Xin Wei
;
Yi Yao
;
Miklos
Feher
;
Fuqiang Ban
;
Reza Kiarash
;
Erin Green
;
Tak W. Mak
;
Guohua Pan
;
Henry W. Pauls
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Numerical Errors and Chaotic Behavior in Docking Simulations
作者:
Miklos
Feher
;
Christopher I. Williams
刊名:Journal of Chemical Information and Modeling
出版年:2012
7.
Numerical Errors in Minimization Based Binding Energy Calculations
作者:
Miklos
Feher
;
Christopher I. Williams
刊名:Journal of Chemical Information and Modeling
出版年:2012
8.
Structural Chemistry of the Histone Methyltransferases Cofactor Binding Site
作者:
Vale虂rie Campagna-Slater
;
Man Wai Mok
;
Kong T. Nguyen
;
Miklos
Feher
;
Rafael Najmanovich
;
Matthieu Schapira
刊名:Journal of Chemical Information and Modeling
出版年:2011
9.
Reducing Docking Score Variations Arising from Input Differences
作者:
Miklos
Feher
;
Christopher I. Williams
刊名:Journal of Chemical Information and Modeling
出版年:2010
10.
Effect of Input Differences on the Results of Docking Calculations
作者:
Miklos
Feher
;
Christopher I. Williams
刊名:Journal of Chemical Information and Modeling
出版年:2009
1
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