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知网期刊论文(2)
在“
ACS电子期刊
”中,
命中:
12
条,耗时:小于0.01 秒
在所有数据库中总计命中:
5
条
1.
Discovery and Optimization of Quinazolinone-pyrrolopyrrolones as Potent and Orally Bioavailable Pan-Pim Kinase Inhibitors
作者:
Liping H. Pettus
;
Kristin L. Andrews
;
Shon K. Booker
;
Jie Chen
;
Victor J. Cee
;
Frank Chavez Jr.
;
Yuping Chen
;
Heather Eastwood
;
Nadia Guerrero
;
Bradley Herberich
;
Dean Hickman
;
Brian A. Lanman
;
Jimmy Laszlo III
;
Matthew R. Lee
;
J. Russell Lipford
;
Bethany Mattson
;
Christopher Mohr
;
Yen Nguyen
;
Mark H. Norman
;
David Powers
;
Anthony B. Reed
;
Karen Rex
;
Christine Sastri
;
Nuria
Tamayo
;
Paul Wang
;
Jeffrey T. Winston
;
Bin Wu
;
Tian Wu
;
Ryan P. Wurz
;
Yang Xu
;
Yihong Zhou
;
Andrew S. Tasker
;
Hui-Ling Wang
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis
作者:
Nuria
A.
Tamayo
;
Mark H. Norman
;
Michael D. Bartberger
;
Fang-Tsao Hong
;
Yunxin Bo
;
Longbin Liu
;
Nobuko Nishimura
;
Kevin C. Yang
;
Seifu Tadesse
;
Christopher Fotsch
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Clarence Hale
;
Steven R. Jordan
;
David J. Lloyd
;
Glenn Sivits
;
Gwyneth Van
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2015
3.
Optimization of Potency and Pharmacokinetic Properties of Tetrahydroisoquinoline Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists
作者:
Daniel B. Horne
;
Nuria
A.
Tamayo
;
Michael D. Bartberger
;
Yunxin Bo
;
Jeffrey Clarine
;
Carl D. Davis
;
Vijay K. Gore
;
Matthew R. Kaller
;
Sonya G. Lehto
;
Vu V. Ma
;
Nobuko Nishimura
;
Thomas T. Nguyen
;
Phi Tang
;
Weiya Wang
;
Beth D. Youngblood
;
Maosheng Zhang
;
Narender R. Gavva
;
Holger Monenschein
;
Mark H. Norman
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 2. Leveraging Structure-Based Drug Design to Identify Analogues with Improved Pharmacokinetic Profiles
作者:
David J. St. Jean
;
Jr.
;
Kate S. Ashton
;
Michael D. Bartberger
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Elizabeth Galbreath
;
Joan Helmering
;
Fang-Tsao Hong
;
Steven R. Jordan
;
Longbin Liu
;
Roxanne K. Kunz
;
Klaus Michelsen
;
Nobuko Nishimura
;
Lewis D. Pennington
;
Steve F. Poon
;
Darren Reid
;
Glenn Sivits
;
Markian M. Stec
;
Seifu Tadesse
;
Nuria
Tamayo
;
Gwyneth Van
;
Kevin C. Yang
;
Jiandong Zhang
;
Mark H. Norman
;
Christopher Fotsch
;
David J. Lloyd
;
Clarence Hale
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Fused Piperidines as a Novel Class of Potent and Orally Available Transient Receptor Potential Melastatin Type 8 (TRPM8) Antagonists
作者:
Nuria
A.
Tamayo
;
Yunxin Bo
;
Vijay Gore
;
Vu Ma
;
Nobuko Nishimura
;
Phi Tang
;
Hong Deng
;
Lana Klionsky
;
Sonya G. Lehto
;
Weiya Wang
;
Brad Youngblood
;
Jiyun Chen
;
Tiffany L. Correll
;
Michael D. Bartberger
;
Narender R. Gavva
;
Mark H. Norman
刊名:Journal of Medicinal Chemistry
出版年:2012
6.
Selective Class I Phosphoinositide 3-Kinase Inhibitors: Optimization of a Series of Pyridyltriazines Leading to the Identification of a Clinical Candidate, AMG 511
作者:
Mark H. Norman
;
Kristin L. Andrews
;
Yunxin Y. Bo
;
Shon K. Booker
;
Sean Caenepeel
;
Victor J. Cee
;
Noel D. D鈥橝ngelo
;
Daniel J. Freeman
;
Bradley J. Herberich
;
Fang-Tsao Hong
;
Claire L. M. Jackson
;
Jian Jiang
;
Brian A. Lanman
;
Longbin Liu
;
John D. McCarter
;
Erin L. Mullady
;
Nobuko Nishimura
;
Liping H. Pettus
;
Anthony B. Reed
;
Tisha San Miguel
;
Adrian L. Smith
;
Markian M. Stec
;
Seifu Tadesse
;
Andrew Tasker
;
Divesh Aidasani
;
Xiaochun Zhu
;
Raju Subramanian
;
Nuria
A.
Tamayo
;
Ling Wang
;
Douglas A. Whittington
;
Bin Wu
;
Tian Wu
;
Ryan P. Wurz
;
Kevin Yang
;
Leeanne Zalameda
;
Nancy Zhang
;
Paul E. Hughes
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
Structure-Based Design of a Novel Series of Potent, Selective Inhibitors of the Class I Phosphatidylinositol 3-Kinases
作者:
Adrian L. Smith
;
Noel D. D鈥橝ngelo
;
Yunxin Y. Bo
;
Shon K. Booker
;
Victor J. Cee
;
Brad Herberich
;
Fang-Tsao Hong
;
Claire L. M. Jackson
;
Brian A. Lanman
;
Longbin Liu
;
Nobuko Nishimura
;
Liping H. Pettus
;
Anthony B. Reed
;
Seifu Tadesse
;
Nuria
A.
Tamayo
;
Ryan P. Wurz
;
Kevin Yang
;
Kristin L. Andrews
;
Douglas A. Whittington
;
John D. McCarter
;
Tisha San Miguel
;
Leeanne Zalameda
;
Jian Jiang
;
Raju Subramanian
;
Erin L. Mullady
;
Sean Caenepeel
;
Daniel J. Freeman
;
Ling Wang
;
Nancy Zhang
;
Tian Wu
;
Paul E. Hughes
;
Mark H. Norman
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
Correction to Selective Class I Phosphoinositide 3-Kinase Inhibitors: Optimization of a Series of Pyridyltriazines Leading to the Identification of a Clinical Candidate, AMG 511
作者:
Mark H. Norman
;
Kristin L. Andrews
;
Yunxin Y. Bo
;
Shon K. Booker
;
Sean Caenepeel
;
Victor J. Cee
;
Noel D. D鈥橝ngelo
;
Daniel J. Freeman
;
Bradley J. Herberich
;
Fang-Tsao Hong
;
Claire L. M. Jackson
;
Jian Jiang
;
Brian A. Lanman
;
Longbin Liu
;
John D. McCarter
;
Erin L. Mullady
;
Nobuko Nishimura
;
Liping H. Pettus
;
Anthony B. Reed
;
Tisha San Miguel
;
Adrian L. Smith
;
Markian M. Stec
;
Seifu Tadesse
;
Andrew Tasker
;
Divesh Aidasani
;
Xiaochun Zhu
;
Raju Subramanian
;
Nuria
A.
Tamayo
;
Ling Wang
;
Douglas A. Whittington
;
Bin Wu
;
Tian Wu
;
Ryan P. Wurz
;
Kevin Yang
;
Leeanne Zalameda
;
Nancy Zhang
;
Paul E. Hughes
刊名:Journal of Medicinal Chemistry
出版年:2012
9.
Structure鈥揂ctivity Relationships of Phosphoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors: Investigations of Various 6,5-Heterocycles to Improve Metabolic Stability
作者:
Markian M. Stec
;
Kristin L. Andrews
;
Shon K. Booker
;
Sean Caenepeel
;
Daniel J. Freeman
;
Jian Jiang
;
Hongyu Liao
;
John McCarter
;
Erin L. Mullady
;
Tisha San Miguel
;
Raju Subramanian
;
Nuria
Tamayo
;
Ling Wang
;
Kevin Yang
;
Leeanne P. Zalameda
;
Nancy Zhang
;
Paul E. Hughes
;
Mark H. Norman
刊名:Journal of Medicinal Chemistry
出版年:2011
10.
Phospshoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors: Discovery and Structure鈥揂ctivity Relationships of a Series of Quinoline and Quinoxaline Derivatives
作者:
Nobuko Nishimura
;
Aaron Siegmund
;
Longbin Liu
;
Kevin Yang
;
Marian C. Bryan
;
Kristin L. Andrews
;
Yunxin Bo
;
Shon K. Booker
;
Sean Caenepeel
;
Daniel Freeman
;
Hongyu Liao
;
John McCarter
;
Erin L. Mullady
;
Tisha San Miguel
;
Raju Subramanian
;
Nuria
Tamayo
;
Ling Wang
;
Douglas A. Whittington
;
Leeanne Zalameda
;
Nancy Zhang
;
Paul E. Hughes
;
Mark H. Norman
刊名:Journal of Medicinal Chemistry
出版年:2011
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