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内部出版物
在“
ACS电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
1.
Left-Hand Side Exploration of Novel Bacterial Topoisomerase Inhibitors to Improve Selectivity against hERG Binding
作者:
Shahul Hameed P
;
Praveena Manjrekar
;
Anandkumar Raichurkar
;
Vikas Shinde
;
Jayashree Puttur
;
Gajanan Shanbhag
;
Murugan Chinnapattu
;
Vikas Patil
;
Suresh Rudrapatana
;
Sreevalli Sharma
;
C. N. Naveen Kumar
;
Radha Nandishaiah
;
Prashanti
Madhavapeddi
;
D. Sriram
;
Suresh Solapure
;
Vasan K. Sambandamurthy
刊名:ACS Medicinal Chemistry Letters
出版年:2015
2.
Benzimidazoles: Novel Mycobacterial Gyrase Inhibitors from Scaffold Morphing
作者:
Shahul Hameed P
;
Anandkumar Raichurkar
;
Prashanti
Madhavapeddi
;
Sreenivasaiah Menasinakai
;
Sreevalli Sharma
;
Parvinder Kaur
;
Radha Nandishaiah
;
Vijender Panduga
;
Jitendar Reddy
;
Vasan K. Sambandamurthy
;
D. Sriram
刊名:ACS Medicinal Chemistry Letters
出版年:2014
3.
Novel N-Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis
作者:
Shahul Hameed P
;
Vikas Patil
;
Suresh Solapure
;
Umender Sharma
;
Prashanti
Madhavapeddi
;
Anandkumar Raichurkar
;
Murugan Chinnapattu
;
Praveena Manjrekar
;
Gajanan Shanbhag
;
Jayashree Puttur
;
Vikas Shinde
;
Sreenivasaiah Menasinakai
;
Suresh Rudrapatana
;
Vijayashree Achar
;
Disha Awasthy
;
Radha Nandishaiah
;
Vaishali Humnabadkar
;
Anirban Ghosh
;
Chandan Narayan
;
V. K. Ramya
;
Parvinder Kaur
;
Sreevalli Sharma
;
Jim Werngren
;
Sven Hoffner
;
Vijender Panduga
;
C. N. Naveen Kumar
;
Jitendar Reddy
;
Mahesh Kumar KN
;
Samit Ganguly
;
Sowmya Bharath
;
Ugarkar Bheemarao
;
Kakoli Mukherjee
;
Uma Arora
;
Sheshagiri Gaonkar
;
Michelle Coulson
;
David Waterson
;
Vasan K. Sambandamurthy
;
Sunita M. de Sousa
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity
作者:
Maruti Naik
;
Vaishali Humnabadkar
;
Subramanyam J. Tantry
;
Manoranjan Panda
;
Ashwini Narayan
;
Supreeth Guptha
;
Vijender Panduga
;
Praveena Manjrekar
;
Lalit kumar Jena
;
Krishna Koushik
;
Gajanan Shanbhag
;
Sandesh Jatheendranath
;
M. R. Manjunatha
;
Gopinath Gorai
;
Chandramohan Bathula
;
Suresh Rudrapatna
;
Vijayashree Achar
;
Sreevalli Sharma
;
Anisha Ambady
;
Naina Hegde
;
Jyothi Mahadevaswamy
;
Parvinder Kaur
;
Vasan K. Sambandamurthy
;
Disha Awasthy
;
Chandan Narayan
;
Sudha Ravishankar
;
Prashanti
Madhavapeddi
;
Jitendar Reddy
;
KR Prabhakar
;
Ramanatha Saralaya
;
Monalisa Chatterji
;
James Whiteaker
;
Bob McLaughlin
;
Laurent R. Chiarelli
;
Giovanna Riccardi
;
Maria Rosalia Pasca
;
Claudia Binda
;
Jo茫o Neres
;
Neeraj Dhar
;
Fran莽ois Signorino-Gelo
;
John D. McKinney
;
Vasanthi Ramachandran
;
Radha Shandil
;
Ruben Tommasi
;
Pravin S. Iyer
;
Shridhar Narayanan
;
Vinayak Hosagrahara
;
Stefan Kavanagh
;
Neela Dinesh
;
Sandeep R. Ghorpade
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Thiazolopyridine Ureas as Novel Antitubercular Agents Acting through Inhibition of DNA Gyrase B
作者:
Manoj G. Kale
;
Anandkumar Raichurkar
;
Shahul Hameed P
;
David Waterson
;
David McKinney
;
M. R. Manjunatha
;
Usha Kranthi
;
Krishna Koushik
;
Lalit kumar Jena
;
Vikas Shinde
;
Suresh Rudrapatna
;
Shubhada Barde
;
Vaishali Humnabadkar
;
Prashanti
Madhavapeddi
;
Halesha Basavarajappa
;
Anirban Ghosh
;
VK Ramya
;
Supreeth Guptha
;
Sreevalli Sharma
;
Prakash Vachaspati
;
K.N. Mahesh Kumar
;
Jayashree Giridhar
;
Jitendar Reddy
;
Vijender Panduga
;
Samit Ganguly
;
Vijaykamal Ahuja
;
Sheshagiri Gaonkar
;
C. N. Naveen Kumar
;
Derek Ogg
;
Julie A. Tucker
;
P. Ann Boriack-Sjodin
;
Sunita M. de Sousa
;
Vasan K. Sambandamurthy
;
Sandeep R. Ghorpade
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Methyl-Thiazoles: A Novel Mode of Inhibition with the Potential to Develop Novel Inhibitors Targeting InhA in Mycobacterium tuberculosis
作者:
Pravin S. Shirude
;
Prashanti
Madhavapeddi
;
Maruti Naik
;
Kannan Murugan
;
Vikas Shinde
;
Radha Nandishaiah
;
Jyothi Bhat
;
Anupriya Kumar
;
Shahul Hameed
;
Geoffrey Holdgate
;
Gareth Davies
;
Helen McMiken
;
Naina Hegde
;
Anisha Ambady
;
Janani Venkatraman
;
Manoranjan Panda
;
Balachandra Bandodkar
;
Vasan K. Sambandamurthy
;
Jon A. Read
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo
作者:
Pravin S. Shirude
;
Radha Shandil
;
Claire Sadler
;
Maruti Naik
;
Vinayak Hosagrahara
;
Shahul Hameed
;
Vikas Shinde
;
Chandramohan Bathula
;
Vaishali Humnabadkar
;
Naveen Kumar
;
Jitendar Reddy
;
Vijender Panduga
;
Sreevalli Sharma
;
Anisha Ambady
;
Naina Hegde
;
James Whiteaker
;
Robert E. McLaughlin
;
Humphrey Gardner
;
Prashanti
Madhavapeddi
;
Vasanthi Ramachandran
;
Parvinder Kaur
;
Ashwini Narayan
;
Supreeth Guptha
;
Disha Awasthy
;
Chandan Narayan
;
Jyothi Mahadevaswamy
;
KG Vishwas
;
Vijaykamal Ahuja
;
Abhishek Srivastava
;
KR Prabhakar
;
Sowmya Bharath
;
Ramesh Kale
;
Manjunatha Ramaiah
;
Nilanjana Roy Choudhury
;
Vasan K. Sambandamurthy
;
Suresh Solapure
;
Pravin S. Iyer
;
Shridhar Narayanan
;
Monalisa Chatterji
刊名:Journal of Medicinal Chemistry
出版年:2013
8.
Aminopyrazinamides: Novel and Specific GyrB Inhibitors that Kill Replicating and Nonreplicating Mycobacterium tuberculosis
作者:
Pravin S. Shirude
;
Prashanti
Madhavapeddi
;
Julie A. Tucker
;
Kannan Murugan
;
Vikas Patil
;
Halesha Basavarajappa
;
Anandkumar V. Raichurkar
;
Vaishali Humnabadkar
;
Syeed Hussein
;
Sreevalli Sharma
;
V. K. Ramya
;
Chandan B. Narayan
;
Tanjore S. Balganesh
;
Vasan K. Sambandamurthy
刊名:ACS Chemical Biology
出版年:2013
9.
Pre-Steady-State Kinetic Studies on the Glu171Gln Active Site Mutant of Adenosylcobalamin-Dependent Glutamate Mutase
作者:
Prashanti
Madhavapeddi
;
David P. Ballou
;
and E. Neil G. Marsh
刊名:Biochemistry
出版年:2002
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