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CNKI学位论文(8)
知网期刊论文(3)
在“
ACS电子期刊
”中,
命中:
14
条,耗时:小于0.01 秒
在所有数据库中总计命中:
11
条
1.
Lead Optimization of 2-Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of Gliomas
作者:
Simona Daniele
;
Valeria
La
Pietra
;
Elisabetta Barresi
;
Salvatore Di Maro
;
Eleonora Da Pozzo
;
Marco Robello
;
Concettina
La
Motta
;
Sandro Cosconati
;
Sabrina Taliani
;
Luciana Marinelli
;
Ettore Novellino
;
C
la
udia Martini
;
Federico Da Settimo
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Exploring the N-Terminal Region of C-X-C Motif Chemokine 12 (CXCL12): Identification of P
la
sma-Stable Cyclic Peptides As Novel, Potent C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonists
作者:
Salvatore Di Maro
;
Anna Maria Trotta
;
Diego Brancaccio
;
Francesco Saverio Di Leva
;
Valeria
La
Pietra
;
Caterina Ieranò
;
Maria Napolitano
;
Luigi Portel
la
;
Crescenzo D’Alterio
;
Rosa Anna Siciliano
;
Deborah Sementa
;
Stefano Tomassi
;
Alfonso Carotenuto
;
Ettore Novellino
;
Stefania Sca
la
;
Luciana Marinelli
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Structure-Based Lead Optimization and Biological Evaluation of BAX Direct Activators as Novel Potential Anticancer Agents
作者:
Mariano Stornaiuolo
;
Giuseppe
La
Regina
;
Sara Passacantilli
;
Gianluca Grassia
;
Antonio Coluccia
;
Valeria
La
Pietra
;
Mariateresa Giustiniano
;
Hilde Cassese
;
Salvatore Di Maro
;
Diego Brancaccio
;
Sabrina Taliani
;
Armando Ialenti
;
Romano Silvestri
;
C
la
udia Martini
;
Ettore Novellino
;
Luciana Marinelli
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
A Novel Cell-Permeable, Selective, and Noncompetitive Inhibitor of KAT3 Histone Acetyltransferases from a Combined Molecu
la
r Pruning/C
la
ssical Isosterism Approach
作者:
Ciro Milite
;
Alessandra Feoli
;
Kazuki Sasaki
;
Valeria
La
Pietra
;
Amodio Luca Balzano
;
Luciana Marinelli
;
Antonello Mai
;
Ettore Novellino
;
Sabrina Castel
la
no
;
Alessandra Tosco
;
Gianluca Sbardel
la
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Structure-Based Optimization of Tyrosine Kinase Inhibitor CLM3. Design, Synthesis, Functional Evaluation, and Molecu
la
r Modeling Studies.
作者:
Stefania Sartini
;
Vito Coviello
;
Agostino Bruno
;
Valeria
La
Pietra
;
Luciana Marinelli
;
Francesca Simorini
;
Sabrina Taliani
;
Silvia Salerno
;
Anna Maria Marini
;
Anna Fioravanti
;
Pao
la
Or
la
ndi
;
Alessandro Antonelli
;
Federico Da Settimo
;
Ettore Novellino
;
Guido Bocci
;
Concettina
La
Motta
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
p53 Functional Inhibitors Behaving Like Pifithrin-尾 Counteract the Alzheimer Peptide Non-尾-amyloid Component Effects in Human SH-SY5Y Cells
作者:
Eleonora Da Pozzo
;
Valeria
La
Pietra
;
Barbara Cosimelli
;
Federico Da Settimo
;
Chiara Giacomelli
;
Luciana Marinelli
;
C
la
udia Martini
;
Ettore Novellino
;
Sabrina Taliani
;
Giovanni Greco
刊名:ACS Chemical Neuroscience
出版年:2014
7.
Discovery of Covalent Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase, A Target for the Treatment of Ma
la
ria
作者:
Stefano Bruno
;
Andrea Pinto
;
Gianluca Paredi
;
Lucia Tamborini
;
Carlo De Micheli
;
Valeria
La
Pietra
;
Luciana Marinelli
;
Ettore Novellino
;
Pao
la
Conti
;
Andrea Mozzarelli
刊名:Journal of Medicinal Chemistry
出版年:2014
8.
Design, Synthesis, and Biological Evaluation of 1-Phenylpyrazolo[3,4-e]pyrrolo[3,4-g]indolizine-4,6(1H,5H)-diones as New Glycogen Synthase Kinase-3β Inhibitors
作者:
Valeria
La
Pietra
;
Giuseppe
La
Regina
;
Antonio Coluccia
;
Valeria
Famiglini
;
Sveva Pelliccia
;
Batya Plotkin
;
Hagit Eldar-Finkelman
;
Andrea Brancale
;
Carlo Bal
la
tore
;
Alex Crowe
;
Kurt R. Brunden
;
Luciana Marinelli
;
Ettore Novellino
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2013
9.
Selective Arylsulfonamide Inhibitors of ADAM-17: Hit Optimization and Activity in Ovarian Cancer Cell Models
作者:
Elisa Nuti
;
Francesca Casalini
;
Salvatore Santamaria
;
Marina Fabbi
;
Grazia Carbotti
;
Silvano Ferrini
;
Luciana Marinelli
;
Valeria
La
Pietra
;
Ettore Novellino
;
Caterina Camodeca
;
Elisabetta Or
la
ndini
;
Susanna Nencetti
;
Armando Rossello
刊名:Journal of Medicinal Chemistry
出版年:2013
10.
Protein Flexibility in Virtual Screening: The BACE-1 Case Study
作者:
Sandro Cosconati
;
Luciana Marinelli
;
Francesco Saverio Di Leva
;
Valeria
La
Pietra
;
Ange
la
De Simone
;
Francesca Mancini
;
Vincenza Andrisano
;
Ettore Novellino
;
David S. Goodsell
;
Arthur J. Olson
刊名:Journal of Chemical Information and Modeling
出版年:2012
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