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知网期刊论文(423)
在“
ACS电子期刊
”中,
命中:
38
条,耗时:0.0789269 秒
在所有数据库中总计命中:
2,711
条
1.
Fragment-Based Discovery of a Selective
and
Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637)
作者:
Alex
and
er M. Taylor
;
Alex
and
re Côté
;
Michael C. Hewitt
;
Richard
Pastor
;
Yves Leblanc
;
Christopher G. Nasveschuk
;
F. Anthony Romero
;
Terry D. Crawford
;
Nico Cantone
;
Hariharan Jayaram
;
Jeremy Setser
;
Jeremy Murray
;
Maureen H. Beresini
;
Gladys de Leon Boenig
;
Zhongguo Chen
;
And
rew R. Conery
;
Richard
T.
Cummings
;
Leslie A. Dakin
;
E. Megan Flynn
;
Oscar W. Huang
;
Susan Kaufman
;
Patricia J. Keller
;
James R. Kiefer
;
Tommy Lai
;
Yingjie Li
;
Jiangpeng Liao
;
Wenfeng Liu
;
Henry Lu
;
Eneida Pardo
;
Vickie Tsui
;
Jian Wang
;
Yongyun Wang
;
Zhaowu Xu
;
Fen Yan
;
Dong Yu
;
Laura Zawadzke
;
Xiaoqin Zhu
;
Xiaoyu Zhu
;
Robert J. Sims III
;
And
rea G. Cochran
;
Steve Bellon
;
James E. Audia
;
Steven Magnuson
;
Brian K. Albrecht
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9,
and
CECR2 Bromodomains
作者:
Terry D. Crawford
;
Vickie Tsui
;
E. Megan Flynn
;
Shumei Wang
;
Alex
and
er M. Taylor
;
Alex
and
re Côté
;
James E. Audia
;
Maureen H. Beresini
;
Daniel J. Burdick
;
Richard
Cummings
;
Les A. Dakin
;
Martin Duplessis
;
And
rew C. Good
;
Michael C. Hewitt
;
Hon-Ren Huang
;
Hariharan Jayaram
;
James R. Kiefer
;
Ying Jiang
;
Jeremy Murray
;
Christopher G. Nasveschuk
;
Eneida Pardo
;
Florence Poy
;
F. Anthony Romero
;
Yong Tang
;
Jian Wang
;
Zhaowu Xu
;
Laura E. Zawadzke
;
Xiaoyu Zhu
;
Brian K. Albrecht
;
Steven R. Magnuson
;
Steve Bellon
;
And
rea G. Cochran
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery of a Potent
and
Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300
作者:
Terry D. Crawford
;
F. Anthony Romero
;
Kwong Wah Lai
;
Vickie Tsui
;
Alex
and
er M. Taylor
;
Gladys de Leon Boenig
;
Cameron L. Nol
and
;
Jeremy Murray
;
Justin Ly
;
Edna F. Choo
;
Thomas L. Hunsaker
;
Emily W. Chan
;
Mark Merchant
;
Samir Kharb
and
a
;
Karen E. Gascoigne
;
Susan Kaufman
;
Maureen H. Beresini
;
Jiangpeng Liao
;
Wenfeng Liu
;
Kevin X. Chen
;
Zhongguo Chen
;
And
rew R. Conery
;
Alex
and
re Côté
;
Hariharan Jayaram
;
Ying Jiang
;
James R. Kiefer
;
Tracy Kleinheinz
;
Yingjie Li
;
Jonathan Maher
;
Eneida Pardo
;
Florence Poy
;
Kerry L. Spillane
;
Fei Wang
;
Jian Wang
;
Xiaocang Wei
;
Zhaowu Xu
;
Zhongya Xu
;
Ivana Yen
;
Laura Zawadzke
;
Xiaoyu Zhu
;
Steven Bellon
;
Richard
Cummings
;
And
rea G. Cochran
;
Brian K. Albrecht
;
Steven Magnuson
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent
and
Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymp
作者:
Rishi G. Vaswani
;
Victor S. Gehling
;
Les A. Dakin
;
And
rew S. Cook
;
Christopher G. Nasveschuk
;
Martin Duplessis
;
Priyadarshini Iyer
;
Srividya Balasubramanian
;
Feng Zhao
;
And
rew C. Good
;
Robert Campbell
;
Christina Lee
;
Nico Cantone
;
Richard
T.
Cummings
;
Emmanuel Normant
;
Steven F. Bellon
;
Brian K. Albrecht
;
Jean-Christophe Harmange
;
Patrick Trojer
;
James E. Audia
;
Ying Zhang
;
Neil Justin
;
Shuyang Chen
;
Jon R. Wilson
;
Steven J. Gamblin
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain
and
Extra-Terminal (BET) Family as a C
and
idate for Human Clinical Trials
作者:
Brian K. Albrecht
;
Victor S. Gehling
;
Michael C. Hewitt
;
Rishi G. Vaswani
;
Alex
and
re Côté
;
Yves Leblanc
;
Christopher G. Nasveschuk
;
Steve Bellon
;
Louise Bergeron
;
Robert Campbell
;
Nico Cantone
;
Michael R. Cooper
;
Richard
T.
Cummings
;
Hariharan Jayaram
;
Shivangi Joshi
;
Jennifer A. Mertz
;
Adrianne Neiss
;
Emmanuel Normant
;
Michael O’Meara
;
Eneida Pardo
;
Florence Poy
;
Peter S
and
y
;
Jeffrey Supko
;
Robert J. Sims III
;
Jean-Christophe Harmange
;
Alex
and
er M. Taylor
;
James E. Audia
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Discovery of Benzotriazolo[4,3-d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains
作者:
Alex
and
er M. Taylor
;
Rishi G. Vaswani
;
Victor S. Gehling
;
Michael C. Hewitt
;
Yves Leblanc
;
James E. Audia
;
Steve Bellon
;
Richard
T.
Cummings
;
Alex
and
re C?té
;
Jean-Christophe Harmange
;
Hari Jayaram
;
Shivangi Joshi
;
Jose M. Lora
;
Jennifer A. Mertz
;
Adrianne Neiss
;
Eneida Pardo
;
Christopher G. Nasveschuk
;
Florence Poy
;
Peter S
and
y
;
Jeremy W. Setser
;
Robert J. Sims III
;
Yong Tang
;
Brian K. Albrecht
刊名:ACS Medicinal Chemistry Letters
出版年:2016
7.
Thiolactomycin-Based Inhibitors of Bacterial β-Ketoacyl-ACP Synthases with in Vivo Activity
作者:
Gopal R. Bommineni
;
Kanishk Kapilashrami
;
Jason E.
Cummings
;
Yang Lu
;
Susan E. Knudson
;
Chendi Gu
;
Stephen G. Walker
;
Richard
A. Slayden
;
Peter J. Tonge
刊名:Journal of Medicinal Chemistry
出版年:2016
8.
Dramatically Increased pH
and
Temperature Stability of Chymotrypsin Using Dual Block Polymer-Based Protein Engineering
作者:
Chad
Cummings
;
Hironobu Murata
;
Richard
Koepsel
;
Alan J. Russell
刊名:Biomacromolecules
出版年:2014
9.
Rational Tailoring of Substrate
and
Inhibitor Affinity via ATRP Polymer-Based Protein Engineering
作者:
Hironobu Murata
;
Chad S.
Cummings
;
Richard
R. Koepsel
;
Alan J. Russell
刊名:Biomacromolecules
出版年:2014
10.
Discovery
and
Optimization of Tetramethylpiperidinyl Benzamides as Inhibitors of EZH2
作者:
Christopher G. Nasveschuk
;
Alex
and
re Gagnon
;
Shivani Garapaty-Rao
;
Srividya Balasubramanian
;
Robert Campbell
;
Christina Lee
;
Feng Zhao
;
Louise Bergeron
;
Richard
Cummings
;
Patrick Trojer
;
James E. Audia
;
Brian K. Albrecht
;
Jean-Christophe P. Harmange
刊名:ACS Medicinal Chemistry Letters
出版年:2014
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