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在“
ACS电子期刊
”中,
命中:
5
条,耗时:0.0189648 秒
在所有数据库中总计命中:
5
条
1.
Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein–Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery
作者:
Thomas G. Davies
;
William E. Wixted
;
J
oseph E. Coyle
;
Charlotte Griffiths-
J
ones
;
Keisha Hearn
;
Rachel McMenamin
;
David Norton
;
Sharna
J
. Rich
;
Caroline Richardson
;
Gordon Saxty
;
Henriëtte M. G. Willems
;
Alison
J
.-A.
Woolford
;
J
oshua E. Cottom
;
J
en-Pyng Kou
;
J
ohn G. Yonchuk
;
Heidi G. Feldser
;
Yolanda Sanchez
;
J
oseph P. Foley
;
Brian
J
. Bolognese
;
Gregory Logan
;
Patricia L. Podolin
;
Hongxing Yan
;
J
ames F. Callahan
;
Tom D. Heightman
;
J
effrey K. Kerns
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
2.
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening
作者:
Alison
J
.-A.
Woolford
;
J
oseph E. Pero
;
Sridhar Aravapalli
;
Valerio Berdini
;
J
oseph E. Coyle
;
Philip
J
. Day
;
Andrew M. Dodson
;
Pascal Grondin
;
Finn P. Holding
;
Lydia Y. W. Lee
;
Peng Li
;
Eric S. Manas
;
J
oseph Marino Jr.
;
Agnes C. L. Martin
;
Brent W. McCleland
;
Rachel L. McMenamin
;
Christopher W. Murray
;
Christopher E. Neipp
;
Lee W. Page
;
Vipulkumar K. Patel
;
Florent Potvain
;
Sharna Rich
;
Ralph A. Rivero
;
Kirsten Smith
;
Donald O. Somers
;
Lionel Trottet
;
Ranganadh Velagaleti
;
Glyn Williams
;
Ren Xie
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
3.
Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)
作者:
Alison
J
.-A.
Woolford
;
Philip
J
. Day
;
Véronique Bénéton
;
Valerio Berdini
;
J
oseph E. Coyle
;
Yann Dudit
;
Pascal Grondin
;
Pascal Huet
;
Lydia Y. W. Lee
;
Eric S. Manas
;
Rachel L. McMenamin
;
Christopher W. Murray
;
Lee W. Page
;
Vipulkumar K. Patel
;
Florent Potvain
;
Sharna
J
. Rich
;
Yingxia Sang
;
Don O. Somers
;
Lionel Trottet
;
Zehong Wan
;
Xiaomin Zhang
刊名:
J
ournal of Medicinal Chemistry
出版年:2016
4.
Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Discovery of a Non-Alanine Lead Series with Dual Activity Against cIAP1 and XIAP
作者:
Gianni Chessari
;
Ildiko M. Buck
;
J
ames E. H. Day
;
Philip
J
. Day
;
Aman Iqbal
;
Christopher N.
J
ohnson
;
Edward
J
. Lewis
;
Vanessa Martins
;
Darcey Miller
;
Michael Reader
;
David C. Rees
;
Sharna
J
. Rich
;
Emiliano Tamanini
;
Marc Vitorino
;
George A. Ward
;
Pamela A. Williams
;
Glyn Williams
;
Nicola E. Wilsher
;
Alison
J
.-A.
Woolford
刊名:
J
ournal of Medicinal Chemistry
出版年:2015
5.
Fragment-Based Discovery of 7-Azabenzimidazoles as Potent, Highly Selective, and Orally Active CDK4/6 Inhibitors
作者:
Young Shin Cho
;
Hayley Angove
;
Christopher Brain
;
Christine Hiu-Tung Chen
;
Hong Cheng
;
Robert Cheng
;
Ra
j
iv Chopra
;
Kristy Chung
;
Miles Congreve
;
Claudio Dagostin
;
Deborah
J
. Davis
;
Ruth Feltell
;
J
ohn Giraldes
;
Steven D. Hiscock
;
Sunkyu Kim
;
Steven Kovats
;
Bharat Lagu
;
Kim Lewry
;
Alice Loo
;
Yipin Lu
;
Michael Luzzio
;
Wiesia Maniara
;
Rachel McMenamin
;
Paul N. Mortenson
;
Ra
j
deep Benning
;
Marc O'Reilly
;
David C. Rees
;
J
unqing Shen
;
Troy Smith
;
Yaping Wang
;
Glyn Williams
;
Alison
J
.-A.
Woolford
;
Wo
j
ciech Wrona
;
Mei Xu
;
Fan Yang
;
Steven Howard
刊名:ACS Medicinal Chemistry Letters
出版年:2012
1
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