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在“
ACS电子期刊
”中,
命中:
17
条,耗时:小于0.01 秒
在所有数据库中总计命中:
3
条
1.
Discovery of Benzotriazolo[4,3-d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains
作者:
Alexander M. Taylor
;
Rishi G. Vaswani
;
Victor S. Gehling
;
Michael C. Hewitt
;
Yves Leblanc
;
James E. Audia
;
Steve Bellon
;
Richard T. Cummings
;
Alexandre C?té
;
Jean
-
Christophe
Harmange
;
Hari Jayaram
;
Shivangi Joshi
;
Jose M. Lora
;
Jennifer A. Mertz
;
Adrianne Neiss
;
Eneida Pardo
;
Christophe
r G. Nasveschuk
;
Florence Poy
;
Peter Sandy
;
Jeremy W. Setser
;
Robert J. Sims III
;
Yong Tang
;
Brian K. Albrecht
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials
作者:
Brian K. Albrecht
;
Victor S. Gehling
;
Michael C. Hewitt
;
Rishi G. Vaswani
;
Alexandre Côté
;
Yves Leblanc
;
Christophe
r G. Nasveschuk
;
Steve Bellon
;
Louise Bergeron
;
Robert Campbell
;
Nico Cantone
;
Michael R. Cooper
;
Richard T. Cummings
;
Hariharan Jayaram
;
Shivangi Joshi
;
Jennifer A. Mertz
;
Adrianne Neiss
;
Emmanuel Normant
;
Michael O’Meara
;
Eneida Pardo
;
Florence Poy
;
Peter Sandy
;
Jeffrey Supko
;
Robert J. Sims III
;
Jean
-
Christophe
Harmange
;
Alexander M. Taylor
;
James E. Audia
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymp
作者:
Rishi G. Vaswani
;
Victor S. Gehling
;
Les A. Dakin
;
Andrew S. Cook
;
Christophe
r G. Nasveschuk
;
Martin Duplessis
;
Priyadarshini Iyer
;
Srividya Balasubramanian
;
Feng Zhao
;
Andrew C. Good
;
Robert Campbell
;
Christina Lee
;
Nico Cantone
;
Richard T. Cummings
;
Emmanuel Normant
;
Steven F. Bellon
;
Brian K. Albrecht
;
Jean
-
Christophe
Harmange
;
Patrick Trojer
;
James E. Audia
;
Ying Zhang
;
Neil Justin
;
Shuyang Chen
;
Jon R. Wilson
;
Steven J. Gamblin
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery of (R)-6-(1-(8-Fluoro-6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl)-3-(2-methoxyethoxy)-1,6-naphthyridin-5(6H)-one (AMG 337), a Potent and Selective Inhibitor of MET with High Unbound Target Coverage and Robust In Vivo A
作者:
Alessandro A. Boezio
;
Katrina W. Copeland
;
Karen Rex
;
Brian K. Albrecht
;
David Bauer
;
Steven F. Bellon
;
Christiane Boezio
;
Martin A. Broome
;
Deborah Choquette
;
Angela Coxon
;
Isabelle Dussault
;
Satoko Hirai
;
Richard Lewis
;
Min-Hwa Jasmine Lin
;
Julia Lohman
;
Jingzhou Liu
;
Emily A. Peterson
;
Michele Potashman
;
Roman Shimanovich
;
Yohannes Teffera
;
Douglas A. Whittington
;
Karina R. Vaida
;
Jean
-
Christophe
Harmange
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Correction to Discovery of Potent and Selective 8-Fluorotriazolopyridine c-Met Inhibitors
作者:
Emily A. Peterson
;
Yohannes Teffera
;
Brian K. Albrecht
;
David Bauer
;
Steven F. Bellon
;
Alessandro Boezio
;
Christiane Boezio
;
Martin A. Broome
;
Deborah Choquette
;
Katrina W. Copeland
;
Isabelle Dussault
;
Richard Lewis
;
Min-Hwa Jasmine Lin
;
Julia Lohman
;
Jingzhou Liu
;
Michele Potashman
;
Karen Rex
;
Roman Shimanovich
;
Douglas A. Whittington
;
Karina R. Vaida
;
Jean
-
Christophe
Harmange
刊名:Journal of Medicinal Chemistry
出版年:2015
6.
Discovery and Optimization of Tetramethylpiperidinyl Benzamides as Inhibitors of EZH2
作者:
Christophe
r G. Nasveschuk
;
Alexandre Gagnon
;
Shivani Garapaty-Rao
;
Srividya Balasubramanian
;
Robert Campbell
;
Christina Lee
;
Feng Zhao
;
Louise Bergeron
;
Richard Cummings
;
Patrick Trojer
;
James E. Audia
;
Brian K. Albrecht
;
Jean
-
Christophe
P.
Harmange
刊名:ACS Medicinal Chemistry Letters
出版年:2014
7.
A Practical Synthesis of Indoles via a Pd-Catalyzed C鈥揘 Ring Formation
作者:
Rishi G. Vaswani
;
Brian K. Albrecht
;
James E. Audia
;
Alexandre C么t茅
;
Les A. Dakin
;
Martin Duplessis
;
Victor S. Gehling
;
Jean
-
Christophe
Harmange
;
Michael C. Hewitt
;
Yves Leblanc
;
Christophe
r G. Nasveschuk
;
Alexander M. Taylor
刊名:Organic Letters
出版年:2014
8.
Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors
作者:
Victor S. Gehling
;
Michael C. Hewitt
;
Rishi G. Vaswani
;
Yves Leblanc
;
Alexandre C么t茅
;
Christophe
r G. Nasveschuk
;
Alexander M. Taylor
;
Jean
-
Christophe
Harmange
;
James E. Audia
;
Eneida Pardo
;
Shivangi Joshi
;
Peter Sandy
;
Jennifer A. Mertz
;
Robert J. Sims
;
III
;
Louise Bergeron
;
Barbara M. Bryant
;
Steve Bellon
;
Florence Poy
;
Hariharan Jayaram
;
Ravichandran Sankaranarayanan
;
Sreegouri Yellapantula
;
Nandana Bangalore Srinivasamurthy
;
Swarnakumari Birudukota
;
Brian K. Albrecht
刊名:ACS Medicinal Chemistry Letters
出版年:2013
9.
Structure-Based Design of Novel Class II c-Met Inhibitors: 2. SAR and Kinase Selectivity Profiles of the Pyrazolone Series
作者:
Longbin Liu
;
Mark H. Norman
;
Matthew Lee
;
Ning Xi
;
Aaron Siegmund
;
Alessandro A. Boezio
;
Shon Booker
;
Debbie Choquette
;
Noel D. D鈥橝ngelo
;
Julie Germain
;
Kevin Yang
;
Yajing Yang
;
Yihong Zhang
;
Steven F. Bellon
;
Douglas A. Whittington
;
Jean
-
Christophe
Harmange
;
Celia Dominguez
;
Tae-Seong Kim
;
Isabelle Dussault
刊名:Journal of Medicinal Chemistry
出版年:2012
10.
Chemical Reactivity of Methoxy 4-O-Aryl Quinolines: Identification of Glutathione Displacement Products in Vitro and in Vivo
作者:
Yohannes Teffera
;
Adria E. Colletti
;
Jean
Christophe
Harmange
;
L. Steven Hollis
;
Brian K. Albrecht
;
Alessandro A. Boezio
;
Jingzhou Liu
;
Zhiyang Zhao
刊名:Chemical Research in Toxicology
出版年:2008
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