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CNKI学位论文(41)
知网期刊论文(6)
在“
ACS电子期刊
”中,
命中:
14
条,耗时:小于0.01 秒
在所有数据库中总计命中:
47
条
1.
N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase
作者:
Luca Pescatori
;
Mathieu M茅tifiot
;
Suhman Chung
;
Takashi Masoaka
;
Giuliana Cuzzucoli Crucitti
;
Antonella Messore
;
Giovanni Pupo
;
Valentina Noemi Madia
;
Francesco Saccoliti
;
Luigi Scipione
;
Silvano Tortorella
;
Francesco Saverio Di Leva
;
Sandro Cosconati
;
Luciana Marinelli
;
Ettore Novellino
;
Stuart F. J. Le Grice
;
Yves Pommier
;
Christophe Marchand
;
Roberta
Costi
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2015
2.
Structure鈥揂ctivity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain
作者:
Giuliana Cuzzucoli Crucitti
;
Mathieu M茅tifiot
;
Luca Pescatori
;
Antonella Messore
;
Valentina Noemi Madia
;
Giovanni Pupo
;
Francesco Saccoliti
;
Luigi Scipione
;
Silvano Tortorella
;
Francesca Esposito
;
Angela Corona
;
Marta Cadeddu
;
Christophe Marchand
;
Yves Pommier
;
Enzo Tramontano
;
Roberta
Costi
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2015
3.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
作者:
Roberta
Costi
;
Mathieu M茅tifiot
;
Suhman Chung
;
Giuliana Cuzzucoli Crucitti
;
Kasthuraiah Maddali
;
Luca Pescatori
;
Antonella Messore
;
Valentina Noemi Madia
;
Giovanni Pupo
;
Luigi Scipione
;
Silvano Tortorella
;
Francesco Saverio Di Leva
;
Sandro Cosconati
;
Luciana Marinelli
;
Ettore Novellino
;
Stuart F. J. Le Grice
;
Angela Corona
;
Yves Pommier
;
Christophe Marchand
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi
作者:
Laura Friggeri
;
Luigi Scipione
;
Roberta
Costi
;
Marcel Kaiser
;
Francesca Moraca
;
Claudio Zamperini
;
Bruno Botta
;
Roberto Di Santo
;
Daniela De Vita
;
Reto Brun
;
Silvano Tortorella
刊名:ACS Medicinal Chemistry Letters
出版年:2013
5.
Pharmacophore Assessment Through 3-D QSAR: Evaluation of the Predictive Ability on New Derivatives by the Application on a Series of Antitubercular Agents
作者:
Laura Friggeri
;
Flavio Ballante
;
Rino Ragno
;
Ira Musmuca
;
Daniela De Vita
;
Fabrizio Manetti
;
Mariangela Biava
;
Luigi Scipione
;
Roberto Di Santo
;
Roberta
Costi
;
Marta Feroci
;
Silvano Tortorella
刊名:Journal of Chemical Information and Modeling
出版年:2013
6.
New Nucleotide-Competitive Non-Nucleoside Inhibitors of Terminal Deoxynucleotidyl Transferase: Discovery, Characterization, and Crystal Structure in Complex with the Target
作者:
Roberta
Costi
;
Giuliana Cuzzucoli Crucitti
;
Luca Pescatori
;
Antonella Messore
;
Luigi Scipione
;
Silvano Tortorella
;
Alessandra Amoroso
;
Emmanuele Crespan
;
Pietro Campiglia
;
Bruno Maresca
;
Amalia Porta
;
Ilaria Granata
;
Ettore Novellino
;
J茅r么me Gouge
;
Marc Delarue
;
Giovanni Maga
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic Acids as Dual Inhibitors of Recombinant HIV-1 Integrase and Ribonuclease H, Synthesized by a Parallel Synthesis Approach
作者:
Roberta
Costi
;
Mathieu M茅tifiot
;
Francesca Esposito
;
Giuliana Cuzzucoli Crucitti
;
Luca Pescatori
;
Antonella Messore
;
Luigi Scipione
;
Silvano Tortorella
;
Luca Zinzula
;
Ettore Novellino
;
Yves Pommier
;
Enzo Tramontano
;
Christophe Marchand
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2013
8.
Design, Synthesis, and Structure鈥揂ctivity Relationship of N-Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors
作者:
Roberto Di Santo
;
Roberta
Costi
;
Giuliana Cuzzucoli Crucitti
;
Luca Pescatori
;
Federica Rosi
;
Luigi Scipione
;
Diana Celona
;
Mario Vertechy
;
Orlando Ghirardi
;
Paola Piovesan
;
Mauro Marzi
;
Silvio Caccia
;
Giovanna Guiso
;
Fabrizio Giorgi
;
Patrizia Minetti
刊名:Journal of Medicinal Chemistry
出版年:2012
9.
Discovery and Pharmacological Profile of New 1H-Indazole-3-carboxamide and 2H-Pyrrolo[3,4-c]quinoline Derivatives as Selective Serotonin 4 Receptor Ligands
作者:
Guido Furlotti
;
Maria Alessandra Alisi
;
Claudia Apicella
;
Alessandra Capezzone de Joannon
;
Nicola Cazzolla
;
Roberta
Costi
;
Giuliana Cuzzucoli Crucitti
;
Beatrice Garrone
;
Alberto Iacovo
;
Gabriele Magar貌
;
Giorgina Mangano
;
Gaetano Miele
;
Rosella Ombrato
;
Luca Pescatori
;
Lorenzo Polenzani
;
Federica Rosi
;
Marco Vitiello
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2012
10.
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-Associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity
作者:
Donghang Cheng
;
Sergio Valente
;
Sabrina Castellano
;
Gianluca Sbardella
;
Roberto Di Santo
;
Roberta
Costi
;
Mark T. Bedford
;
Antonello Mai
刊名:Journal of Medicinal Chemistry
出版年:2011
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