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内部出版物
在“
ACS电子期刊
”中,
命中:
36
条,耗时:小于0.01 秒
1.
Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma
作者:
Daniela Vullo
;
Mariaconcetta Durante
;
Francesco Saverio Di Leva
;
Sandro
Cosconati
;
Emanuela Masini
;
Andrea Scozzafava
;
Ettore Novellino
;
Claudiu T. Supuran
;
Fabrizio Carta
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Lead Optimization of 2-Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of Gliomas
作者:
Simona Daniele
;
Valeria La Pietra
;
Elisabetta Barresi
;
Salvatore Di Maro
;
Eleonora Da Pozzo
;
Marco Robello
;
Concettina La Motta
;
Sandro
Cosconati
;
Sabrina Taliani
;
Luciana Marinelli
;
Ettore Novellino
;
Claudia Martini
;
Federico Da Settimo
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Switchable Protecting Strategy for Solid Phase Synthesis of DNA and RNA Interacting Nucleopeptides
作者:
Maria Emilia Mercurio
;
Stefano Tomassi
;
Maria Gaglione
;
Rosita Russo
;
Angela Chambery
;
Stefania Lama
;
Paola Stiuso
;
Sandro
Cosconati
;
Ettore Novellino
;
Salvatore Di Maro
;
Anna Messere
刊名:Journal of Organic Chemistry
出版年:2016
4.
Deepening the Topology of the Translocator Protein Binding Site by Novel N,N-Dialkyl-2-arylindol-3-ylglyoxylamides
作者:
Elisabetta Barresi
;
Agostino Bruno
;
Sabrina Taliani
;
Sandro
Cosconati
;
Eleonora Da Pozzo
;
Silvia Salerno
;
Francesca Simorini
;
Simona Daniele
;
Chiara Giacomelli
;
Anna Maria Marini
;
Concettina La Motta
;
Luciana Marinelli
;
Barbara Cosimelli
;
Ettore Novellino
;
Giovanni Greco
;
Federico Da Settimo
;
Claudia Martini
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity
作者:
Thomas C. Eadsforth
;
Andrea Pinto
;
Rosaria Luciani
;
Lucia Tamborini
;
Gregorio Cullia
;
Carlo De Micheli
;
Luciana Marinelli
;
Sandro
Cosconati
;
Ettore Novellino
;
Leonardo Lo Presti
;
Anabela Cordeiro da Silva
;
Paola Conti
;
William N. Hunter
;
Maria P. Costi
刊名:Journal of Medicinal Chemistry
出版年:2015
6.
N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase
作者:
Luca Pescatori
;
Mathieu M茅tifiot
;
Suhman Chung
;
Takashi Masoaka
;
Giuliana Cuzzucoli Crucitti
;
Antonella Messore
;
Giovanni Pupo
;
Valentina Noemi Madia
;
Francesco Saccoliti
;
Luigi Scipione
;
Silvano Tortorella
;
Francesco Saverio Di Leva
;
Sandro
Cosconati
;
Luciana Marinelli
;
Ettore Novellino
;
Stuart F. J. Le Grice
;
Yves Pommier
;
Christophe Marchand
;
Roberta Costi
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2015
7.
Design, Synthesis, and Biological Evaluation of Novel 2-((2-(4-(Substituted)phenylpiperazin-1-yl)ethyl)amino)-5鈥?N-ethylcarboxamidoadenosines as Potent and Selective Agonists of the A2A
作者:
Delia Preti
;
Pier Giovanni Baraldi
;
Giulia Saponaro
;
Romeo Romagnoli
;
Mojgan Aghazadeh Tabrizi
;
Stefania Baraldi
;
Sandro
Cosconati
;
Agostino Bruno
;
Ettore Novellino
;
Fabrizio Vincenzi
;
Annalisa Ravani
;
Pier Andrea Borea
;
Katia Varani
刊名:Journal of Medicinal Chemistry
出版年:2015
8.
A Unique Capsular Polysaccharide Structure from the Psychrophilic Marine Bacterium Colwellia psychrerythraea 34H That Mimics Antifreeze (Glyco)proteins
作者:
Sara Carillo
;
Angela Casillo
;
Giuseppina Pieretti
;
Ermenegilda Parrilli
;
Filomena Sannino
;
Maddalena Bayer-Giraldi
;
Sandro
Cosconati
;
Ettore Novellino
;
Marcela Ewert
;
Jody W. Deming
;
Rosa Lanzetta
;
Gennaro Marino
;
Michelangelo Parrilli
;
Antonio Randazzo
;
Maria L. Tutino
;
M. Michela Corsaro
刊名:Journal of the American Chemical Society
出版年:2015
9.
Structure鈥揂ctivity Relationship Refinement and Further Assessment of 4-Phenylquinazoline-2-carboxamide Translocator Protein Ligands as Antiproliferative Agents in Human Glioblastoma Tumors
作者:
Sabrina Castellano
;
Sabrina Taliani
;
Monica Viviano
;
Ciro Milite
;
Eleonora Da Pozzo
;
Barbara Costa
;
Elisabetta Barresi
;
Agostino Bruno
;
Sandro
Cosconati
;
Luciana Marinelli
;
Giovanni Greco
;
Ettore Novellino
;
Gianluca Sbardella
;
Federico Da Settimo
;
Claudia Martini
刊名:Journal of Medicinal Chemistry
出版年:2014
10.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
作者:
Roberta Costi
;
Mathieu M茅tifiot
;
Suhman Chung
;
Giuliana Cuzzucoli Crucitti
;
Kasthuraiah Maddali
;
Luca Pescatori
;
Antonella Messore
;
Valentina Noemi Madia
;
Giovanni Pupo
;
Luigi Scipione
;
Silvano Tortorella
;
Francesco Saverio Di Leva
;
Sandro
Cosconati
;
Luciana Marinelli
;
Ettore Novellino
;
Stuart F. J. Le Grice
;
Angela Corona
;
Yves Pommier
;
Christophe Marchand
;
Roberto Di Santo
刊名:Journal of Medicinal Chemistry
出版年:2014
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