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SpringerLink电子期刊(13)
Elsevier电子期刊(18)
ACS电子期刊(3)
在“
SpringerLink电子期刊
”中,
命中:
13
条,耗时:0.0109948 秒
在所有数据库中总计命中:
34
条
1.
Exploring structural requirements for peripherally acting 1,5-diaryl pyrazole-containing cannabinoid 1 receptor antagonists for the treatment of obesity
作者:
Mayank Kumar Sharma
;
Prashant R. Murumkar
;
Rajani
Giridhar
…
关键词:
3D
;
QSAR
;
Endocannabinoids
;
CB1 receptor antagonists
;
1
;
5
;
Diaryl pyrazole
;
Rimonabant
刊名:Molecular Diversity
出版年:2015
2.
Regioselective alkylation of 1,3,4,5-tetrahydrobenzo[d]azepin-2-one and biological evaluation of the resulting alkylated products as potentially selective
作者:
Navnit Prajapati
;
Rajani
Giridhar
;
Anshuman Sinha
;
Ashish M. Kanhed…
关键词:3 ;
Benzazepine
;
Regioselective alkylation
;
Phenethyl fragment
;
Selective $$\hbox {5
;
HT}_{\mathrm{2C}}$$ 5
;
HT 2 C agonists
;
Anti
;
obesity agents
刊名:Molecular Diversity
出版年:2015
3.
Virtual screening-based identification of lead molecules as selective TACE inhibitors
作者:
Prashant R. Murumkar
;
Mayank Kumar Sharma
;
Rajani
Giridhar
…
关键词:
TNF
α ;
TACE inhibitors
;
IK
;
682
;
Docking
;
Virtual screening
刊名:Medicinal Chemistry Research
出版年:2015
4.
Potential of Piperazinylalkylester Prodrugs of 6-Methoxy-2-Naphthylacetic Acid (6-MNA) for Percutaneous Drug Delivery
作者:
Vijay Pawar
;
Rushabh Thosani
;
Ashish Kanhed
;
Rajani
Giridhar
…
关键词:6 ;
MNA
;
NSAID
;
piperazinylalkylester
;
prodrug
;
skin permeation
刊名:AAPS PharmSciTech
出版年:2015
5.
Erratum to: Potential of Piperazinylalkylester Prodrugs of 6-Methoxy-2-Naphthylacetic Acid (6-MNA) for Percutaneous Drug Delivery
作者:
Vijay Pawar
;
Rushabh Thosani
;
Ashish Kanhed
;
Rajani
Giridhar
…
刊名:AAPS PharmSciTech
出版年:2015
6.
Structural requirements for imidazo[1,2-a]pyrazine derivatives as Aurora A kinase inhibitors and validation of the model
作者:
Ashish M. Kanhed (1)
Vishal P. Zambre (1)
Vijay A. Pawar (1)
Mayank Kumar Sharma (1)
Rajani
Giridhar
(1)
Mange Ram Yadav (1)
关键词:
Aurora A kinase
;
Cancer
;
Imidazo[1
2 ;
a]pyrazine
;
AutoDock
;
CoMFA and CoMSIA
;
3D
;
QSAR
刊名:Medicinal Chemistry Research
出版年:2014
7.
Pharmacophore modeling and 3D-QSAR (CoMSIA) studies for structural requirements of some triazine derivatives as G-quadruplex binders for telomerase inhibition
作者:
Vishal P. Zambre (1)
Rajani
Giridhar
(1)
Mange Ram Yadav (1)
关键词:
Telomerase inhibitors
;
G
;
Quadruplex binders
;
Triazine derivatives
;
CoMSIA
;
Pharmacophore
刊名:Medicinal Chemistry Research
出版年:2013
8.
Synthesis of novel 4,6-diaryl-2-aminopyrimidines as potential antiplasmodial agents
作者:
Rajani
Giridhar
(1)
Riyaj S. Tamboli (1)
Dhaval G. Prajapati (1)
Sanket Soni (2)
Sarita Gupta (2)
M. R. Yadav (1)
关键词:2 ;
Aminopyrimidines
;
Chloroquine
;
Plasmodium falciparum
;
Antiplasmodial agents
刊名:Medicinal Chemistry Research
出版年:2013
9.
3D-QSAR studies of 4-quinolone derivatives as high-affinity ligands at the benzodiazepine site of brain GABAA receptors
作者:
Anand Gaurav (1)
Mange R. Yadav (2)
Rajani
Giridhar
(2)
Vertika Gautam (1)
Ranjit Singh (1)
关键词:
GABA
;
3D
;
QSAR
;
CoMFA
;
CoMSIA
;
Leave one out
;
PLS analysis
刊名:Medicinal Chemistry Research
出版年:2011
10.
Substituted aminoalcohol ester analogs of indomethacin with reduced toxic effects
作者:
Parmeshwari K. Halen (1)
Kewal K. Chagti (1)
Rajani
Giridhar
(1)
Mange Ram Yadav (1)
关键词:
Antiinflammatory
;
Indomethacin
;
Ulceration
刊名:Medicinal Chemistry Research
出版年:2007
1
2
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