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内部出版物
在“
SpringerLink电子期刊
”中,
命中:
21
条,耗时:小于0.01 秒
1.
The antimitotic pyrimido[4,5-c]quinolin-1(2H)-one scaffold: probing substituents at position 3
作者:
Kamel Metwally
;
Harris Pratsinis
;
Dimitris Kletsas
关键词:
Cytotoxic agents
;
Anticancer
;
Antimitotic
;
Pyrimido[4
5 ;
c]quinolin
;
1(2H)
;
ones
刊名:Medicinal Chemistry Research
出版年:2015
2.
Quinoline-Based Compound BPIQ Exerts Anti-Proliferative Effects on Human Retinoblastoma Cells via Modulating Intracellular Reactive Oxygen Species
作者:
Kai-Chun Cheng
;
Chun-Tzu Hung
;
Kuo-Jen Chen…
关键词:
BPIQ
;
Quinoline
;
Retinoblastoma
;
Reactive oxygen species
;
DNA damage
;
Apoptosis
刊名:Archivum Immunologiae et Therapiae Experimentalis
出版年:2016
3.
Structure–activity relationship investigation of methoxy substitution on anticancer pyrimido[4,5-c]quinolin-1(2H)-ones
作者:
Kamel Metwally (1)
Ashraf Khalil (2)
Asmaa Sallam (3)
Harris Pratsinis (4)
Dimitris Kletsas (4)
Khalid El Sayed (3)
关键词:
Anticancer
;
Cytotoxicity
;
Methoxy substitution
;
Pyrimido[4
5 ;
c]quinolin
;
1(2H)
;
ones
;
Migration
;
Tubulin
;
Wound
;
healing
刊名:Medicinal Chemistry Research
出版年:2013
4.
PQ-69, a novel and selective adenosine A1 receptor antagonist with inverse agonist activity
作者:
Min Lu
;
Bo Wang
;
Cheng Zhang
;
Xiaomei Zhuang
;
Mei Yuan…
关键词:4 ;
butylamino
2 ;
(3
;
fluorophenyl)[4
3 ;
c]quinolin
3 ;
one
;
Non
;
xanthine adenosine A1 receptor (A1AR) antagonist
;
Inverse agonism
;
Diuresis
刊名:Purinergic Signalling
出版年:2014
5.
BPIQ, a novel synthetic quinoline derivative, inhibits growth and induces mitochondrial apoptosis of lung cancer cells in vitro and in zebrafish xenograft model
作者:
Chien-Chih Chiu
;
Han-Lin Chou
;
Bing-Hung Chen
;
Kuo-Feng Chang
;
Chih-Hua Tseng…
关键词:
Indeno[1
2 ;
c]quinolinequinoline
;
BPIQ
;
Lung cancer
;
Apoptosis
;
Polyploidy
;
Zebrafish xenograft
刊名:BMC Cancer
出版年:2015
6.
Synthesis of azabicyclo[4.2.0]octa-1,3,5-trien-8-one analogues of 1H-imidazo[4,5-c]quinoline and evaluation of their antimicrobial and anticancer activities
作者:
Reshma Kayarmar (1) (2)
G. K. Nagaraja (1) (2)
Manjunath Bhat (1) (2)
Prashantha Naik (3)
K. P. Rajesh (4)
Suchetha Shetty (5)
T. Arulmoli (2)
关键词:
Imidazoquinoline
;
Antimicrobial activity
;
Anticancer activity
;
Docking study
;
β
;
Tubulin
刊名:Medicinal Chemistry Research
出版年:2014
7.
Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β?Site
作者:
Pantea Mirheydari (1)
Joachim Ramerstorfer (1)
Zdravko Varagic (1)
Petra Scholze (3)
Laurin Wimmer (2)
Marko M. Mihovilovic (2)
Werner Sieghart (1)
Margot Ernst (1)
关键词:
GABAA
;
CGS 9895
;
Pyrazoloquinolinones
;
α+ β?Binding site
;
Positive modulators
;
Null modulators
;
δ Subunit
;
Extrasynaptic receptor
刊名:Neurochemical Research
出版年:2014
8.
A Drug Mystery of Heterocycles: Various Molecules for One Target or One Compound for Multiple Targets?
作者:
I. Shcherbakova (1)
关键词:
ambocarb
;
2
347 ;
tetrahydroindolo[2
3 ;
c]quinolin
1 ;
ones
;
inhibitors of MT3/QR2 receptor/enzyme
;
DYRK1A kinase and L
;
type calcium channels
;
multitarget CNS drugs
刊名:Chemistry of Heterocyclic Compounds
出版年:2013
9.
Photo-induced antimicrobial and DNA cleavage studies of indoloquinolines and 1,8-naphtharidine
作者:
MALATHI MAHALINGAM (1)
PALATHURAI SUBRAMANIAM MOHAN (1)
KASIRAJAN GAYATHRI (1)
RAMADOSS GOMATHI (1)
PUSHPARAJA SUBHAPRIYA (2)
关键词:
Vilsmeier–Haack reagent
;
indoloquinolines
;
photosensitizer
;
photoinduced antibacterial activity
;
photo
;
DNA binding
刊名:Journal of Chemical Sciences
出版年:2013
10.
Highly Sensitive Quantitative Analysis of 1-[3-(Furo[3,2-
c
]quinolin-4-ylamino)phenyl]ethanone Oxime, a New Antitumor Agent, in Rat Plasma by LC with Electrochemical Detection
作者:
Pao-Chu Wu
;
Yaw-Bin Huang
;
Chih-Kai Chang
;
Yeh-Long Chen
;
Cherng-Chyi Tzeng and Yi-Hung Tsai
关键词:
Column liquid chromatography
;
Amsacrine
;
Antitumor
;
1
;
[3
;
(Furo[3
2 ;
c]quinolin
4 ;
ylamino)phenyl]ethanone oxime
;
Pharmacokinetics
刊名:Chromatographia
出版年:2009
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