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SpringerLink电子期刊(10)
NATURE电子期刊(2)
Elsevier电子期刊(3)
ACS电子期刊(9)
在“
ACS电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
24
条
1.
Discovery of N-(4-Fluoro-3-methoxybenzyl)-6-(2-(((2S,5R)-5-(hydroxymethyl)-1,4-dioxan-2-yl)methyl)-2H-tetrazol-5-yl)-2-methylpyrimidine-4-carboxamide. A Highly Selective and Orally Bioavailable Matrix
作者:
Peter G. Ruminski
;
Mark Massa
;
Joseph Strohbach
;
Cathleen E. Hanau
;
Michelle Schmidt
;
Jeffrey A. Scholten
;
Theresa R. Fletcher
;
Bruce C. Hamper
;
Jeffery N. Carroll
;
Huey S. Shieh
;
Nicole Caspers
;
Brandon
Collins
;
Margaret Grapperhaus
;
Katherine E. Palmquist
;
Joe
Collins
;
John E. Baldus
;
Jeffrey Hitchcock
;
H. Peter Kleine
;
Michael D. Rogers
;
Joseph McDonald
;
Grace E. Munie
;
Dean M. Messing
;
Silvia Portolan
;
Laurence O. Whiteley
;
Teresa Sunyer
;
Mark E. Schnute
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Multiparameter Lead Optimization to Give an Oral Checkpoint Kinase 1 (CHK1) Inhibitor Clinical Candidate: (R)-5-((4-((Morpholin-2-ylmethyl)amino)-5-(trifluoromethyl)pyridin-2-yl)amino)pyrazine-2-carbonitrile (CCT245737)
作者:
James D. Osborne
;
Thomas P. Matthews
;
Tatiana McHardy
;
Nicolas Proisy
;
Kwai-Ming J. Cheung
;
Michael Lainchbury
;
Nathan Brown
;
Michael I. Walton
;
Paul D. Eve
;
Katherine J. Boxall
;
Angela Hayes
;
Alan T. Henley
;
Melanie R. Valenti
;
Alexis K. De Haven
Brandon
;
Gary Box
;
Yann Jamin
;
Simon P. Robinson
;
Isaac M. Westwood
;
Rob L. M. van Montfort
;
Philip M. Leonard
;
Marieke B. A. C. Lamers
;
John C. Reader
;
G. Wynne Aherne
;
Florence I. Raynaud
;
Suzanne A. Eccles
;
Michelle D. Garrett
;
Ian
Collins
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Correction to Fragment-Based Discovery of Indole Inhibitors of Matrix Metalloproteinase-13
作者:
Steven J. Taylor
;
Asitha Abeywardane
;
Shuang Liang
;
Ingo Muegge
;
Anil K. Padyana
;
Zhaoming Xiong
;
Melissa Hill-Drzewi
;
Bennett Farmer
;
Xiang Li
;
Brandon
Collins
;
John Xiang Li
;
Alexander Heim-Riether
;
John Proudfoot
;
Qiang Zhang
;
Daniel Goldberg
;
Ljiljana Zuvela-Jelaska
;
Hani Zaher
;
Jun Li
;
Neil A. Farrow
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Discovery of Potent, Selective Chymase Inhibitors via Fragment Linking Strategies
作者:
Steven J. Taylor
;
Anil K. Padyana
;
Asitha Abeywardane
;
Shuang Liang
;
Ming-Hong Hao
;
St茅phane De Lombaert
;
John Proudfoot
;
Bennett S. Farmer
;
III
;
Xiang Li
;
Brandon
Collins
;
Leslie Martin
;
Daniel R. Albaugh
;
Melissa Hill-Drzewi
;
Steven S. Pullen
;
Hidenori Takahashi
刊名:Journal of Medicinal Chemistry
出版年:2013
5.
Discovery of 3-Alkoxyamino-5-(pyridin-2-ylamino)pyrazine-2-carbonitriles as Selective, Orally Bioavailable CHK1 Inhibitors
作者:
Michael Lainchbury
;
Thomas P. Matthews
;
Tatiana McHardy
;
Kathy J. Boxall
;
Michael I. Walton
;
Paul D. Eve
;
Angela Hayes
;
Melanie R. Valenti
;
Alexis K. de Haven
Brandon
;
Gary Box
;
G. Wynne Aherne
;
John C. Reader
;
Florence I. Raynaud
;
Suzanne A. Eccles
;
Michelle D. Garrett
;
Ian
Collins
刊名:Journal of Medicinal Chemistry
出版年:2012
6.
Fragment-Based Discovery of Indole Inhibitors of Matrix Metalloproteinase-13
作者:
Steven J. Taylor
;
Asitha Abeywardane
;
Shuang Liang
;
Ingo Muegge
;
Anil K. Padyana
;
Zhaoming Xiong
;
Melissa Hill-Drzewi
;
Bennett Farmer
;
Xiang Li
;
Brandon
Collins
;
John Xiang Li
;
Alexander Heim-Riether
;
John Proudfoot
;
Qiang Zhang
;
Daniel Goldberg
;
Ljiljana Zuvela-Jelaska
;
Hani Zaher
;
Jun Li
;
Neil A. Farrow
刊名:Journal of Medicinal Chemistry
出版年:2011
7.
Structure-Guided Evolution of Potent and Selective CHK1 Inhibitors through Scaffold Morphing
作者:
John C. Reader
;
Thomas P. Matthews
;
Suki Klair
;
Kwai-Ming J. Cheung
;
Jane Scanlon
;
Nicolas Proisy
;
Glynn Addison
;
John Ellard
;
Nelly Piton
;
Suzanne Taylor
;
Michael Cherry
;
Martin Fisher
;
Kathy Boxall
;
Samantha Burns
;
Michael I. Walton
;
Isaac M. Westwood
;
Angela Hayes
;
Paul Eve
;
Melanie Valenti
;
Alexis de Haven
Brandon
;
Gary Box
;
Rob L. M. van Montfort
;
David H. Williams
;
G. Wynne Aherne
;
Florence I. Raynaud
;
Suzanne A. Eccles
;
Michelle D. Garrett
;
Ian
Collins
刊名:Journal of Medicinal Chemistry
出版年:2011
8.
Sterically Hindered Aluminum Alkyls: Weakly Interacting Scavenging Agents of Use in Olefin Polymerization
作者:
Russell A. Stapleton
;
Abdulaziz Al-Humydi
;
Jianfang Chai
;
Brandon
R. Galan
;
Scott
Collins
刊名:Organometallics
出版年:2006
9.
Bulky Aluminum Alkyl Scavengers in Olefin Polymerization with Group 4 Catalysts
作者:
Russell A. Stapleton
;
Brandon
R. Galan
;
Scott
Collins
;
Richard S. Simons
;
Jered C. Garrison
;
and Wiley J. Youngs
刊名:Journal of the American Chemical Society
出版年:2003
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