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SpringerLink电子期刊(3)
Elsevier电子期刊(7)
ACS电子期刊(24)
在“
ACS电子期刊
”中,
命中:
24
条,耗时:0.0319862 秒
在所有数据库中总计命中:
34
条
1.
The Discove
r
y and Cha
r
acte
r
ization of the 伪-Amino-3-hyd
r
oxy-5-methyl-4-isoxazolep
r
opionic Acid (AMPA) Recepto
r
Potentiato
r
N-{(3S,4S)-4-[4-(5-Cyano-2-thienyl)phenoxy]tet
r
ahyd
r
ofu
r
作者:
Ch
r
istophe
r
L. Shaffe
r
;
Nandini C. Patel
;
Jacob Schwa
r
z
;
R
enato J. Scialis
;
Yunjing Wei
;
Xinjun J. Hou
;
Longfei Xie
;
Kapil Ka
r
ki
;
Dianne K. B
r
yce
;
Sa
r
ah M. Osgood
;
William E. Hoffmann
;
John T. Lazza
r
o
;
Cheng Chang
;
Dina F. McGinnis
;
Susan M. Lota
r
ski
;
JianHua Liu
;
R
.
Scott
Obach
;
Ma
r
k L. Webe
r
;
Laigao Chen
;
Kenneth
R
. Zasadny
;
Pat
r
icia A. Seymou
r
;
Ch
r
istophe
r
J. Schmidt
;
Mih谩ly Haj贸s
;
R
aymond S. Hu
r
st
;
Jayva
r
dhan Pandit
;
Ch
r
istophe
r
J. O鈥橠onnell
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2015
2.
Unbiased Scanning Method and Data Banking App
r
oach Using Ult
r
a-High Pe
r
fo
r
mance Liquid Ch
r
omatog
r
aphy Coupled with High-Resolution Mass Spect
r
omet
r
y fo
r
Quantitative Compa
r
ison of Metabolite Exposu
r
e
作者:
Hongying Gao
;
Shibing Deng
;
R
.
Scott
Obach
刊名:Analytical Chemist
r
y
出版年:2015
3.
Chemical and Computational Methods fo
r
the Cha
r
acte
r
ization of Covalent Reactive G
r
oups fo
r
the P
r
ospective Design of I
rr
eve
r
sible Inhibito
r
s
作者:
Ma
r
k E. Flanagan
;
Joseph A. Ab
r
amite
;
Dennis P. Ande
r
son
;
Ann Aulabaugh
;
Upend
r
a P. Dahal
;
Adam M. Gilbe
r
t
;
Chao Li
;
Justin Montgome
r
y
;
Stacey
R
. Oppenheime
r
;
Tim
R
yde
r
;
B
r
andon P. Schuff
;
Daniel P. Uccello
;
G
r
ego
r
y S. Walke
r
;
Yan Wu
;
Matthew F. B
r
own
;
Jinshan M. Chen
;
Matthew M. Haywa
r
d
;
Ma
r
k C. Noe
;
R
.
Scott
Obach
;
Lau
r
ence Philippe
;
Vee
r
abahu Shanmugasunda
r
am
;
Michael J. Shapi
r
o
;
Je
r
emy Sta
rr
;
Justin St
r
oh
;
Ye Che
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2014
4.
Clea
r
ance Mechanism Assignment and Total Clea
r
ance P
r
ediction in Human Based upon in Silico Models
作者:
F
r
anco Lomba
r
do
;
R
.
Scott
Obach
;
Manthena V. Va
r
ma
;
R
owan St
r
inge
r
;
Giuliano Be
r
ellini
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2014
5.
Mechanism-Based Inactivation (MBI) of Cytoch
r
ome P450 Enzymes: St
r
uctu
r
e鈥揂ctivity Relationships and Discove
r
y St
r
ategies To Mitigate D
r
ug鈥揇
r
ug Inte
r
action Risks
作者:
Suvi T. M. O
rr
;
Sha
r
on L. Ripp
;
T. E
r
ic Balla
r
d
;
Jaclyn L. Hende
r
son
;
Dennis O.
Scott
;
R
.
Scott
Obach
;
Hao Sun
;
Amit S. Kalgutka
r
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2012
6.
Benchma
r
king in Vit
r
o Covalent Binding Bu
r
den As a Tool To Assess Potential Toxicity Caused by Nonspecific Covalent Binding of Covalent D
r
ugs
作者:
Upend
r
a P. Dahal
;
R
.
Scott
Obach
;
Adam M. Gilbe
r
t
刊名:Chemical
R
esea
r
ch in Toxicology
出版年:2013
7.
Identification of P
r
otein Ta
r
gets of Reactive Metabolites of Tienilic Acid in Human Hepatocytes
作者:
Yakov M. Koen
;
Diganta Sa
r
ma
;
Todd D. Williams
;
Nadezhda A. Galeva
;
R
.
Scott
Obach
;
R
obe
r
t P. Hanzlik
刊名:Chemical
R
esea
r
ch in Toxicology
出版年:2012
8.
Metabolism-Di
r
ected Design of Oxetane-Containing A
r
ylsulfonamide De
r
ivatives as 纬-Sec
r
etase Inhibito
r
s
作者:
Antonia F. Stepan
;
Kapil Ka
r
ki
;
W.
Scott
McDonald
;
Pete
r
H. Do
r
ff
;
Jason K. Dut
r
a
;
Kenneth J. Di
R
ico
;
Annie Won
;
Chak
r
apani Sub
r
amanyam
;
Ivan V. Ef
r
emov
;
Ch
r
istophe
r
J. O鈥橠onnell
;
Cha
r
les E. Nolan
;
Stacey L. Becke
r
;
Leslie
R
. Pustilnik
;
Blossom Sneed
;
Hao Sun
;
Yasong Lu
;
Ashley E.
R
obshaw
;
David
R
iddell
;
The
r
esa J. O'Sullivan
;
Evelyn Sibley
;
Steven Capetta
;
Kevin Atchison
;
And
r
ew J. Hallg
r
en
;
Emily Mille
r
;
Anthony Wood
;
R
.
Scott
Obach
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2011
9.
Physicochemical Space fo
r
Optimum O
r
al Bioavailability: Cont
r
ibution of Human Intestinal Abso
r
ption and Fi
r
st-Pass Elimination
作者:
Manthena V. S. Va
r
ma
;
R
.
Scott
Obach
;
Cha
r
les Rotte
r
;
Howa
r
d R. Mille
r
;
Geo
r
ge Chang
;
Stefanus J. Steyn
;
Ayman El-Kattan
;
Matthew D. T
r
outman
刊名:Jou
r
nal of Medicinal Chemist
r
y
出版年:2010
10.
NADPH-Dependent Covalent Binding of [3H]Pa
r
oxetine to Human Live
r
Mic
r
osomes and S-9 F
r
actions: Identification of an Elect
r
ophilic Quinone Metabolite of Pa
r
oxetine
作者:
Sab
r
ina X. Zhao
;
Deepak K. Dalvie
;
Joan M. Kelly
;
John
R
. Soglia
;
Kosea S. F
r
ede
r
ick
;
Evan B. Smith
;
R
.
Scott
Obach
;
Amit S. Kalgutka
r
刊名:Chemical
R
esea
r
ch in Toxicology
出版年:2007
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