设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Wiley电子期刊(1)
SpringerLink电子期刊(2)
Elsevier电子期刊(30)
ACS电子期刊(33)
在“
ACS电子期刊
”中,
命中:
33
条,耗时:小于0.01 秒
在所有数据库中总计命中:
66
条
1.
Fragment-Linking Approach Using 19F NMR Spectroscopy To Obtain Highly Potent and Selective Inhibitors of β-Secretase
作者:
John B. Jordan
;
Douglas
A.
Whittington
;
Michael D. Bartberger
;
E. Allen Sickmier
;
Kui Chen
;
Yuan Cheng
;
Ted Judd
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quino
作者:
Felix Gonzalez-Lopez de Turiso
;
Xiaolin Hao
;
Youngsook Shin
;
Minna Bui
;
Iain D. G. Campuzano
;
Mario Cardozo
;
Michelle C. Dunn
;
Jason Duquette
;
Benjamin Fisher
;
Robert S. Foti
;
Kirk Henne
;
Xiao He
;
Yi-Ling Hu
;
Ron C. Kelly
;
Michael G. Johnson
;
Brian S. Lucas
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Sharon Wannberg
;
Douglas
A.
Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery of (R)-6-(1-(8-Fluoro-6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl)-3-(2-methoxyethoxy)-1,6-naphthyridin-5(6H)-one (AMG 337), a Potent and Selective Inhibitor of MET with High Unbound Target Coverage and Robust In Vivo A
作者:
Alessandro A. Boezio
;
Katrina W. Copeland
;
Karen Rex
;
Brian K. Albrecht
;
David Bauer
;
Steven F. Bellon
;
Christiane Boezio
;
Martin A. Broome
;
Deborah Choquette
;
Angela Coxon
;
Isabelle Dussault
;
Satoko Hirai
;
Richard Lewis
;
Min-Hwa Jasmine Lin
;
Julia Lohman
;
Jingzhou Liu
;
Emily A. Peterson
;
Michele Potashman
;
Roman Shimanovich
;
Yohannes Teffera
;
Douglas
A.
Whittington
;
Karina R. Vaida
;
Jean-Christophe Harmange
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery, Optimization, and in Vivo Evaluation of Benzimidazole Derivatives AM-8508 and AM-9635 as Potent and Selective PI3Kδ Inhibitors
作者:
Youngsook Shin
;
Julia Suchomel
;
Mario Cardozo
;
Jason Duquette
;
Xiao He
;
Kirk Henne
;
Yi-Ling Hu
;
Ron C. Kelly
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Simon Wong
;
Sharon Wannberg
;
Douglas
A.
Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
An Orally Available BACE1 Inhibitor That Affords Robust CNS A尾 Reduction without Cardiovascular Liabilities
作者:
Yuan Cheng
;
James Brown
;
Ted C. Judd
;
Patricia Lopez
;
Wenyuan Qian
;
Timothy S. Powers
;
Jian Jeffrey Chen
;
Michael D. Bartberger
;
Kui Chen
;
Robert T. Dunn
;
II
;
Oleg Epstein
;
Robert T. Fremeau
;
Jr.
;
Scott Harried
;
Dean Hickman
;
Stephen A. Hitchcock
;
Yi Luo
;
Ana Elena Minatti
;
Vinod F. Patel
;
Hugo M. Vargas
;
Robert C. Wahl
;
Matthew M. Weiss
;
Paul H. Wen
;
Ryan D. White
;
Douglas
A.
Whittington
;
Xiao Mei Zheng
;
Stephen Wood
刊名:ACS Medicinal Chemistry Letters
出版年:2015
6.
Correction to Discovery of Potent and Selective 8-Fluorotriazolopyridine c-Met Inhibitors
作者:
Emily A. Peterson
;
Yohannes Teffera
;
Brian K. Albrecht
;
David Bauer
;
Steven F. Bellon
;
Alessandro Boezio
;
Christiane Boezio
;
Martin A. Broome
;
Deborah Choquette
;
Katrina W. Copeland
;
Isabelle Dussault
;
Richard Lewis
;
Min-Hwa Jasmine Lin
;
Julia Lohman
;
Jingzhou Liu
;
Michele Potashman
;
Karen Rex
;
Roman Shimanovich
;
Douglas
A.
Whittington
;
Karina R. Vaida
;
Jean-Christophe Harmange
刊名:Journal of Medicinal Chemistry
出版年:2015
7.
Discovery and in Vivo Evaluation of (S)-N-(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and Related PI3K未 Inhibitors for Inflammation and Autoimmune
作者:
Timothy D. Cushing
;
Xiaolin Hao
;
Youngsook Shin
;
Kristin Andrews
;
Matthew Brown
;
Mario Cardozo
;
Yi Chen
;
Jason Duquette
;
Ben Fisher
;
Felix Gonzalez-Lopez de Turiso
;
Xiao He
;
Kirk R. Henne
;
Yi-Ling Hu
;
Randall Hungate
;
Michael G. Johnson
;
Ron C. Kelly
;
Brian Lucas
;
John D. McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Tisha San Miguel
;
Deanna Mohn
;
Vatee Pattaropong
;
Liping H. Pettus
;
Andreas Reichelt
;
Robert M. Rzasa
;
Jennifer Seganish
;
Andrew S. Tasker
;
Robert C. Wahl
;
Sharon Wannberg
;
Douglas
A.
Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Dawei Zhang
;
Daniela P. Metz
刊名:Journal of Medicinal Chemistry
出版年:2015
8.
Inhibitors of 尾-Site Amyloid Precursor Protein Cleaving Enzyme (BACE1): Identification of (S)-7-(2-Fluoropyridin-3-yl)-3-((3-methyloxetan-3-yl)ethynyl)-5鈥?i>H-spiro[chromeno[2,3-b]py
作者:
Thomas A. Dineen
;
Kui Chen
;
Alan C. Cheng
;
Katayoun Derakhchan
;
Oleg Epstein
;
Joel Esmay
;
Dean Hickman
;
Chuck E. Kreiman
;
Isaac E. Marx
;
Robert C. Wahl
;
Paul H. Wen
;
Matthew M. Weiss
;
Douglas
A.
Whittington
;
Stephen Wood
;
Robert T. Fremeau
;
Jr.
;
Ryan D. White
;
Vinod F. Patel
刊名:Journal of Medicinal Chemistry
出版年:2014
9.
Lead Optimization and Modulation of hERG Activity in a Series of Aminooxazoline Xanthene 尾-Site Amyloid Precursor Protein Cleaving Enzyme (BACE1) Inhibitors
作者:
Oleg Epstein
;
Marian C. Bryan
;
Alan C. Cheng
;
Katayoun Derakhchan
;
Thomas A. Dineen
;
Dean Hickman
;
Zihao Hua
;
Jason B. Human
;
Charles Kreiman
;
Isaac E. Marx
;
Matthew M. Weiss
;
Robert C. Wahl
;
Paul H. Wen
;
Douglas
A.
Whittington
;
Stephen Wood
;
Xiao Mei Zheng
;
Robert T. Fremeau
;
Jr.
;
Ryan D. White
;
Vinod F. Patel
刊名:Journal of Medicinal Chemistry
出版年:2014
10.
The Discovery and Optimization of a Novel Class of Potent, Selective, and Orally Bioavailable Anaplastic Lymphoma Kinase (ALK) Inhibitors with Potential Utility for the Treatment of Cancer
作者:
Richard T. Lewis
;
Christiane M. Bode
;
Deborah M. Choquette
;
Michele Potashman
;
Karina Romero
;
John C. Stellwagen
;
Yohannes Teffera
;
Earl Moore
;
Douglas
A.
Whittington
;
Hao Chen
;
Linda F. Epstein
;
Renee Emkey
;
Paul S. Andrews
;
Violeta L. Yu
;
Douglas
C. Saffran
;
Man Xu
;
Allison Drew
;
Patricia Merkel
;
Steven Szilvassy
;
Rachael L. Brake
刊名:Journal of Medicinal Chemistry
出版年:2012
1
2
3
4
按检索点细分(33)
题名(33)
按出版年细分(33)
2016年(4)
2015年(3)
2014年(2)
2012年(10)
2011年(3)
2009年(1)
2003年(1)
2002年(1)
2001年(5)
2000年(1)
2000年及以前(2)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.