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SpringerLink电子期刊(4)
NATURE电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
25
条
1.
The Discovery and Hit-to-Lead Optimization of Tricyclic Sulfonamides as Potent and Efficacious Potentiators of Glycine Receptors
作者:
Howard BregmanJeffrey R. Simard
;
Kristin L. Andrews
;
Shawn Ayube
;
Hao Chen
;
Hakan Gunaydin
;
Angel Guzman-Perez
;
Jiali Hu
;
Liyue
Huang
;
Xin
Huang
;
Paul H. Krolikowski
;
Sonya G. Lehto
;
Richard T. Lewis
;
Klaus Michelsen
;
Pamela Pegman
;
Matthew H. Plant
;
Paul L. Shaffer
;
Yohannes Teffera
;
Shuyan Yi
;
Maosheng Zhang
;
Jacinthe Gingras
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2017
2.
Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement
作者:
Isaac E. Marx
;
Thomas A. Dineen
;
Jessica Able
;
Christiane Bode
;
Howard Bregman
;
Margaret Chu-Moyer
;
Erin F. DiMauro
;
Bingfan Du
;
Robert S. Foti
;
Robert T. Fremeau Jr.
;
Hua Gao
;
Hakan Gunaydin
;
Brian E. Hall
;
Liyue
Huang
;
Thomas Kornecook
;
Charles R. Kreiman
;
Daniel S. La
;
Joseph Ligutti
;
Min-Hwa Jasmine Lin
;
Dong Liu
;
Jeff S. McDermott
;
Bryan D. Moyer
;
Emily A. Peterson
;
Jonathan T. Roberts
;
Paul Rose
;
Jean Wang
;
Beth D. Youngblood
;
Violeta Yu
;
Matthew M. Weiss
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery of N-(4-(3-(2-Aminopyrimidin-4-yl)pyridin-2-yloxy)phenyl)-4-(4-methylthiophen-2-yl)phthalazin-1-amine (AMG 900), A Highly Selective, Orally Bioavailable Inhibitor of Aurora Kinases wi
作者:
Stephanie Geuns-Meyer
;
Victor J. Cee
;
Holly L. Deak
;
Bingfan Du
;
Brian L. Hodous
;
Hanh Nho Nguyen
;
Philip R. Olivieri
;
Laurie B. Schenkel
;
Karina R. Vaida
;
Paul Andrews
;
Annette Bak
;
Xuhai Be
;
Pedro J. Beltran
;
Tammy L. Bush
;
Mary K. Chaves
;
Grace Chung
;
Yang Dai
;
Patrick Eden
;
Kelly Hanestad
;
Liyue
Huang
;
Min-Hwa Jasmine Lin
;
Jin Tang
;
Beth Ziegler
;
Robert Radinsky
;
Richard Kendall
;
Vinod F. Patel
;
Marc Payton
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Structure-Based Design of 2-Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors
作者:
Hongbing
Huang
;
Angel Guzman-Perez
;
Lisa Acquaviva
;
Virginia Berry
;
Howard Bregman
;
Jennifer Dovey
;
Hakan Gunaydin
;
Xin
Huang
;
Liyue
Huang
;
Doug Saffran
;
Randy Serafino
;
Steve Schneider
;
Cindy Wilson
;
Erin F. DiMauro
刊名:ACS Medicinal Chemistry Letters
出版年:2013
5.
Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Howard Bregman
;
Nagasree Chakka
;
Angel Guzman-Perez
;
Hakan Gunaydin
;
Yan Gu
;
Xin
Huang
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue
Huang
;
Bryan Egge
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Ankita Mishra
;
John Newcomb
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Zihao Hua
;
Howard Bregman
;
John L. Buchanan
;
Nagasree Chakka
;
Angel Guzman-Perez
;
Hakan Gunaydin
;
Xin
Huang
;
Yan Gu
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue
Huang
;
Bryan Egge
;
Renee Emkey
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Lisa Acquaviva
;
Jennifer Dovey
;
Ankita Mishra
;
John Newcomb
;
Douglas Saffran
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Mary Stanton
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Structure-Based Design of Potent and Selective CK1纬 Inhibitors
作者:
Hongbing
Huang
;
Lisa Acquaviva
;
Virginia Berry
;
Howard Bregman
;
Nagasree Chakka
;
Anne O鈥機onnor
;
Erin F. DiMauro
;
Jennifer Dovey
;
Oleg Epstein
;
Barbara Grubinska
;
Jon Goldstein
;
Hakan Gunaydin
;
Zihao Hua
;
Xin
Huang
;
Liyue
Huang
;
Jason Human
;
Alex Long
;
John Newcomb
;
Vinod F. Patel
;
Doug Saffran
;
Randy Serafino
;
Steve Schneider
;
Craig Strathdee
;
Jin Tang
;
Susan Turci
;
Ryan White
;
Violeta Yu
;
Huilin Zhao
;
Cindy Wilson
;
Matthew W. Martin
刊名:ACS Medicinal Chemistry Letters
出版年:2012
8.
Identification of a Potent, State-Dependent Inhibitor of Nav1.7 with Oral Efficacy in the Formalin Model of Persistent Pain
作者:
Howard Bregman
;
Loren Berry
;
John L. Buchanan
;
April Chen
;
Bingfan Du
;
Elma Feric
;
Markus Hierl
;
Liyue
Huang
;
David Immke
;
Brett Janosky
;
Danielle Johnson
;
Xingwen Li
;
Joseph Ligutti
;
Dong Liu
;
Annika Malmberg
;
David Matson
;
Jeff McDermott
;
Peter Miu
;
Hanh Nho Nguyen
;
Vinod F. Patel
;
Daniel Waldon
;
Ben Wilenkin
;
Xiao Mei Zheng
;
Anruo Zou
;
Stefan I. McDonough
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2011
9.
Discovery and Optimization of a Novel Series of N-Arylamide Oxadiazoles as Potent, Highly Selective and Orally Bioavailable Cannabinoid Receptor 2 (CB2) Agonists
作者:
Yuan Cheng
;
Brian K. Albrecht
;
James Brown
;
John L. Buchanan
;
William H. Buckner
;
Erin F. DiMauro
;
Renee Emkey
;
Robert T. Fremeau
;
Jean-Christophe Harmange
;
Beth J. Hoffman
;
Liyue
Huang
;
Ming
Huang
刊名:Journal of Medicinal Chemistry
出版年:2008
10.
Discovery of a Potent, Selective, and Orally Bioavailable c-Met Inhibitor: 1-(2-Hydroxy-2-methylpropyl)-N-(5-(7-methoxyquinolin-4-yloxy)pyridin-2-yl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H
作者:
Longbin Liu
;
Aaron Siegmund
;
Ning Xi
;
Paula Kaplan-Lefko
;
Karen Rex
;
April Chen
;
Jasmine Lin
;
Jodi Moriguchi
;
Loren Berry
;
Liyue
Huang
;
Yohannes Teffera
;
Yajing Yang
;
Yihong Zhang
;
Steven F. Bellon
;
M
刊名:Journal of Medicinal Chemistry
出版年:2008
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