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NATURE电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(25)
在“
ACS电子期刊
”中,
命中:
25
条,耗时:小于0.01 秒
在所有数据库中总计命中:
36
条
1.
Facile Modulation of Antibody Fucosylation with Small Molecule Fucostatin Inhibitors and Cocrystal Structure with GDP-Mannose 4,6-Dehydratase
作者:
John G. Allen
;
Mirna Mujacic
;
Michael J. Frohn
;
Alex J. Pickrell
;
Paul Kodama
;
Dhanashri Bagal
;
Tisha San Miguel
;
E. Allen Sickmier
;
Steve Osgood
;
Aleksander Swietlow
;
Vivian Li
;
John B. Jordan
;
Ki-Won Kim
;
Anne-Marie C. Rousseau
;
Yong-Jae Kim
;
Seb Caille
;
Mike Achmatowicz
;
Oliver Thiel
;
Christopher
H.
Fotsch
;
Pranhitha Reddy
;
John D. McCarter
刊名:ACS Chemical Biology
出版年:2016
2.
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase–Glucokinase Regulatory Protein (GK–GKRP) Binding: Strategic Use of a N → S (nN → σ*S–X) Interaction fo
作者:
Lewis D. Pennington
;
Michael D. Bartberger
;
Michael D. Croghan
;
Kristin L. Andrews
;
Kate S. Ashton
;
Matthew P. Bourbeau
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Christopher
Fotsch
;
Joan Helmering
;
Fang-Tsao Hong
;
Randall W. Hungate
;
Steven R. Jordan
;
Ke Kong
;
Longbin Liu
;
Klaus Michelsen
;
Carolyn Moyer
;
Nobuko Nishimura
;
Mark H. Norman
;
Andreas Reichelt
;
Aaron C. Siegmund
;
Glenn Sivits
;
Seifu Tadesse
;
Christopher
M. Tegley
;
Gwyneth Van
;
Kevin C. Yang
;
Guomin Yao
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean Jr.
刊名:Journal of Medicinal Chemistry
出版年:2015
3.
Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis
作者:
Nuria A. Tamayo
;
Mark H. Norman
;
Michael D. Bartberger
;
Fang-Tsao Hong
;
Yunxin Bo
;
Longbin Liu
;
Nobuko Nishimura
;
Kevin C. Yang
;
Seifu Tadesse
;
Christopher
Fotsch
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Clarence Hale
;
Steven R. Jordan
;
David J. Lloyd
;
Glenn Sivits
;
Gwyneth Van
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Systematic Study of the Glutathione (GSH) Reactivity of N-Arylacrylamides: 1. Effects of Aryl Substitution
作者:
Victor J. Cee
;
Laurie P. Volak
;
Yuping Chen
;
Michael D. Bartberger
;
Chris Tegley
;
Tara Arvedson
;
John McCarter
;
Andrew S. Tasker
;
Christopher
Fotsch
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 3. Structure鈥揂ctivity Relationships within the Aryl Carbinol Region of the N-Arylsulfonamido-N鈥?a
作者:
Nobuko Nishimura
;
Mark H. Norman
;
Longbin Liu
;
Kevin C. Yang
;
Kate S. Ashton
;
Michael D. Bartberger
;
Samer Chmait
;
Jie Chen
;
Rod Cupples
;
Christopher
Fotsch
;
Joan Helmering
;
Steven R. Jordan
;
Roxanne K. Kunz
;
Lewis D. Pennington
;
Steve F. Poon
;
Aaron Siegmund
;
Glenn Sivits
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept
作者:
Kate S. Ashton
;
Kristin L. Andrews
;
Marion C. Bryan
;
Jie Chen
;
Kui Chen
;
Michelle Chen
;
Samer Chmait
;
Michael Croghan
;
Rod Cupples
;
Christopher
Fotsch
;
Joan Helmering
;
Steve R. Jordan
;
Robert J. M. Kurzeja
;
Klaus Michelsen
;
Lewis D. Pennington
;
Steve F. Poon
;
Glenn Sivits
;
Gwyneth Van
;
Steve L. Vonderfecht
;
Robert C. Wahl
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
7.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 2. Leveraging Structure-Based Drug Design to Identify Analogues with Improved Pharmacokinetic Profiles
作者:
David J. St. Jean
;
Jr.
;
Kate S. Ashton
;
Michael D. Bartberger
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Elizabeth Galbreath
;
Joan Helmering
;
Fang-Tsao Hong
;
Steven R. Jordan
;
Longbin Liu
;
Roxanne K. Kunz
;
Klaus Michelsen
;
Nobuko Nishimura
;
Lewis D. Pennington
;
Steve F. Poon
;
Darren Reid
;
Glenn Sivits
;
Markian M. Stec
;
Seifu Tadesse
;
Nuria Tamayo
;
Gwyneth Van
;
Kevin C. Yang
;
Jiandong Zhang
;
Mark H. Norman
;
Christopher
Fotsch
;
David J. Lloyd
;
Clarence Hale
刊名:Journal of Medicinal Chemistry
出版年:2014
8.
Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 4. Exploration of a Novel Binding Pocket
作者:
Fang-Tsao Hong
;
Mark H. Norman
;
Kate S. Ashton
;
Michael D. Bartberger
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Christopher
Fotsch
;
Steven R. Jordan
;
David J. Lloyd
;
Glenn Sivits
;
Seifu Tadesse
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
9.
Correction to Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept
作者:
Kate S. Ashton
;
Kristin L. Andrews
;
Marian C. Bryan
;
Jie Chen
;
Kui Chen
;
Michelle Chen
;
Samer Chmait
;
Michael Croghan
;
Rod Cupples
;
Christopher
Fotsch
;
Joan Helmering
;
Steve R. Jordan
;
Robert J. M. Kurzeja
;
Klaus Michelsen
;
Lewis D. Pennington
;
Steve F. Poon
;
Glenn Sivits
;
Gwyneth Van
;
Steve L. Vonderfecht
;
Robert C. Wahl
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
10.
Piperazine Oxadiazole Inhibitors of Acetyl-CoA Carboxylase
作者:
Matthew P. Bourbeau
;
Aaron Siegmund
;
John G. Allen
;
Hong Shu
;
Christopher
Fotsch
;
Michael D. Bartberger
;
Ki-Won Kim
;
Renee Komorowski
;
Melissa Graham
;
James Busby
;
Minghan Wang
;
James Meyer
;
Yang Xu
;
Kevin Salyers
;
Mark Fielden
;
Murielle M. Véniant
;
Wei Gu
刊名:Journal of Medicinal Chemistry
出版年:2013
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