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Elsevier电子期刊(10)
ACS电子期刊(8)
在“
ACS电子期刊
”中,
命中:
8
条,耗时:0.0299858 秒
在所有数据库中总计命中:
18
条
1.
8-Substituted Pyrido[3,4-d]pyri
m
idin-4(3H)-one Derivatives As Potent, Cell Per
m
eable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine De
m
ethylase Inhibitors
作者:
Vassilios Bavetsias
;
Rachel
M
. Lanigan
;
Gian Filippo Ruda
;
Butrus Atrash
;
M
ark G. McLaughlin
;
Anthony Tu
m
ber
;
N. Yi
M
ok
;
Yann-Vaï Le Bihan
;
Sally De
m
pster
;
Katherine J. Boxall
;
Fiona Jeganathan
;
Stephanie B. Hatch
;
Pavel Savitsky
;
Srikannathasan Velupillai
;
Tobias Krojer
;
Katherine S. England
;
Ji
mm
y Sejberg
;
Ching Thai
;
Ada
m
Donovan
;
Akos Pal
;
Giuseppe Scozzafava
;
Ja
m
es M. Bennett
;
Akane Kawa
m
ura
;
Catrine Johansson
;
Aleksandra Szykowska
;
Carina Gileadi
;
Nicola A. Burgess-Brown
;
Frank von Delft
;
Udo Opper
m
ann
;
Zoe Walters
;
Janet Shipley
;
Florence I. Raynaud
;
Susan
M
.
Westaway
;
Rab K. Prinjha
;
Oleg Fedorov
;
Rose
m
ary Burke
;
Christopher J. Schofield
;
Isaac
M
. Westwood
;
Chas Bountra
;
Susan
ne
M
üller
;
Rob L.
M
. van Montfort
;
Paul E. Brennan
;
Julian Blagg
刊名:Journal of
M
edicinal Che
m
istry
出版年:2016
2.
Cell Penetrant Inhibitors of the KD
M
4 and KDM5 Fa
m
ilies of Histone Lysine De
m
ethylases. 1. 3-A
m
ino-4-pyridine Carboxylate Derivatives
作者:
Susan
M
.
Westaway
;
Alex G. S. Preston
;
M
ichael D. Barker
;
Fiona Brown
;
Jack A. Brown
;
M
atthew Ca
m
pbell
;
Chun-wa Chung
;
Hawa Diallo
;
Cle
m
ent Douault
;
Gerard Drewes
;
Robert Eagle
;
Laurie Gordon
;
Carl Hasla
m
;
Tho
m
as G. Hayhow
;
Philip G. Hu
m
phreys
;
Gerard Joberty
;
Roy Katso
;
Laurens Kruidenier
;
M
elanie Leveridge
;
John Liddle
;
Julie
M
osley
;
M
arcel Muelbaier
;
Rebecca Randle
;
In
m
a Rioja
;
Anne Rueger
;
Gail A. Seal
;
Robert J. Sheppard
;
Onkar Singh
;
Joanna Taylor
;
Pa
m
ela Tho
m
as
;
Douglas Tho
m
son
;
David
M
. Wilson
;
Kevin Lee
;
Rab K. Prinjha
刊名:Journal of
M
edicinal Che
m
istry
出版年:2016
3.
Cell Penetrant Inhibitors of the KD
M
4 and KDM5 Fa
m
ilies of Histone Lysine De
m
ethylases. 2. Pyrido[3,4-d]pyri
m
idin-4(3H)-one Derivatives
作者:
Susan
M
.
Westaway
;
Alex G. S. Preston
;
M
ichael D. Barker
;
Fiona Brown
;
Jack A. Brown
;
M
atthew Ca
m
pbell
;
Chun-wa Chung
;
Gerard Drewes
;
Robert Eagle
;
Neil Garton
;
Laurie Gordon
;
Carl Hasla
m
;
Tho
m
as G. Hayhow
;
Philip G. Hu
m
phreys
;
Gerard Joberty
;
Roy Katso
;
Laurens Kruidenier
;
M
elanie Leveridge
;
M
ichelle Pe
m
berton
;
In
m
a Rioja
;
Gail A. Seal
;
Tracy Shipley
;
Onkar Singh
;
Colin J. Suckling
;
Joanna Taylor
;
Pa
m
ela Tho
m
as
;
David
M
. Wilson
;
Kevin Lee
;
Rab K. Prinjha
刊名:Journal of
M
edicinal Che
m
istry
出版年:2016
4.
Interrogating the Druggability of the 2-Oxoglutarate-Dependent Dioxygenase Target Class by Che
m
ical Proteo
m
ics
作者:
Gérard Joberty
;
M
arkus Boesche
;
Jack A. Brown
;
Dirk Eberhard
;
Neil S. Garton
;
Philip G. Hu
m
phreys
;
Toby
M
athieson
;
M
arcel Muelbaier
;
Nigel G. Ra
m
sden
;
Valérie Reader
;
Anne Rueger
;
Robert J. Sheppard
;
Susan
M
.
Westaway
;
M
arcus Bantscheff
;
Kevin Lee
;
David
M
. Wilson
;
Rab K. Prinjha
;
Gerard Drewes
刊名:ACS Che
m
ical Biology
出版年:2016
5.
Discovery of N-(3-Fluorophenyl)-1-[(4-([(3S)-3-
m
ethyl-1-piperazinyl]
m
ethyl)phenyl)acetyl]-4-piperidina
m
ine (GSK962040), the First S
m
all Molecule Motilin Receptor Agonist Clinical Candida
作者:
Susan
M
.
Westaway
*
†
;
;
Sa
m
antha L. Brown
†
;
;
Stephen C.
M
. Fell
†
;
;
Christopher N. Johnson
‡
;
;
David T.
M
acPherson
‡
;
;
Darren
刊名:Journal of
M
edicinal Che
m
istry
出版年:2009
6.
Deter
m
ining the Transition-State Structure for Different SN2 Reactions Using Experi
m
ental Nucleophile Carbon and Secondary α-Deuteriu
m
Kinetic Isotope Effects and Theory
作者:
Kenneth C.
Westaway
;
Yao-ren Fang
;
Susan
na
M
acMillar
;
Olle
M
atsson
;
Ray
m
ond A. Poirier
;
Shahidul
M
. Isla
m
刊名:Journal of Physical Che
m
istry A
出版年:2008
7.
A New Insight into Using Chlorine Leaving Group and Nucleophile Carbon Kinetic Isotope Effects To Deter
m
ine Substituent Effects on the Structure of SN2 Transition States
作者:
Kenneth C.
Westaway
;
Yao-ren Fang
;
Susan
na
M
acMillar
;
Olle
M
atsson
;
Ray
m
ond A. Poirier
;
Shahidul
M
. Isla
m
刊名:Journal of Physical Che
m
istry A
出版年:2007
8.
The Potential of Transient Receptor Potential Vanilloid Type 1 Channel
M
odulators for the Treat
m
ent of Pain
作者:
Susan
M
.
Westaway
刊名:Journal of
M
edicinal Che
m
istry
出版年:2007
1
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