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SpringerLink电子期刊(2)
Elsevier电子期刊(6)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:0.0309846 秒
在所有数据库中总计命中:
15
条
1.
Design and Synthesis of a Pan-Janus Kinase Inhibitor Clinical Candidate (PF-06263276) Suitable for Inhaled and Topical Delivery for the Treat
m
ent of Infla
mm
atory Diseases of the Lungs and Skin
作者:
Peter JonesR. Ian Storer
;
Yogesh A. Sabnis
;
Florian
M
. Wakenhut
;
Gavin A. Whitlock
;
Katherine S. England
;
Takasuke
M
ukaiya
m
a
;
Christoph
M
.
Dehnhardt
;
Jotha
m
W. Coe
;
Steve W. Kortu
m
;
Jill E. Chrencik
;
David G. Brown
;
Rhys
M
. Jones
;
John R.
M
urphy
;
Thean Yeoh
;
Paul
M
organ
;
Iain Kilty
刊名:Journal of
M
edicinal Che
m
istry
出版年:2017
2.
Discovery of Aryl Sulfona
m
ides as Isofor
m
-Selective Inhibitors of NaV1.7 with Efficacy in Rodent Pain Models
作者:
Thilo Focken
;
Shifeng Liu
;
Navjot Chahal
;
M
axi
m
Dauphinais
;
M
ichael E. Gri
m
wood
;
Sultan Chowdhury
;
Ivan He
m
eon
;
Paul Bichler
;
David Bogucki
;
M
atthew Waldbrook
;
Girish Bankar
;
Luis E. Sojo
;
Clint Young
;
Sophia Lin
;
Noah Shuart
;
Rainbow Kwan
;
Jodie Pang
;
Jae H. Chang
;
Brian S. Safina
;
Daniel P. Sutherlin
;
J. P. Johnson Jr.
;
Christoph
M
.
Dehnhardt
;
Tarek S.
M
ansour
;
Renata
M
. Oballa
;
Charles J. Cohen
;
C. Lee Robinette
刊名:ACS
M
edicinal Che
m
istry Letters
出版年:2016
3.
Synthesis and SAR of Novel 4-
M
orpholinopyrrolopyri
m
idine Derivatives as Potent Phosphatidylinositol 3-Kinase Inhibitors
作者:
Zecheng Chen
;
Aranapaka
m
M. Venkatesan
;
Christoph
M
.
Dehnhardt
;
Se
m
ira
m
is Ayral-Kaloustian
;
Natasja Brooij
m
ans
;
Robert
M
allon
;
Larry Feldberg
;
Irwin Hollander
;
Judy Lucas
;
Ker Yu
;
Fang
m
ing Kong
;
Tarek
刊名:Journal of
M
edicinal Che
m
istry
出版年:2010
4.
Design and Synthesis of Novel Dia
m
inoquinazolines with in Vivo Efficacy for β-Catenin/T-Cell Transcriptional Factor 4 Pathway Inhibition
作者:
Christoph
M
.
Dehnhardt
;
Aranapaka
m
M. Venkatesan
;
Zecheng Chen
;
Se
m
ira
m
is Ayral-Kaloustian
;
Osvaldo Dos Santos
;
Efren Delos Santos
;
Kevin Curran
;
M
ax T. Follettie
;
Veronica Diesl
;
Judy Lucas
;
Yi Geng
刊名:Journal of
M
edicinal Che
m
istry
出版年:2010
5.
Lead Opti
m
ization of N-3-Substituted 7-Morpholinotriazolopyri
m
idines as Dual Phosphoinositide 3-Kinase/Ma
mm
alian Target of Rapa
m
ycin Inhibitors: Discovery of PKI-402
作者:
Christoph
M
.
Dehnhardt
;
Aranapaka
m
M. Venkatesan
;
Efren Delos Santos
;
Zecheng Chen
;
Osvaldo Santos
;
Se
m
ira
m
is Ayral-Kaloustian
;
Natasja Brooij
m
ans
;
Robert
M
allon
;
Irwin Hollander
;
Larry Feldberg
;
Judy
刊名:Journal of
M
edicinal Che
m
istry
出版年:2010
6.
Bis(
m
orpholino-1,3,5-triazine) Derivatives: Potent Adenosine 5′-Triphosphate Co
m
petitive Phosphatidylinositol-3-kinase/Ma
mm
alian Target of Rapa
m
ycin Inhibitors: Discovery of Co
m
pound 26 (
作者:
Aranapaka
m
M. Venkatesan
;
Christoph
M
.
Dehnhardt
;
Efren Delos Santos
;
Zecheng Chen
;
Osvaldo Dos Santos
;
Se
m
ira
m
is Ayral-Kaloustian
;
Gulnaz Khafizova
;
Natasja Brooij
m
ans
;
Robert
M
allon
;
Irwin Hollander
刊名:Journal of
M
edicinal Che
m
istry
出版年:2010
7.
Stereoselective Synthesis of an Active
M
etabolite of the Potent PI3 Kinase Inhibitor PKI-179
作者:
Zecheng Chen
;
Aranapaka
m
M. Venkatesan
;
Osvaldo Dos Santos
;
Efren Delos Santos
;
Christoph
M
.
Dehnhardt
;
Se
m
ira
m
is Ayral-Kaloustian
;
Joseph Ashcroft
;
Leonard A.
M
cDonald
;
Tarek S.
M
ansour
刊名:Journal of Organic Che
m
istry
出版年:2010
1
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