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3.Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quino
6.Discovery and in Vivo Evaluation of (S)-N-(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and Related PI3K未 Inhibitors for Inflammation and Autoimmune
7.Discovery of AMG 925, a FLT3 and CDK4 Dual Kinase Inhibitor with Preferential Affinity for the Activated State of FLT3
作者:Zhihong Li ; Xianghong Wang ; John Eksterowicz ; Michael W. Gribble ; Jr. ; Grace Q. Alba ; Merrill Ayres ; Timothy J. Carlson ; Ada Chen ; Xiaoqi Chen ; Robert Cho ; Richard V. Connors ; Michael DeGraffenreid ; Jeffrey T. Deignan ; Jason Duquette ; Pingchen Fan ; Benjamin Fisher ; Jiasheng Fu ; Justin N. Huard ; Jacob Kaizerman ; Kathleen S. Keegan ; Cong Li ; Kexue Li ; Yunxiao Li ; Lingming Liang ; Wen Liu ; Sarah E. Lively ; Mei-Chu Lo ; Ji Ma ; Dustin L. McMinn ; Jeffrey T. Mihalic ; Kriti Modi ; Rachel Ngo ; Kanaka Pattabiraman ; Derek E. Piper ; Christophe Queva ; Mark L. Ragains ; Julia Suchomel ; Steve Thibault ; Nigel Walker ; Xiaodong Wang ; Zhulun Wang ; Malgorzata Wanska ; Paul M. Wehn ; Margaret F. Weidner ; Alex J. Zhang ; Xiaoning Zhao ; Alexander Kamb ; Dineli Wickramasinghe ; Kang Dai ; Lawrence R. McGee ; Julio C. Medina
刊名:Journal of Medicinal Chemistry
出版年:2014
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