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255
条
1.
Ch
e
mical and Computational M
e
thods for th
e
Charact
e
rization of Coval
e
nt R
e
activ
e
Groups for th
e
Prosp
e
ctiv
e
D
e
sign of Irr
e
v
e
rsibl
e
Inhibitors
作者:
Mark
E
.
Flanagan
;
Jos
e
ph A. Abramit
e
;
D
e
nnis P. And
e
rson
;
Ann Aulabaugh
;
Up
e
ndra P. Dahal
;
Adam M. Gilb
e
rt
;
Chao Li
;
Justin Montgom
e
ry
;
Stac
e
y R. Opp
e
nh
e
im
e
r
;
Tim Ryd
e
r
;
Brandon P. Schuff
;
Dani
e
l P. Ucc
e
llo
;
Gr
e
gory S. Walk
e
r
;
Yan Wu
;
Matth
e
w F. Brown
;
Jinshan M. Ch
e
n
;
Matth
e
w M. Hayward
;
Mark
C. No
e
;
R. Scott Obach
;
Laur
e
nc
e
Philipp
e
;
V
ee
rabahu Shanmugasundaram
;
Micha
e
l J. Shapiro
;
J
e
r
e
my Starr
;
Justin Stroh
;
Y
e
Ch
e
刊名:Journal of M
e
dicinal Ch
e
mistry
出版年:2014
2.
Discov
e
ry and D
e
v
e
lopm
e
nt of Janus Kinas
e
(JAK) Inhibitors for Inflammatory Dis
e
as
e
s
作者:
Jam
e
s D. Clark
;
Mark
E
.
Flanagan
;
J
e
an-Baptist
e
T
e
lli
e
z
刊名:Journal of M
e
dicinal Ch
e
mistry
出版年:2014
3.
Discov
e
ry of Dap-3 Polymyxin Analogu
e
s for th
e
Tr
e
atm
e
nt of Multidrug-R
e
sistant Gram-N
e
gativ
e
Nosocomial Inf
e
ctions
作者:
Thomas V. Mag
ee
;
Matth
e
w F. Brown
;
J
e
r
e
my T. Starr
;
David C. Ackl
e
y
;
Jos
e
ph A. Abramit
e
;
Jiri Aubr
e
cht
;
Andr
e
w Butl
e
r
;
Jar
e
d L. Crandon
;
Fadia Dib-Hajj
;
Mark
E
.
Flanagan
;
Karl Granskog
;
Jo
e
l R. Hardink
;
Micha
e
l D. Huband
;
R
e
b
e
cca Irvin
e
;
Micha
e
l Kuhn
;
Kar
e
n L. L
e
ach
;
Bryan Li
;
Jian Lin
;
David R. Luk
e
;
Shawn H. MacVan
e
;
Alita A. Mill
e
r
;
Sandra McCurdy
;
Jam
e
s M. McKim
;
Jr.
;
David P. Nicolau
;
Thuy-Trinh Nguy
e
n
;
Mark
C. No
e
;
John P. O鈥橠onn
e
ll
;
Scott B. S
e
ib
e
l
;
Yu
e
Sh
e
n
;
Antonia F. St
e
pan
;
Andr
e
w P. Tomaras
;
Paul C. Wilga
;
Li Zhang
;
Jinf
e
ng Xu
;
Jinshan Micha
e
l Ch
e
n
刊名:Journal of M
e
dicinal Ch
e
mistry
出版年:2013
4.
Proc
e
ss D
e
v
e
lopm
e
nt of a Nov
e
l Az
e
tidinyl K
e
tolid
e
Antibiotic
作者:
Bryan Li
;
Thomas V. Mag
ee
;
Richard A. Buzon
;
Dani
e
l W. Widlicka
;
Dav
e
R. Bill
;
Thomas Brandt
;
Xiaoping Cao
;
Micha
e
l Coutant
;
Haijian Dou
;
Karl Granskog
;
Mark
E
.
Flanagan
;
Ch
e
ryl M. Hayward
;
Bin Li
;
F
e
ngw
e
i Liu
;
W
e
i Liu
;
Thuy-Trinh Nguy
e
n
;
J
e
ffr
e
y W. Raggon
;
P
e
t
e
r Ros
e
;
Jos
e
ph Rainvill
e
;
Usa Datta R
e
illy
;
Yu
e
Sh
e
n
;
Jianmin Sun
;
Gl
e
nn E. Wilcox
刊名:Organic Proc
e
ss R
e
s
e
arch & D
e
v
e
lopm
e
nt
出版年:2012
5.
D
e
v
e
lopm
e
nt and Charact
e
rization of N
e
w Inhibitors of th
e
Human and Mous
e
H
e
matopoi
e
tic Prostaglandin D2 Synthas
e
s
作者:
Ang
e
lika N. Christ
;
Larisa Labzin
;
Gr
e
gory T. Bourn
e
;
Hirotada Fukunishi
;
Jan
e
E. W
e
b
e
r
;
Matth
e
w J. Sw
ee
t
;
Mark
L. Smyth
e
;
Jack U.
Flanagan
刊名:Journal of M
e
dicinal Ch
e
mistry
出版年:2010
6.
Discov
e
ry of CP-690,550: A Pot
e
nt and S
e
l
e
ctiv
e
Janus Kinas
e
(JAK) Inhibitor for th
e
Tr
e
atm
e
nt of Autoimmun
e
Dis
e
as
e
s and Organ Transplant R
e
j
e
ction
作者:
Mark
E
.
Flanagan
;
Todd A. Blum
e
nkopf
;
William H. Briss
e
tt
e
;
Matth
e
w F. Brown
;
J
e
ffr
e
y M. Casavant
;
Chang Shang-Poa
;
Jonathan L. Doty
;
E
il
ee
n A. Elliott
;
Micha
e
l B. Fish
e
r
;
Micha
e
l Hin
e
s
;
Craig K
e
nt
;
E
刊名:Journal of M
e
dicinal Ch
e
mistry
出版年:2010
7.
A Ligand-Fi
e
ld Analysis of th
e
tr
e
nsal (H3tr
e
nsal = 2,2',2' '-Tris(salicylid
e
n
e
imino)tri
e
thylamin
e
) Ligand. An Application of th
e
Angular Ov
e
rlap Mod
e
l to Lanthanid
e
s
作者:
B
e
rnadin
e
M.
Flanagan
;
Paul V. B
e
rnhardt
;
E
lmars R. Krausz
;
St
e
fan R. Lü
;
thi
;
and
Mark
J. Ril
e
y
刊名:Inorganic Ch
e
mistry
出版年:2002
8.
D
e
v
e
lopm
e
nt of a Scal
e
abl
e
Rout
e
for th
e
Production of cis-N-B
e
nzyl-3-m
e
thylamino-4-m
e
thylpip
e
ridin
e
作者:
David H. Brown Ripin
;
St
e
fan Ab
e
l
e
;
W
e
iling Cai
;
Todd Blum
e
nkopf
;
J
e
ffr
e
y M. Casavant
;
Jonathan L. Doty
;
Mark
Flanagan
;
Christian Ko
e
ch
e
r
;
Klaus W. Lau
e
;
K
e
ith McCarthy
;
Cliff M
e
ltz
;
Mik
e
Munchhoff
;
K
刊名:Organic Proc
e
ss R
e
s
e
arch & D
e
v
e
lopm
e
nt
出版年:2003
9.
M
e
chanistic Studi
e
s of an Antibody-Catalyz
e
d Elimination R
e
action
作者:
Floyd
E
. Rom
e
sb
e
rg
;
Mark
E
.
Flanagan
;
T
e
tsuo Uno
;
and P
e
t
e
r G. Schultz
刊名:Journal of th
e
Am
e
rican Ch
e
mical Soci
e
ty
出版年:1998
10.
Multipl
e
Int
e
ractions of th
e
Asp2.61(98) Sid
e
Chain of th
e
Gonadotropin-R
e
l
e
asing Hormon
e
R
e
c
e
ptor Contribut
e
Diff
e
r
e
ntially to Ligand Int
e
raction
作者:
Coll
ee
n A.
Flanagan
;
Vladimir Rodic
;
Kar
e
l Konvicka
;
Tony Yu
e
n
;
Ling Chi
;
J
e
an E. Rivi
e
r
;
Rob
e
rt P. Millar
;
Har
e
l W
e
inst
e
in
;
and Stuart C. S
e
alfon
刊名:Bioch
e
mistry
出版年:2000
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