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Wiley电子期刊(3)
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ACS电子期刊(45)
NATURE电子期刊(1)
Elsevier电子期刊(29)
在“
ACS电子期刊
”中,
命中:
45
条,耗时:0.0239872 秒
在所有数据库中总计命中:
79
条
1.
High-
T
hroughpu
t
Screening and Hi
t
Valida
t
ion of Ex
t
racellular-Rela
t
ed Kinase 5 (ERK5) Inhibi
t
ors
作者:
S
t
ephanie M. Myers
;
Ru
t
h H. Bawn
;
Louise C. Bisse
t
;
T
imo
t
hy J. Blackburn
;
Be
tt
y Co
tt
yn
;
Lauren Molyneux
;
Ai-Ching Wong
;
Celine Cano
;
William Clegg
;
Ross. W. Harring
t
on
;
Hing Leung
;
Lauren
t
Rigoreau
;
Sandrine Vido
t
;
Bernard
T
.
Golding
;
Roger J. Griffin
;
T
im Hammonds
;
David R. Newell
;
Ian R. Hardcas
t
le
刊名:ACS Combina
t
orial Science
出版年:2016
2.
8-Subs
t
i
t
u
t
ed O6-Cyclohexylme
t
hylguanine CDK2 Inhibi
t
ors: Using S
t
ruc
t
ure-Based Inhibi
t
or Design
t
o Op
t
imize an Al
t
erna
t
ive Binding Mode
作者:
Benoi
t
Carbain
;
David J. Pa
t
erson
;
Elizabe
t
h Anscombe
;
Allyson J. Campbell
;
Celine Cano
;
Aude Echalier
;
Jane A. Endico
tt
;
Bernard
T
.
Golding
;
Karen Hagger
t
y
;
Ian R. Hardcas
t
le
;
Philip J. Jewsbury
;
David R. Newell
;
Mar
t
in E. M. Noble
;
Celine Roche
;
Lan Z. Wang
;
Roger J. Griffin
刊名:Journal of Medicinal Chemis
t
ry
出版年:2014
3.
Nucleoside
T
ranspor
t
Inhibi
t
ors: S
t
ruc
t
ure鈭扐c
t
ivi
t
y Rela
t
ionships for Pyrimido[5,4-d]pyrimidine Deriva
t
ives Tha
t
Po
t
en
t
ia
t
e Peme
t
rexed Cy
t
o
t
oxici
t
y in
t
he Presence of 伪1-Acid Glycopr
作者:
Kappusamy Saravanan
;
Hannah C. Barlow
;
Marion Bar
t
on
;
A. Hilary Calver
t
;
Bernard
T
.
Golding
;
David R. Newell
;
Julian S. Nor
t
hen
;
Nicola J. Cur
t
in
;
Huw D.
T
homas
;
Roger J. Griffin
刊名:Journal of Medicinal Chemis
t
ry
出版年:2011
4.
1-Subs
t
i
t
u
t
ed (Dibenzo[b,d]
t
hiophen-4-yl)-2-morpholino-4H-chromen-4-ones Endowed wi
t
h Dual DNA-PK/PI3-K Inhibi
t
ory Ac
t
ivi
t
y
作者:
C茅line Cano
;
Kappusamy Saravanan
;
Chris Bailey
;
Julia Bardos
;
Nicola J. Cur
t
in
;
Mark Frigerio
;
Bernard
T
.
Golding
;
Ian R. Hardcas
t
le
;
Marc G. Hummersone
;
Kei
t
h A. Menear
;
David R. Newell
;
Caroline J. Richardson
;
K. Shea
;
Graeme C. M. Smi
t
h
;
Pia
T
hommes
;
A
tt
illa Ting
;
Roger J. Griffin
刊名:Journal of Medicinal Chemis
t
ry
出版年:2013
5.
Isoindolinone Inhibi
t
ors of
t
he Murine Double Minu
t
e 2 (MDM2)-p53 Pro
t
ein鈭扨ro
t
ein In
t
erac
t
ion: S
t
ruc
t
ure鈭扐c
t
ivi
t
y S
t
udies Leading
t
o Improved Po
t
ency
作者:
Ian R. Hardcas
t
le
;
Junfeng Liu
;
Eric Valeur
;
Anna Wa
t
son
;
Shafiq U. Ahmed
;
T
imo
t
hy J. Blackburn
;
Karim Bennaceur
;
William Clegg
;
Ca
t
herine Drummond
;
Jane A. Endico
tt
;
Bernard
T
.
Golding
;
Roger J. Griffin
;
Jan Gruber
;
Karen Hagger
t
y
;
Ross W. Harring
t
on
;
Claire Hu
tt
on
;
S
t
uar
t
Kemp
;
Xiaohong Lu
;
James M. McDonnell
;
David R. Newell
;
Mar
t
in E. M. Noble
;
Sara L. Payne
;
Charlo
tt
e H. Revill
;
Chris
t
iane Riedinger
;
Qing Xu
;
John Lunec
刊名:Journal of Medicinal Chemis
t
ry
出版年:2011
6.
Iden
t
ifica
t
ion and Charac
t
eriza
t
ion of 2鈥?Deoxyadenosine Adduc
t
s Formed by Isoprene Monoepoxides in Vi
t
ro
作者:
Pe
t
ra Begemann
;
Gunnar Boysen
;
Nadia I. Georgieva
;
Ramiah Sangaiah
;
Karl M. Koshlap
;
Hasan Koc
;
Daping Zhang
;
Bernard
T
.
Golding
;
Avram Gold
;
James A. Swenberg
刊名:Chemical Research in
T
oxicology
出版年:2011
7.
DNA-Dependen
t
Pro
t
ein Kinase (DNA-PK) Inhibi
t
ors. Syn
t
hesis and Biological Ac
t
ivi
t
y of Quinolin-4-one and Pyridopyrimidin-4-one Surroga
t
es for
t
he Chromen-4-one Chemo
t
ype
作者:
Cline Cano
;
Olivier R. Barbeau
;
Chris
t
ine Bailey
;
Xiao-Ling Cockcrof
t
;
Nicola J. Cur
t
in
;
Hea
t
her Duggan
;
Mark Frigerio
;
Bernard
T
.
Golding
;
Ian R. Hardcas
t
le
;
Marc G. Hummersone
;
Charlo
tt
e Knigh
t
s
;
Ke
刊名:Journal of Medicinal Chemis
t
ry
出版年:2010
8.
Cob(I)alamin for
T
rapping Bu
t
adiene Epoxides in Me
t
abolism wi
t
h Ra
t
S9 and for De
t
ermining Associa
t
ed Kine
t
ic Parame
t
ers
作者:
Hi
t
esh V. Mo
t
wani
;
Charlo
tt
a Fred
;
Johanna Haglund
;
Bernard
T
.
Golding
;
Margare
t
a Trnqvis
t
刊名:Chemical Research in
T
oxicology
出版年:2009
9.
Mechanism of Enzyma
t
ic Birch Reduc
t
ion: S
t
ereochemical Course and Exchange Reac
t
ions of Benzoyl-CoA Reduc
t
ase
作者:
Bä
;
rbel
T
hiele
;
Oliver Rieder
;
Bernard
T
.
Golding
;
Michael Mü
;
ller
;
Ma
tt
hias Boll
刊名:Journal of
t
he American Chemical Socie
t
y
出版年:2008
10.
Analysis of Chemical Shif
t
Changes Reveals
t
he Binding Modes of Isoindolinone Inhibi
t
ors of
t
he MDM2-p53 In
t
erac
t
ion
作者:
Chris
t
iane Riedinger
;
Jane A. Endico
tt
;
S
t
uar
t
J. Kemp
;
Lyne
tt
e A. Smy
t
h
;
Anna Wa
t
son
;
Eric Valeur
;
Bernard
T
.
Golding
;
Roger J. Griffin
;
Ian R. Hardcas
t
le
;
Mar
t
in E. Noble
;
James M. McDonnell
刊名:Journal of
t
he American Chemical Socie
t
y
出版年:2008
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