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SpringerLink电子期刊(2)
NATURE电子期刊(7)
Elsevier电子期刊(10)
ACS电子期刊(15)
在“
ACS电子期刊
”中,
命中:
15
条,耗时:小于0.01 秒
在所有数据库中总计命中:
34
条
1.
Discovery and Preclinical Characterization of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577), a Direct Activator of Adenosine Monophosphate-activated Protein Kinase (AMPK), for the Potential Treatment of Diabetic Nephropathy
作者:
Kimberly O. Cameron
;
Daniel W. Kung
;
Amit S. Kalgutkar
;
Ravi G. Kurumbail
;
Russell Miller
;
Christopher T. Salatto
;
Jessica Ward
;
Jane M. Withka
;
Samit K. Bhattacharya
;
Markus Boehm
;
Kris A. Borzilleri
;
Janice A. Brown
;
Matthew Calabrese
;
Nicole L. Caspers
;
Emily Cokorinos
;
Edward L. Conn
;
Matthew S. Dowling
;
David
J. Edmonds
;
Heather Eng
;
Dilinie P. Fernando
;
Richard Frisbie
;
David
Hepworth
;
James Landro
;
Yuxia Mao
;
Francis Rajamohan
;
Allan R. Reyes
;
Colin R. Rose
;
Tim Ryder
;
Andre Shavnya
;
Aaron C. Smith
;
Meihua Tu
;
Angela C. Wolford
;
Jun Xiao
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of an in Vivo Tool to Establish Proof-of-Concept for MAP4K4-Based Antidiabetic Treatment
作者:
Mark Ammirati
;
Scott W. Bagley
;
Samit K. Bhattacharya
;
Leonard Buckbinder
;
Anthony A. Carlo
;
Rebecca Conrad
;
Christian Cortes
;
Robert L. Dow
;
Matthew S. Dowling
;
Ayman El-Kattan
;
Kristen Ford
;
Cristiano R. W. Guimar茫es
;
David
Hepworth
;
Wenhua Jiao
;
Jennifer LaPerle
;
Shenping Liu
;
Allyn Londregan
;
Paula M. Loria
;
Alan M. Mathiowetz
;
Michael Munchhof
;
Suvi T. M. Orr
;
Donna N. Petersen
;
David
A. Price
;
Athanasia Skoura
;
Aaron C. Smith
;
Jian Wang
刊名:ACS Medicinal Chemistry Letters
出版年:2015
3.
Evaluation and Synthesis of Polar Aryl- and Heteroaryl Spiroazetidine-Piperidine Acetamides as Ghrelin Inverse Agonists
作者:
Suvi T. M. Orr
;
Ramsay Beveridge
;
Samit K. Bhattacharya
;
Kimberly O. Cameron
;
Steven Coffey
;
Dilinie Fernando
;
David
Hepworth
;
Margaret V. Jackson
;
Vishal Khot
;
Rachel Kosa
;
Kimberly Lapham
;
Paula M. Loria
;
Kim F. McClure
;
Jigna Patel
;
Colin Rose
;
James Saenz
;
Ingrid A. Stock
;
Gregory Storer
;
Maria von Volkenburg
;
Derek Vrieze
;
Guoqiang Wang
;
Jun Xiao
;
Yingxin Zhang
刊名:ACS Medicinal Chemistry Letters
出版年:2015
4.
Discovery of 2-(6-(5-Chloro-2-methoxyphenyl)-4-oxo-2-thioxo-3,4-dihydropyrimidin-1(2H)-yl)acetamide (PF-06282999): A Highly Selective Mechanism-Based Myeloperoxidase Inhibitor for the Treatment of Car
作者:
Roger B. Ruggeri
;
Leonard Buckbinder
;
Scott W. Bagley
;
Philip A. Carpino
;
Edward L. Conn
;
Matthew S. Dowling
;
Dilinie P. Fernando
;
Wenhua Jiao
;
Daniel W. Kung
;
Suvi T. M. Orr
;
Yingmei Qi
;
Benjamin N. Rocke
;
Aaron Smith
;
Joseph S. Warmus
;
Yan Zhang
;
Daniel Bowles
;
Daniel W. Widlicka
;
Heather Eng
;
Tim Ryder
;
Raman Sharma
;
Angela Wolford
;
Carlin Okerberg
;
Karen Walters
;
Tristan S. Maurer
;
Yanwei Zhang
;
Paul D. Bonin
;
Samantha N. Spath
;
Gang Xing
;
David
Hepworth
;
Kay Ahn
;
Amit S. Kalgutkar
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Discovery and Optimization of Imidazopyridine-Based Inhibitors of Diacylglycerol Acyltransferase 2 (DGAT2)
作者:
Kentaro Futatsugi
;
Daniel W. Kung
;
Suvi T. M. Orr
;
Shawn Cabral
;
David
Hepworth
;
Gary Aspnes
;
Scott Bader
;
Jianwei Bian
;
Markus Boehm
;
Philip A. Carpino
;
Steven B. Coffey
;
Matthew S. Dowling
;
Michael Herr
;
Wenhua Jiao
;
Sophie Y. Lavergne
;
Qifang Li
;
Ronald W. Clark
;
Derek M. Erion
;
Kou Kou
;
Kyuha Lee
;
Brandon A. Pabst
;
Sylvie M. Perez
;
Julie Purkal
;
Csilla C. Jorgensen
;
Theunis C. Goosen
;
James R. Gosset
;
Mark Niosi
;
John C. Pettersen
;
Jeffrey A. Pfefferkorn
;
Kay Ahn
;
Bryan Goodwin
刊名:Journal of Medicinal Chemistry
出版年:2015
6.
Discovery of Selective Small Molecule Inhibitors of Monoacylglycerol Acyltransferase 3
作者:
Kim Huard
;
Allyn T. Londregan
;
Gregory Tesz
;
Kevin B. Bahnck
;
Thomas V. Magee
;
David
Hepworth
;
Jana Polivkova
;
Steven B. Coffey
;
Brandon A. Pabst
;
James R. Gosset
;
Anu Nigam
;
Kou Kou
;
Hao Sun
;
Kyuha Lee
;
Michael Herr
;
Markus Boehm
;
Philip A. Carpino
;
Bryan Goodwin
;
Christian Perreault
;
Qifang Li
;
Csilla C. Jorgensen
;
George T. Tkalcevic
;
Timothy A. Subashi
;
Kay Ahn
刊名:Journal of Medicinal Chemistry
出版年:2015
7.
Identification of (R)-6-(1-(4-Cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro-1H-pyrazol-3-yl)-2-methoxynicotinic Acid, a Highly Potent and Selective Nonsteroidal Mineralocorticoid Recep
作者:
Agustin Casimiro-Garcia
;
David
W. Piotrowski
;
Catherine Ambler
;
Graciela B. Arhancet
;
Mary Ellen Banker
;
Tereece Banks
;
Carine M. Boustany-Kari
;
Cuiman Cai
;
Xiangyang Chen
;
Rena Eudy
;
David
Hepworth
;
Catherine A. Hulford
;
Sandra M. Jennings
;
Paula M. Loria
;
Marvin J. Meyers
;
Donna N. Petersen
;
Neil K. Raheja
;
Matthew Sammons
;
Li She
;
Kun Song
;
Derek Vrieze
;
Liuqing Wei
刊名:Journal of Medicinal Chemistry
出版年:2014
8.
Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate
作者:
Samit K. Bhattacharya
;
Kim Andrews
;
Ramsay Beveridge
;
Kimberly O. Cameron
;
Chiliu Chen
;
Matthew Dunn
;
Dilinie Fernando
;
Hua Gao
;
David
Hepworth
;
V. Margaret Jackson
;
Vishal Khot
;
Jimmy Kong
;
Rachel E. Kosa
;
Kimberly Lapham
;
Paula M. Loria
;
Allyn T. Londregan
;
Kim F. McClure
;
Suvi T. M. Orr
;
Jigna Patel
;
Colin Rose
;
James Saenz
;
Ingrid A. Stock
;
Gregory Storer
;
Maria VanVolkenburg
;
Derek Vrieze
;
Guoqiang Wang
;
Jun Xiao
;
Yingxin Zhang
刊名:ACS Medicinal Chemistry Letters
出版年:2014
9.
Identification of Tetrahydropyrido[4,3-d]pyrimidine Amides as a New Class of Orally Bioavailable TGR5 Agonists
作者:
David
W. Piotrowski
;
Kentaro Futatsugi
;
Joseph S. Warmus
;
Suvi T. M. Orr
;
Kevin D. Freeman-Cook
;
Allyn T. Londregan
;
Liuqing Wei
;
Sandra M. Jennings
;
Michael Herr
;
Steven B. Coffey
;
Wenhua Jiao
;
Gregory Storer
;
David
Hepworth
;
Jian Wang
;
Sophie Y. Lavergne
;
Janice E. Chin
;
John R. Hadcock
;
Martin B. Brenner
;
Angela C. Wolford
;
Ann M. Janssen
;
Nicole S. Roush
;
Joanne Buxton
;
Terri Hinchey
;
Amit S. Kalgutkar
;
Raman Sharma
;
Declan A. Flynn
刊名:ACS Medicinal Chemistry Letters
出版年:2013
10.
Chemical Probe Identification Platform for Orphan GPCRs Using Focused Compound Screening: GPR39 as a Case Example
作者:
Markus Boehm
;
David
Hepworth
;
Paula M. Loria
;
Lisa D. Norquay
;
Kevin J. Filipski
;
Janice E. Chin
;
Kimberly O. Cameron
;
Martin Brenner
;
Peter Bonnette
;
Shawn Cabral
;
Edward Conn
;
David
C. Ebner
;
Denise Gautreau
;
John Hadcock
;
Esther C. Y. Lee
;
Alan M. Mathiowetz
;
Michelle Morin
;
Lucy Rogers
;
Aaron Smith
;
Maria VanVolkenburg
;
Philip A. Carpino
刊名:ACS Medicinal Chemistry Letters
出版年:2013
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