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SpringerLink电子期刊(15)
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ACS电子期刊(24)
NATURE电子期刊(13)
Elsevier电子期刊(43)
在“
ACS电子期刊
”中,
命中:
24
条,耗时:小于0.01 秒
在所有数据库中总计命中:
97
条
1.
Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor
作者:
Nicholas D. Measom
;
Kenneth D. Down
;
David J. HirstCraig Jamieson
;
Eric S. Manas
;
Vipulkumar K. Patel
;
Don
O.
Somers
刊名:ACS Medicinal Chemistry Letters
出版年:2017
2.
Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors
作者:
Hongfeng Deng
;
Jingye Zhou
;
Flora Sundersingh
;
Jeffrey A. Messer
;
Don
ald O.
Somers
;
Myriam Ajakane
;
Christopher C. Arico-Muendel
;
Arthur Beljean
;
Svetlana L. Belyanskaya
;
Ryan Bingham
;
Emily Blazensky
;
Anne-Benedicte Boullay
;
Eric Boursier
;
Jing Chai
;
Paul Carter
;
Chun-Wa Chung
;
Alain Daugan
;
Yun Ding
;
Kenny Herry
;
Clare Hobbs
;
Eric Humphries
;
Christopher Kollmann
;
Van Loc Nguyen
;
Edwige Nicodeme
;
Sarah E. Smith
;
Nerina Dodic
;
Nicolas Ancellin
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
CSAR 2014: A Benchmark Exercise Using Unpublished Data from Pharma
作者:
Heather A. Carlson
;
Richard D. Smith
;
Kelly L. Damm-Ganamet
;
Jeanne A. Stuckey
;
Aqeel Ahmed
;
Maire A. Convery
;
Don
ald O.
Somers
;
Michael Kranz
;
Patricia A. Elkins
;
Guanglei Cui
;
Catherine E. Peishoff
;
Millard H. Lambert
;
James B. Dunbar Jr.
刊名:Journal of Chemical Information and Modeling
出版年:2016
4.
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening
作者:
Alison J.-A. Woolford
;
Joseph E. Pero
;
Sridhar Aravapalli
;
Valerio Berdini
;
Joseph E. Coyle
;
Philip J. Day
;
Andrew M. Dodson
;
Pascal Grondin
;
Finn P. Holding
;
Lydia Y. W. Lee
;
Peng Li
;
Eric S. Manas
;
Joseph Marino Jr.
;
Agnes C. L. Martin
;
Brent W. McCleland
;
Rachel L. McMenamin
;
Christopher W. Murray
;
Christopher E. Neipp
;
Lee W. Page
;
Vipulkumar K. Patel
;
Florent Potvain
;
Sharna Rich
;
Ralph A. Rivero
;
Kirsten Smith
;
Don
ald O.
Somers
;
Lionel Trottet
;
Ranganadh Velagaleti
;
Glyn Williams
;
Ren Xie
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Structurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment Screening
作者:
Jennifer A. Borthwick
;
Nicolas Ancellin
;
Sophie M. Bertrand
;
Ryan P. Bingham
;
Paul S. Carter
;
Chun-wa Chung
;
Ian Churcher
;
Nerina Dodic
;
Charlène Fournier
;
Peter L. Francis
;
Andrew Hobbs
;
Craig Jamieson
;
Stephen D. Pickett
;
Sarah E. Smith
;
Don
ald O’N.
Somers
;
Claus Spitzfaden
;
Colin J. Suckling
;
Robert J. Young
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)
作者:
Alison J.-A. Woolford
;
Philip J. Day
;
Véronique Bénéton
;
Valerio Berdini
;
Joseph E. Coyle
;
Yann Dudit
;
Pascal Grondin
;
Pascal Huet
;
Lydia Y. W. Lee
;
Eric S. Manas
;
Rachel L. McMenamin
;
Christopher W. Murray
;
Lee W. Page
;
Vipulkumar K. Patel
;
Florent Potvain
;
Sharna J. Rich
;
Yingxia Sang
;
Don
O.
Somers
;
Lionel Trottet
;
Zehong Wan
;
Xiaomin Zhang
刊名:Journal of Medicinal Chemistry
出版年:2016
7.
Discovery, SAR, and X-ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library
作者:
Hongfeng Deng
;
Jingye Zhou
;
Flora S. Sundersingh
;
Jennifer Summerfield
;
Don
Somers
;
Jeffrey A. Messer
;
Alexander L. Satz
;
Nicolas Ancellin
;
Christopher C. Arico-Muendel
;
Katie L. (Sargent) Bedard
;
Arthur Beljean
;
Svetlana L. Belyanskaya
;
Ryan Bingham
;
Sarah E. Smith
;
Eric Boursier
;
Paul Carter
;
Paolo A. Centrella
;
Matthew A. Clark
;
Chun-wa Chung
;
Christopher P. Davie
;
Jennifer L. Delorey
;
Yun Ding
;
G. Joseph Franklin
;
LaShadric C. Grady
;
Kenny Herry
;
Clare Hobbs
;
Christopher S. Kollmann
;
Barry A. Morgan
;
Laura J. (Pothier) Kaushansky
;
Quan Zhou
刊名:ACS Medicinal Chemistry Letters
出版年:2015
8.
The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits
作者:
Sophie M. Bertrand
;
Nicolas Ancellin
;
Benjamin Beaufils
;
Ryan P. Bingham
;
Jennifer A. Borthwick
;
Anne-B茅n茅dicte Boullay
;
Eric Boursier
;
Paul S. Carter
;
Chun-wa Chung
;
Ian Churcher
;
Nerina Dodic
;
Marie-H茅l猫ne Fouchet
;
Charl猫ne Fournier
;
Peter L. Francis
;
Laura A. Gummer
;
Kenny Herry
;
Andrew Hobbs
;
Clare I. Hobbs
;
Paul Homes
;
Craig Jamieson
;
Edwige Nicodeme
;
Stephen D. Pickett
;
Iain H. Reid
;
Graham L. Simpson
;
Lisa A. Sloan
;
Sarah E. Smith
;
Don
ald O鈥橬.
Somers
;
Claus Spitzfaden
;
Colin J. Suckling
;
Klara Valko
;
Yoshiaki Washio
;
Robert J. Young
刊名:Journal of Medicinal Chemistry
出版年:2015
9.
Chiral Conjugated Corrals
作者:
Melissa Ball
;
Bran
don
Fowler
;
Panpan Li
;
Leo A. Joyce
;
Fang Li
;
Taifeng Liu
;
Daniel Paley
;
Yu Zhong
;
Hexing Li
;
Shengxiong Xiao
;
Fay Ng
;
Michael L. Steigerwald
;
Colin Nuckolls
刊名:Journal of the American Chemical Society
出版年:2015
10.
Spin I
somers
and Ligand Isomerization in a Three-Coordinate Cobalt(I) Carbonyl Complex
作者:
Malik H. Al-Afyouni
;
Elizaveta Suturina
;
Shubhrodeep Pathak
;
Mihail Atanasov
;
Eckhard Bill
;
Daniel E. DeRosha
;
William W. Brennessel
;
Frank Neese
;
Patrick L. Holland
刊名:Journal of the American Chemical Society
出版年:2015
1
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