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ACS电子期刊(38)
在“
ACS电子期刊
”中,
命中:
38
条,耗时:0.0189921 秒
在所有数据库中总计命中:
1,098
条
1.
Discovery of VU0409551/
J
NJ-46778212: An mGlu5 Positive Allosteric Modulator Clinical Candidate Targeting Schizophrenia
作者:
Susana Conde-Ceide
;
Carlos M. Mart铆nez-Viturro
;
J
es煤s Alc谩zar
;
Pedro M. Garcia-Barrantes
;
Hilde Lavreysen
;
Claire Mackie
;
Paige N. Vinson
;
J
erri M. Rook
;
Thomas M. Bridges
;
J
.
Scott
Daniels
;
Anton Megens
;
Xavier Langlois
;
Wilhelmus H. Drinkenburg
;
Abdellah Ahnaou
;
Colleen M. Niswender
;
Carrie K.
J
ones
;
Gregor
J
. Macdonald
;
Thomas Steckler
;
P.
J
effrey Conn
;
Shaun R. Stauffer
;
J
os茅 Manuel Bartolom茅-Nebreda
;
Craig W. Lindsley
刊名:ACS Medicinal Chemistry Letters
出版年:2015
2.
Discovery, Synthesis, and Preclinical Characterization of N-(3-Chloro-4-fluorophenyl)-1H-pyrazolo[4,3-b]pyridin-3-amine (VU0418506), a Novel Positive Allosteric Modulator of the Metabotropic Glutamate Receptor 4 (mGlu4)
作者:
Darren W. Engers
;
Anna L. Blobaum
;
Rocco D. Gogliotti
;
Yiu-Yin Cheung
;
J
ames M. Salovich
;
Pedro M. Garcia-Barrantes
;
J
.
Scott
Daniels
;
Ryan Morrison
;
Carrie K.
J
ones
;
Matthew G. Soars
;
Xiaoliang Zhuo
;
J
eremy Hurley
;
J
ohn E. Macor
;
J
oanne J. Bronson
;
P.
J
effrey Conn
;
Craig W. Lindsley
;
Colleen M. Niswender
;
Corey R. Hopkins
刊名:ACS Chemical Neuroscience
出版年:2016
3.
Development and Antiparkinsonian Activity of VU0418506, a Selective Positive Allosteric Modulator of Metabotropic Glutamate Receptor 4 Homomers without Activity at mGlu2/4 Heteromers
作者:
Colleen M. Niswender
;
Carrie K.
J
ones
;
Xin Lin
;
Michael Bubser
;
Analisa Thompson Gray
;
Anna L. Blobaum
;
Darren W. Engers
;
Alice L. Rodriguez
;
Matthew T. Loch
;
J
.
Scott
Daniels
;
Craig W. Lindsley
;
Corey R. Hopkins
;
J
onathan A. Javitch
;
P.
J
effrey Conn
刊名:ACS Chemical Neuroscience
出版年:2016
4.
Lack of Antiparkinsonian Effects of Systemic In
j
ections of the Specific T-Type Calcium Channel Blocker ML218 in MPTP-Treated Monkeys
作者:
Adriana Galvan
;
Annaelle Devergnas
;
Damien Pittard
;
Gunasingh Masilamoni
;
J
ocelyn Vuong
;
J
.
Scott
Daniels
;
Ryan D. Morrison
;
Craig W. Lindsley
;
Thomas Wichmann
刊名:ACS Chemical Neuroscience
出版年:2016
5.
Identification and Characterization of ML352: A Novel, Noncompetitive Inhibitor of the Presynaptic Choline Transporter
作者:
Elizabeth A. Ennis
;
J
ane Wright
;
Cassandra L. Retzlaff
;
Owen B. McManus
;
Zhinong Lin
;
Xiaofang Huang
;
Meng Wu
;
Min Li
;
J
.
Scott
Daniels
;
Craig W. Lindsley
;
Corey R. Hopkins
;
Randy D. Blakely
刊名:ACS Chemical Neuroscience
出版年:2015
6.
Brooktrout Lake Case Study: Biotic Recovery from Acid Deposition 20 Years after the 1990 Clean Air Act Amendments
作者:
J
ames W. Sutherland
;
Frank W. Acker
;
J
ay A. Bloomfield
;
Charles W. Boylen
;
Donald F. Charles
;
Robert A.
Daniels
;
Lawrence W. Eichler
;
J
eremy L. Farrell
;
Robert S. Feranec
;
Matthew P. Hare
;
Sharon L. Kanfoush
;
Richard
J
. Preall
;
Scott
O. Quinn
;
H. Chandler Rowell
;
William F. Schoch
;
William H. Shaw
;
Clifford A. Siegfried
;
Timothy
J
. Sullivan
;
David A. Winkler
;
Sandra A. Nierzwicki-Bauer
刊名:Environmental Science & Technology
出版年:2015
7.
Design of 4-Oxo-1-aryl-1,4-dihydroquinoline-3-carboxamides as Selective Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 2
作者:
Andrew S. Felts
;
Alice L. Rodriguez
;
Katrina A. Smith
;
J
ulie L. Engers
;
Ryan D. Morrison
;
Frank W. Byers
;
Anna L. Blobaum
;
Charles W. Locuson
;
Sichen Chang
;
Daryl F. Venable
;
Colleen M. Niswender
;
J
.
Scott
Daniels
;
P.
J
effrey Conn
;
Craig W. Lindsley
;
Kyle A. Emmitte
刊名:
J
ournal of Medicinal Chemistry
出版年:2015
8.
Discovery of a Selective and CNS Penetrant Negative Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 3 with Antidepressant and Anxiolytic Activity in Rodents
作者:
J
ulie L. Engers
;
Alice L. Rodriguez
;
Leah C. Konkol
;
Ryan D. Morrison
;
Analisa D. Thompson
;
Frank W. Byers
;
Anna L. Blobaum
;
Sichen Chang
;
Daryl F. Venable
;
Matthew T. Loch
;
Colleen M. Niswender
;
J
.
Scott
Daniels
;
Carrie K.
J
ones
;
P.
J
effrey Conn
;
Craig W. Lindsley
;
Kyle A. Emmitte
刊名:
J
ournal of Medicinal Chemistry
出版年:2015
9.
Selective Activation of M4 Muscarinic Acetylcholine Receptors Reverses MK-801-Induced Behavioral Impairments and Enhances Associative Learning in Rodents
作者:
Michael Bubser
;
Thomas M. Bridges
;
Ditte Dencker
;
Robert W. Gould
;
Michael Grannan
;
Meredith
J
. Noetzel
;
Atin Lamsal
;
Colleen M. Niswender
;
J
.
Scott
Daniels
;
Michael S. Poslusney
;
Bruce
J
. Melancon
;
J
ames C. Tarr
;
Frank W. Byers
;
J
眉rgen Wess
;
Mark E. Duggan
;
J
ohn Dunlop
;
Michael W. Wood
;
Nicholas
J
. Brandon
;
Michael R. Wood
;
Craig W. Lindsley
;
P.
J
effrey Conn
;
Carrie K.
J
ones
刊名:ACS Chemical Neuroscience
出版年:2014
10.
Tetrahydronaphthyridine and Dihydronaphthyridinone Ethers As Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 5 (mGlu5)
作者:
Mark Turlington
;
Chrysa Malosh
;
J
on Jacobs
;
J
ason T. Manka
;
Meredith
J
. Noetzel
;
Paige N. Vinson
;
Satyawan
J
adhav
;
Elizabeth
J
. Herman
;
Hilde Lavreysen
;
Claire Mackie
;
J
os茅 M. Bartolom茅-Nebreda
;
Susana Conde-Ceide
;
M. Luz Mart铆n-Mart铆n
;
Han Min Tong
;
Silvia L贸pez
;
Gregor
J
. MacDonald
;
Thomas Steckler
;
J
.
Scott
Daniels
;
C. David Weaver
;
Colleen M. Niswender
;
Carrie K.
J
ones
;
P.
J
effrey Conn
;
Craig W. Lindsley
;
Shaun R. Stauffer
刊名:
J
ournal of Medicinal Chemistry
出版年:2014
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