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SpringerLink电子期刊(1)
NATURE电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(11)
在“
ACS电子期刊
”中,
命中:
11
条,耗时:小于0.01 秒
在所有数据库中总计命中:
23
条
1.
Discovery of a Potent Acyclic, Tripeptidic, Acyl Sulfonamide Inhibitor of Hepatitis C Virus NS3 Protease as a Back-up to Asunaprevir with the Potential for Once-Daily Dosing
作者:
Li-Qiang Sun
;
Eric Mull
;
Barbara Zheng
;
Stanley D’Andrea
;
Qian Zhao
;
Alan Xiangdong Wang
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Jie Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Arvind Mathur
;
Richard Rampulla
;
Bang-Chi Chen
;
Theerthagiri Palani
;
Sivakumar Ganesan
;
Pirama Nayagam Arunachalam
;
Paul Falk
;
Steven Levine
;
Chaoqun Chen
;
Jacques Friborg
;
Fei Yu
;
Dennis Hernandez
;
Amy K. Sheaffer
;
Jay
O.
Knipe
;
Yong-Hae Han
;
Richard Schartman
;
Maria Donoso
;
Kathy Mosure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Kevin Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Gao
;
Alicia Ng
;
Luciano Mueller
;
Dennis M. Grasela
;
Stephen Adams
;
James Loy
;
Paul C. Levesque
;
Huabin Sun
;
Hong Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jialong Zhu
;
Ying-Kai Wang
;
Hua Fang
;
Mark I. Cockett
;
Nicholas A. Meanwell
;
Fiona McPhee
;
Paul M. Scola
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Hepatitis C Virus NS5A Replication Complex Inhibitors. Part 6: Discovery of a Novel and Highly Potent Biarylimidazole Chemotype with Inhibitory Activity Toward Genotypes 1a and 1b Replicons
作者:
Makonen Belema
;
Van N. Nguyen
;
Jeffrey L. Romine
;
Denis R. St. Laurent
;
Omar D. Lopez
;
Jason T. Goodrich
;
Peter T. Nower
;
Donald R. O鈥橞oyle
;
II
;
Julie A. Lemm
;
Robert A. Fridell
;
Min Gao
;
Hua Fang
;
Rudolph G. Krause
;
Ying-Kai Wang
;
A.
Jay
ne Oliver
;
Andrew C. Good
;
Jay
O.
Knipe
;
Nicholas A. Meanwell
;
Lawrence B. Snyder
刊名:Journal of Medicinal Chemistry
出版年:2014
3.
Discovery and Early Clinical Evaluation of BMS-605339, a Potent and Orally Efficacious Tripeptidic Acylsulfonamide NS3 Protease Inhibitor for the Treatment of Hepatitis C Virus Infection
作者:
Paul M. Scola
;
Alan Xiangdong Wang
;
Andrew C. Good
;
Li-Qiang Sun
;
Keith D. Combrink
;
Jeffrey A. Campbell
;
Jie Chen
;
Yong Tu
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Stanley D鈥橝ndrea
;
Barbara Zheng
;
Piyasena Hewawasam
;
Min Ding
;
Jan Thuring
;
Jianqing Li
;
Dennis Hernandez
;
Fei Yu
;
Paul Falk
;
Guangzhi Zhai
;
Amy K. Sheaffer
;
Chaoqun Chen
;
Min S. Lee
;
Diana Barry
;
Jay
O.
Knipe
;
Wenying Li
;
Yong-Hae Han
;
Susan Jenkins
;
Christoph Gesenberg
;
Qi Gao
;
Michael W. Sinz
;
Kenneth S. Santone
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Herbert E. Klei
;
Richard J. Colonno
;
Dennis M. Grasela
;
Eric Hughes
;
Caly Chien
;
Stephen Adams
;
Paul C. Levesque
;
Danshi Li
;
Jialong Zhu
;
Nicholas A. Meanwell
;
Fiona McPhee
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase
作者:
Robert G. Gentles
;
Min Ding
;
John A. Bender
;
Carl P. Bergstrom
;
Katharine Grant-Young
;
Piyasena Hewawasam
;
Thomas Hudyma
;
Scott Martin
;
Andrew Nickel
;
Alicia Regueiro-Ren
;
Yong Tu
;
Zhong Yang
;
Kap-Sun Yeung
;
Xiaofan Zheng
;
Sam Chao
;
Jung-Hui Sun
;
Brett R. Beno
;
Daniel M. Camac
;
Chong-Hwan Chang
;
Mian Gao
;
Paul E. Morin
;
Steven Sheriff
;
Jeff Tredup
;
John Wan
;
Mark R. Witmer
;
Dianlin Xie
;
Umesh Hanumegowda
;
Jay
Knipe
;
Kathy Mosure
;
Kenneth S. Santone
;
Dawn D. Parker
;
Xiaoliang Zhuo
;
Julie Lemm
;
Mengping Liu
;
Lenore Pelosi
;
Karen Rigat
;
Stacey Voss
;
Yi Wang
;
Ying-Kai Wang
;
Richard J. Colonno
;
Min Gao
;
Susan B. Roberts
;
Qi Gao
;
Alicia Ng
;
Nicholas A Meanwell
;
John F. Kadow
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
The Discovery of Asunaprevir (BMS-650032), An Orally Efficacious NS3 Protease Inhibitor for the Treatment of Hepatitis C Virus Infection
作者:
Paul M. Scola
;
Li-Qiang Sun
;
Alan Xiangdong Wang
;
Jie Chen
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Stanley V. D鈥橝ndrea
;
Barbara Zheng
;
Piyasena Hewawasam
;
Yong Tu
;
Jacques Friborg
;
Paul Falk
;
Dennis Hernandez
;
Steven Levine
;
Chaoqun Chen
;
Fei Yu
;
Amy K. Sheaffer
;
Guangzhi Zhai
;
Diana Barry
;
Jay
O.
Knipe
;
Yong-Hae Han
;
Richard Schartman
;
Maria Donoso
;
Kathy Mosure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Andrew C. Good
;
Ramkumar Rajamani
;
Kevin Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Gao
;
Luciano Mueller
;
Richard J. Colonno
;
Dennis M. Grasela
;
Stephen P. Adams
;
James Loy
;
Paul C. Levesque
;
Huabin Sun
;
Hong Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jialong Zhu
;
Nicholas A. Meanwell
;
Fiona McPhee
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
Hepatitis C Virus NS5A Replication Complex Inhibitors: The Discovery of Daclatasvir
作者:
Makonen Belema
;
Van N. Nguyen
;
Carol Bachand
;
Dan H. Deon
;
Jason T. Goodrich
;
Clint A. James
;
Rico Lavoie
;
Omar D. Lopez
;
Alain Martel
;
Jeffrey L. Romine
;
Edward H. Ruediger
;
Lawrence B. Snyder
;
Denis R. St. Laurent
;
Fukang Yang
;
Juliang Zhu
;
Henry S. Wong
;
David R. Langley
;
Stephen P. Adams
;
Glenn H. Cantor
;
Anjaneya Chimalakonda
;
Aberra Fura
;
Benjamin M. Johnson
;
Jay
O.
Knipe
;
Dawn D. Parker
;
Kenneth S. Santone
;
Robert A. Fridell
;
Julie A. Lemm
;
Donald R. O鈥橞oyle
;
II
;
Richard J. Colonno
;
Min Gao
;
Nicholas A. Meanwell
;
Lawrence G. Hamann
刊名:Journal of Medicinal Chemistry
出版年:2014
7.
Cathepsin B-Labile Dipeptide Linkers for Lysosomal Release of Doxorubicin from Internalizing Immunoconjugates: Model Studies of Enzymatic Drug Release and Antigen-Specific In Vitro Anticancer Activity
作者:
Gene M. Dubowchik
;
Raymond A. Firestone
;
Linda Padilla
;
David Willner
;
Sandra J. Hofstead
;
Kathleen Mosure
;
Jay
O.
Knipe
;
Shirley J. Lasch
;
and Pamela A. Trail
刊名:Bioconjugate Chemistry
出版年:2002
8.
New hydrazone derivatives of Adriamycin and their immunoconjugates - a correlation between acid stability and cytotoxicity
作者:
Takushi Kaneko
;
David Willner
;
Ivo Monkovic
;
Jay
O.
Knipe
;
Gary R. Braslawsky
;
Robert S. Greenfield
;
and Dolatrai M. Vyas
刊名:Bioconjugate Chemistry
出版年:1991
9.
Methylase models: studies on general-base vs. nucleophilic catalysis in the intramolecular alkylation of phenols
作者:
Jay
O.
Knipe
;
Peter J. Vasquez
;
and James K. Coward
刊名:Journal of the American Chemical Society
出版年:1982
10.
Role of buffers in a methylase model reaction. General base catalysis by oxyanions vs. nucleophilic dealkylation by amines
作者:
Jay
O.
Knipe
and James K. Coward
刊名:Journal of the American Chemical Society
出版年:1979
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