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内部出版物
SpringerLink电子期刊(4)
NATURE电子期刊(1)
Elsevier电子期刊(12)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
24
条
1.
Discovery of (S)-1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development
作者:
James F. Blake
;
Michael
Burkard
;
Jocelyn Chan
;
Huifen Chen
;
Kang-Jye Chou
;
Dolores Diaz
;
Danette A. Dudley
;
John J. Gaudino
;
Stephen E. Gould
;
Jonas Grina
;
Thomas Hunsaker
;
Lichuan Liu
;
Matthew Martinson
;
David Moreno
;
Lars Mueller
;
Christine Orr
;
Patricia Pacheco
;
Ann Qin
;
Kevin Rasor
;
Li Ren
;
Kirk Robarge
;
Sheerin Shahidi-Latham
;
Jeffrey Stults
;
Francis Sullivan
;
Weiru Wang
;
Jianping Yin
;
Aihe Zhou
;
Marcia Belvin
;
Mark Merchant
;
John Moffat
;
Jacob B. Schwarz
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Diastereoseletive Transannular Oxa-Conjugate Addition Generates the 2,6-cis-Disubstituted Tetrahydropyran of Neopeltolide
作者:
Taylor P. A. Hari
;
Burkard
t I. Wilke
;
James A. Davey
;
Christopher N. Boddy
刊名:Journal of Organic Chemistry
出版年:2016
3.
A Feasible Way to Remove the Heat during Adsorptive Methane Storage
作者:
Stefan G眉tlein
;
Christoph
Burkard
;
Johannes Zeilinger
;
Matthias Niedermaier
;
Michael
Klumpp
;
Veronika Kolb
;
Andreas Jess
;
Bastian J. M. Etzold
刊名:Environmental Science & Technology
出版年:2015
4.
Discovery of Highly Potent, Selective, and Efficacious Small Molecule Inhibitors of ERK1/2
作者:
Li Ren
;
Jonas Grina
;
David Moreno
;
James F. Blake
;
John J. Gaudino
;
Rustam Garrey
;
Andrew T. Metcalf
;
Michael
Burkard
;
Matthew Martinson
;
Kevin Rasor
;
Huifen Chen
;
Brian Dean
;
Stephen E. Gould
;
Patricia Pacheco
;
Sheerin Shahidi-Latham
;
Jianping Yin
;
Kristina West
;
Weiru Wang
;
John G. Moffat
;
Jacob B. Schwarz
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Discovery of 7-Tetrahydropyran-2-yl Chromans: β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors That Reduce Amyloid β-Protein (Aβ) in the Central Nervous System
作者:
Allen A. Thomas
;
Kevin W. Hunt
;
Matthew Volgraf
;
Ryan J. Watts
;
Xingrong Liu
;
Guy Vigers
;
Darin Smith
;
Douglas Sammond
;
Tony P. Tang
;
Susan P. Rhodes
;
Andrew T. Metcalf
;
Karin D. Brown
;
Jennifer N. Otten
;
Michael
Burkard
;
April A. Cox
;
Mary K. Geck Do
;
Darrin Dutcher
;
Sumeet Rana
;
Robert K. DeLisle
;
Kelly Regal
;
Albion D. Wright
;
Robert Groneberg
;
Kimberly Scearce-Levie
;
Michael
Siu
;
Hans E. Purkey
;
Joseph P. Lyssikatos
;
Indrani W. Gunawardana
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
8-Tetrahydropyran-2-yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors
作者:
Allen A. Thomas
;
Kevin W. Hunt
;
Brad Newhouse
;
Ryan J. Watts
;
Xingrong Liu
;
Guy Vigers
;
Darin Smith
;
Susan P. Rhodes
;
Karin D. Brown
;
Jennifer N. Otten
;
Michael
Burkard
;
April A. Cox
;
Mary K. Geck Do
;
Darrin Dutcher
;
Sumeet Rana
;
Robert K. DeLisle
;
Kelly Regal
;
Albion D. Wright
;
Robert Groneberg
;
Jiangpeng Liao
;
Kimberly Scearce-Levie
;
Michael
Siu
;
Hans E. Purkey
;
Joseph P. Lyssikatos
刊名:Journal of Medicinal Chemistry
出版年:2014
7.
Spirocyclic 尾-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors: From Hit to Lowering of Cerebrospinal Fluid (CSF) Amyloid 尾 in a Higher Species
作者:
Kevin W. Hunt
;
Adam W. Cook
;
Ryan J. Watts
;
Christopher T. Clark
;
Guy Vigers
;
Darin Smith
;
Andrew T. Metcalf
;
Indrani W. Gunawardana
;
Michael
Burkard
;
April A. Cox
;
Mary K. Geck Do
;
Darrin Dutcher
;
Allen A. Thomas
;
Sumeet Rana
;
Nicholas C. Kallan
;
Robert K. DeLisle
;
James P. Rizzi
;
Kelly Regal
;
Douglas Sammond
;
Robert Groneberg
;
Michael
Siu
;
Hans Purkey
;
Joseph P. Lyssikatos
;
Allison Marlow
;
Xingrong Liu
;
Tony P. Tang
刊名:Journal of Medicinal Chemistry
出版年:2013
1
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