设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Wiley电子期刊(3)
GSW全文库(4)
Elsevier电子期刊(4)
ACS电子期刊(6)
在“
ACS电子期刊
”中,
命中:
6
条,耗时:小于0.01 秒
在所有数据库中总计命中:
17
条
1.
Discovery of 1-{(3R,4R)-3-[({5-Chloro-2-[(1-methyl-1H-pyrazol-4-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing, Irreversible Inhibitor of T790M-Containing EGFR Mutants
作者:
Hengmiao Cheng
;
Sajiv K. Nair
;
Brion W. Murray
;
Chau Almaden
;
Simon Bailey
;
Sangita Baxi
;
Doug Behenna
;
Sujin Cho-Schultz
;
Deepak Dalvie
;
Dac M. Dinh
;
Martin P. Edwards
;
Jun Li Feng
;
Rose Ann Ferre
;
Ketan S. Gajiwala
;
Michelle D. Hemkens
;
Amy Jackson-Fisher
;
Mehran Jalaie
;
Ted O. Johnson
;
Robert S. Kania
;
Susan Kephart
;
Jennifer Lafontaine
;
Beth Lunney
;
Kevin K.-C. Liu
;
Zhengyu Liu
;
Jean Matthews
;
Asako Nagata
;
Sherry Niessen
;
Martha A. Ornelas
;
Suvi T. M. Orr
;
Mason Pairish
;
Simon Planken
;
Shijian Ren
;
Daniel Richter
;
Kevin Ryan
;
Neal Sach
;
Hong Shen
;
Tod Smeal
;
Jim Solowiej
;
Scott Sutton
;
Khanh Tran
;
Elaine Tseng
;
William Vernier
;
Marlena Walls
;
Shuiwang Wang
;
Scott L. Weinrich
;
Shuibo Xin
;
Haiwei Xu
;
Min-Jean Yin
;
Michael
Zientek
;
Ru Zhou
;
John C. Kath
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of the Highly Potent PI3K/mTOR Dual Inhibitor PF-04979064 through Structure-Based Drug Design
作者:
Hengmiao Cheng
;
Chunze Li
;
Simon Bailey
;
Sangita M. Baxi
;
Lance Goulet
;
Lisa Guo
;
Jacqui Hoffman
;
Ying Jiang
;
Theodore Otto Johnson
;
Ted W. Johnson
;
Daniel R. Knighton
;
John Li
;
Kevin K.-C. Liu
;
Zhengyu Liu
;
Matthew A. Marx
;
Marlena Walls
;
Peter A. Wells
;
Min-Jean Yin
;
Jinjiang Zhu
;
Michael
Zientek
刊名:ACS Medicinal Chemistry Letters
出版年:2013
3.
Dihydroxyphenylisoindoline Amides as Orally Bioavailable Inhibitors of the Heat Shock Protein 90 (Hsp90) Molecular Chaperone
作者:
Pei-Pei Kung
;
Buwen Huang
;
Gang Zhang
;
Joe Zhongxiang Zhou
;
Jeff Wang
;
Jennifer A. Digits
;
Judith Skaptason
;
Shinji Yamazaki
;
David Neul
;
Michael
Zientek
;
Jeff Elleraas
;
Pramod Mehta
;
Min-Jean Yin
;
Mi
刊名:Journal of Medicinal Chemistry
出版年:2010
4.
Integrated in Silico−in Vitro Strategy for Addressing Cytochrome P450 3A4 Time-Dependent Inhibition
作者:
Michael
Zientek
;
Chad Stoner
;
Robyn Ayscue
;
Jacquelyn Klug-McLeod
;
Ying Jiang
;
Michael
West
;
Claire Collins
;
Sean Ekins
刊名:Chemical Research in Toxicology
出版年:2010
5.
Characterization of Cytochrome P450-Mediated Bioactivation of a Compound Containing the Chemical Scaffold, 4,5-Dihydropyrazole-1-carboxylic acid-(4-chlorophenyl amide), to a Chemically Reactive p
作者:
Hao Chen
;
Michael
Zientek
;
Mehran Jalaie
;
Yanhua Zhang
;
Christopher Bigge
;
Abdul Mutlib
刊名:Chemical Research in Toxicology
出版年:2009
6.
Effect of Intestinal Glucuronidation in Limiting Hepatic Exposure and Bioactivation of Raloxifene in Humans and Rats
作者:
Deepak Dalvie
;
Ping Kang
;
Michael
Zientek
;
Cathie Xiang
;
Sue Zhou
;
R. Scott Obach
刊名:Chemical Research in Toxicology
出版年:2008
1
按检索点细分(6)
题名(6)
按出版年细分(6)
2016年(1)
2013年(1)
2010年(2)
2009年(1)
2008年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.