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Wiley电子期刊(2)
NATURE电子期刊(1)
ACS电子期刊(16)
SpringerLink电子期刊(4)
Elsevier电子期刊(43)
在“
ACS电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
66
条
1.
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials
作者:
T. G. Murali Dhar
;
Hai-Yun Xiao
;
Jenny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurng Wu
;
Marta Dabros
;
Xiaoxia Yang
;
Tracy L. Taylor
;
Xia D. Zhou
;
Elizabeth M. Heimrich
;
Rochelle Thomas
;
Kim W. McIntyre
;
Bethanne Warrack
;
Hong Shi
;
Paul C. Levesque
;
Jia L. Zhu
;
James Hennan
;
Praveen Balimane
;
Zheng Yang
;
Anthony M. Marino
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Arvind
Mathur
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
An Efficient Scale-Up Synthesis of BMS-520, a Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
作者:
Xiaoping Hou
;
Juliang Zhu
;
Bang-Chi Chen
;
Scott H. Watterson
;
William J. Pitts
;
Alaric J. Dyckman
;
Percy H. Carter
;
Arvind
Mathur
;
Huiping Zhang
刊名:Organic Process Research & Development
出版年:2016
3.
Regioselective Synthesis of Substituted 4-Alkylamino and 4-Arylaminophthalazin-1(2H)-ones
作者:
Subramaniam Krishnananthan
;
Daniel Smith
;
Dauh-Rurng Wu
;
Shiuhang Yip
;
Prashantha Gunaga
;
Arvind
Mathur
;
Jianqing Li
刊名:Journal of Organic Chemistry
出版年:2016
4.
Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator
作者:
Michael G. YangZili Xiao
;
T. G. Murali Dhar
;
Hai-Yun Xiao
;
John L. Gilmore
;
David Marcoux
;
Jenny H. Xie
;
Kim W. McIntyre
;
Tracy L. Taylor
;
Virna Borowski
;
Elizabeth Heimrich
;
Yu-Wen Li
;
Jianlin Feng
;
Alda Fernandes
;
Zheng Yang
;
Praveen Balimane
;
Anthony M. Marino
;
Georgia Cornelius
;
Bethanne M. Warrack
;
Arvind
Mathur
;
Dauh-Rurng Wu
;
Peng Li
;
Anuradha Gupta
;
Bala Pragalathan
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Lois D. Lehman-McKeeman
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked
作者:
Scott H. Watterson
;
George V. De Lucca
;
Qing Shi
;
Charles M. Langevine
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Hua Gong
;
Jun Dai
;
Shiuhang Yip
;
Peng Li
;
Dawn Sun
;
Dauh-Rurng Wu
;
Chunlei Wang
;
Yingru Zhang
;
Sarah C. Traeger
;
Mark A. Pattoli
;
Stacey Skala
;
Lihong Cheng
;
Mary T. Obermeier
;
Rodney Vickery
;
Lorell N. Discenza
;
Celia J. D’Arienzo
;
Yifan Zhang
;
Elizabeth Heimrich
;
Kathleen M. Gillooly
;
Tracy L. Taylor
;
Claudine Pulicicchio
;
Kim W. McIntyre
;
Michael A. Galella
;
Andy J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing Chang
;
Richard Rampulla
;
Arvind
Mathur
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Aberra Fura
;
James R. Burke
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Small Molecule Reversible Inhibitors of Bruton’s Tyrosine Kinase (BTK): Structure–Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177)
作者:
George V. De Lucca
;
Qing Shi
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Rick Rampulla
;
Arvind
Mathur
;
Lorell Discenza
;
Celia D’Arienzo
;
Jun Dai
;
Mary Obermeier
;
Rodney Vickery
;
Yingru Zhang
;
Zheng Yang
;
Punit Marathe
;
Andrew J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing J. Chang
;
Huiping Zhang
;
Kathleen Gillooly
;
Tracy Taylor
;
Mark A. Pattoli
;
Stacey Skala
;
Daniel W. Kukral
;
Kim W. McIntyre
;
Luisa Salter-Cid
;
Aberra Fura
;
James R. Burke
;
Joel C. Barrish
;
Percy H. Carter
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
7.
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
作者:
Hai-Yun Xiao
;
Scott H. Watterson
;
Charles M. Langevine
;
Anurag S. Srivastava
;
Soo S. Ko
;
Yanlei Zhang
;
Robert J. Cherney
;
Wei-Wei Guo
;
John L. Gilmore
;
James E. Sheppeck II
;
Dauh-Rurng Wu
;
Peng Li
;
Duraisamy Ramasamy
;
Piramanayagam Arunachalam
;
Arvind
Mathur
;
Tracy L. Taylor
;
David J. Shuster
;
Kim W. McIntyre
;
Ding-Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Anthony M. Marino
;
Praveen V. Balimane
;
Zheng Yang
;
Dana M. Banas
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Bethanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Salter-Cid
;
Jenny Xie
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
;
T. G. Murali Dhar
刊名:Journal of Medicinal Chemistry
出版年:2016
8.
Crystallization-Induced Dynamic Resolution toward the Synthesis of (S)-7-Amino-5H,7H-dibenzo[b,d]-azepin-6-one: An Important Scaffold for γ-Secretase Inhibitors
作者:
Sukhen Karmakar
;
Vijay Byri
;
Ashvinikumar V. Gavai
;
Richard Rampulla
;
Arvind
Mathur
;
Anuradha Gupta
刊名:Organic Process Research & Development
出版年:2016
9.
Discovery of a Potent Acyclic, Tripeptidic, Acyl Sulfonamide Inhibitor of Hepatitis C Virus NS3 Protease as a Back-up to Asunaprevir with the Potential for Once-Daily Dosing
作者:
Li-Qiang Sun
;
Eric Mull
;
Barbara Zheng
;
Stanley D’Andrea
;
Qian Zhao
;
Alan Xiangdong Wang
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Jie Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Arvind
Mathur
;
Richard Rampulla
;
Bang-Chi Chen
;
Theerthagiri Palani
;
Sivakumar Ganesan
;
Pirama Nayagam Arunachalam
;
Paul Falk
;
Steven Levine
;
Chaoqun Chen
;
Jacques Friborg
;
Fei Yu
;
Dennis Hernandez
;
Amy K. Sheaffer
;
Jay O. Knipe
;
Yong-Hae Han
;
Richard Schartman
;
Maria Donoso
;
Kathy Mosure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Kevin Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Gao
;
Alicia Ng
;
Luciano Mueller
;
Dennis M. Grasela
;
Stephen Adams
;
James Loy
;
Paul C. Levesque
;
Huabin Sun
;
Hong Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jialong Zhu
;
Ying-Kai Wang
;
Hua Fang
;
Mark I. Cockett
;
Nicholas A. Meanwell
;
Fiona McPhee
;
Paul M. Scola
刊名:Journal of Medicinal Chemistry
出版年:2016
10.
Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors
作者:
Ashvinikumar V. Gavai
;
Claude Quesnelle
;
Derek Norris
;
Wen-Ching Han
;
Patrice Gill
;
Weifang Shan
;
Aaron Balog
;
Ke Chen
;
Andrew Tebben
;
Richard Rampulla
;
Dauh-Rurng Wu
;
Yingru Zhang
;
Arvind
Mathur
;
Ronald White
;
Anne Rose
;
Haiqing Wang
;
Zheng Yang
;
Asoka Ranasinghe
;
Celia D鈥橝rienzo
;
Victor Guarino
;
Lan Xiao
;
Ching Su
;
Gerry Everlof
;
Vinod Arora
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Krista Menard
;
Mei-Li Wen
;
Jere Meredith
;
George Trainor
;
Louis J. Lombardo
;
Richard Olson
;
Phil S. Baran
;
John T. Hunt
;
Gregory D. Vite
;
Bruce S. Fischer
;
Richard A. Westhouse
;
Francis Y. Lee
刊名:ACS Medicinal Chemistry Letters
出版年:2015
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