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SpringerLink电子期刊(2)
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Elsevier电子期刊(3)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
16
条
1.
Chemically Diverse Group I p21-Activated Kinase (PAK) Inhibitors Impart Acute Cardiovascular Toxicity with a Narrow Therapeutic Window
作者:
Joachim Rudolph
;
Lesley J. Murray
;
Chudi O. Ndubaku
;
Thomas O’Brien
;
Elizabeth Blackwood
;
Weiru Wang
;
Ignacio
Aliagas
;
Lewis Gazzard
;
James J. Crawford
;
Joy Drobnick
;
Wendy Lee
;
Xianrui Zhao
;
Klaus P. Hoeflich
;
David A. Favor
;
Ping Dong
;
Haiming Zhang
;
Christopher E. Heise
;
Angela Oh
;
Christy C. Ong
;
Hank La
;
Paroma Chakravarty
;
Connie Chan
;
Diana Jakubiak
;
Jennifer Epler
;
Sreemathy Ramaswamy
;
Roxanne Vega
;
Gary Cain
;
Dolores Diaz
;
Yu Zhong
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pKa Polar Moiety
作者:
Chudi O. Ndubaku
;
James J. Crawford
;
Joy Drobnick
;
Ignacio
Aliagas
;
David Campbell
;
Ping Dong
;
Laura M. Dornan
;
Sergio Duron
;
Jennifer Epler
;
Lewis Gazzard
;
Christopher E. Heise
;
Klaus P. Hoeflich
;
Diana Jakubiak
;
Hank La
;
Wendy Lee
;
Baiwei Lin
;
Joseph P. Lyssikatos
;
Jasna Maksimoska
;
Ronen Marmorstein
;
Lesley J. Murray
;
Thomas O鈥橞rien
;
Angela Oh
;
Sreemathy Ramaswamy
;
Weiru Wang
;
Xianrui Zhao
;
Yu Zhong
;
Elizabeth Blackwood
;
Joachim Rudolph
刊名:ACS Medicinal Chemistry Letters
出版年:2015
3.
Leveraging the Pre-DFG Residue Thr-406 To Obtain High Kinase Selectivity in an Aminopyrazole-Type PAK1 Inhibitor Series
作者:
Joachim Rudolph
;
Ignacio
Aliagas
;
James J. Crawford
;
Simon Mathieu
;
Wendy Lee
;
Qi Chao
;
Ping Dong
;
Lionel Rouge
;
Weiru Wang
;
Christopher Heise
;
Lesley J. Murray
;
Hank La
;
Yanzhou Liu
;
Gerard Manning
;
Fran莽ois Diederich
;
Klaus P. Hoeflich
刊名:ACS Medicinal Chemistry Letters
出版年:2015
4.
Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors
作者:
James J. Crawford
;
Wendy Lee
;
Ignacio
Aliagas
;
Simon Mathieu
;
Klaus P. Hoeflich
;
Wei Zhou
;
Weiru Wang
;
Lionel Rouge
;
Lesley Murray
;
Hank La
;
Ning Liu
;
Peter W. Fan
;
Jonathan Cheong
;
Christopher E. Heise
;
Sreemathy Ramaswamy
;
Robert Mintzer
;
Yanzhou Liu
;
Qi Chao
;
Joachim Rudolph
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Physicochemical and DMPK In Silico Models: Facilitating Their Use by Medicinal Chemists
作者:
Daniel F. Ortwine
;
Ignacio
Aliagas
刊名:Molecular Pharmaceutics
出版年:2013
6.
Identification of C-2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2
作者:
Mark Zak
;
Christopher A. Hurley
;
Stuart I. Ward
;
Philippe Bergeron
;
Kathy Barrett
;
Mercedesz Balazs
;
Wade S. Blair
;
Richard Bull
;
Paroma Chakravarty
;
Christine Chang
;
Peter Crackett
;
Gauri Deshmukh
;
Jason DeVoss
;
Peter S. Dragovich
;
Charles Eigenbrot
;
Charles Ellwood
;
Simon Gaines
;
Nico Ghilardi
;
Paul Gibbons
;
Stefan Gradl
;
Peter Gribling
;
Chris Hamman
;
Eric Harstad
;
Peter Hewitt
;
Adam Johnson
;
Tony Johnson
;
Jane R. Kenny
;
Michael F. T. Koehler
;
Pawan Bir Kohli
;
Sharada Labadie
;
Wyne P. Lee
;
Jiangpeng Liao
;
Marya Liimatta
;
Rohan Mendonca
;
Raman Narukulla
;
Rebecca Pulk
;
Austin Reeve
;
Scott Savage
;
Steven Shia
;
Micah Steffek
;
Savita Ubhayakar
;
Anne van Abbema
;
Ignacio
Aliagas
;
Barbara Avitabile-Woo
;
Yisong Xiao
;
Jing Yang
;
Janusz J. Kulagowski
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Potent and Selective Aminopyrimidine-Based B-Raf Inhibitors with Favorable Physicochemical and Pharmacokinetic Properties
作者:
Simon Mathieu
;
Stefan N. Gradl
;
Li Ren
;
Zhaoyang Wen
;
Ignacio
Aliagas
;
Janet Gunzner-Toste
;
Wendy Lee
;
Rebecca Pulk
;
Guiling Zhao
;
Bruno Alicke
;
Jason W. Boggs
;
Alex J. Buckmelter
;
Edna F. Choo
;
Victoria Dinkel
;
Susan L. Gloor
;
Stephen E. Gould
;
Joshua D. Hansen
;
Gregg Hastings
;
Georgia Hatzivassiliou
;
Ellen R. Laird
;
David Moreno
;
Yingqing Ran
;
Walter C. Voegtli
;
Steve Wenglowsky
;
Jonas Grina
;
Joachim Rudolph
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
DEGAS: Sharing and Tracking Target Compound Ideas with External Collaborators
作者:
Man-Ling Lee
;
Ignacio
Aliagas
;
Jennafer Dotson
;
Jianwen A. Feng
;
Alberto Gobbi
;
Timothy Heffron
刊名:Journal of Chemical Information and Modeling
出版年:2012
9.
Formation of a Quinoneimine Intermediate of 4-Fluoro-N-methylaniline by FMO1: Carbon Oxidation Plus Defluorination
作者:
James P. Driscoll
;
Ignacio
Aliagas
;
Jennifer J. Harris
;
Jason S. Halladay
;
Sheerin Khatib-Shahidi
;
Alan Deese
;
Nathaniel Segraves
;
S. Cyrus Khojasteh-Bakht
刊名:Chemical Research in Toxicology
出版年:2010
10.
A Class of 2,4-Bisanilinopyrimidine Aurora A Inhibitors with Unusually High Selectivity against Aurora B
作者:
Ignacio
Aliagas
-Martin
;
Dan Burdick
;
Laura Corson
;
Jennafer Dotson
;
Jason Drummond
;
Carter Fields
;
Oscar W. Huang
;
Thomas Hunsaker
;
Tracy Kleinheinz
;
Elaine Krueger
;
Jun Liang
;
John Moffat
;
Gail Phill
刊名:Journal of Medicinal Chemistry
出版年:2009
1
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