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SpringerLink电子期刊(1)
Elsevier电子期刊(7)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:0.017992 秒
在所有数据库中总计命中:
15
条
1.
Discovery of a Highly Selective
J
AK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms
作者:
Honghe Wan
;
Gretchen M. Schroeder
;
Amy C. Hart
;
J
ennifer Inghrim
;
J
ames Grebinski
;
J
ohn S. Tokarski
;
Matthew V. Lorenzi
;
Dan You
;
Theresa Mcdevitt
;
Becky Penhallow
;
Ragini Vuppugalla
;
Yueping Zhang
;
Xiaomei Gu
;
Ramaswamy Iyer
;
Louis
J
.
Lombardo
;
George L. Trainor
;
Stefan Ruepp
;
J
onathan Lippy
;
Yuval Blat
;
J
ohn S. Sack
;
J
aved A. Khan
;
Kevin Stefanski
;
Bogdan Sleczka
;
Arvind Mathur
;
J
ung-Hui Sun
;
Michael K. Wong
;
Dauh-Rurng Wu
;
Peng Li
;
Anuradha Gupta
;
P. N. Arunachalam
;
Bala Pragalathan
;
Sankara Narayanan
;
Nan
j
undaswamy K.C.
;
Prakasam Kuppusamy
;
Ashok V. Purandare
刊名:ACS Medicinal Chemistry Letters
出版年:2015
2.
Structure-Based Design of Selective
J
anus Kinase 2 Imidazo[4,5-d]pyrrolo[2,3-b]pyridine Inhibitors
作者:
Amy C. Hart
;
Gretchen M. Schroeder
;
Honghe Wan
;
J
ames Grebinski
;
J
ennifer Inghrim
;
J
ames Kempson
;
J
unqing Guo
;
William
J
. Pitts
;
J
ohn S. Tokarski
;
J
ohn S. Sack
;
J
aved A. Khan
;
J
onathan Lippy
;
Matthew V. Lorenzi
;
Dan You
;
Theresa McDevitt
;
Ragini Vuppugalla
;
Yueping Zhang
;
Louis
J
.
Lombardo
;
George L. Trainor
;
Ashok V. Purandare
刊名:ACS Medicinal Chemistry Letters
出版年:2015
3.
Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors
作者:
Ashvinikumar V. Gavai
;
Claude Quesnelle
;
Derek Norris
;
Wen-Ching Han
;
Patrice Gill
;
Weifang Shan
;
Aaron Balog
;
Ke Chen
;
Andrew Tebben
;
Richard Rampulla
;
Dauh-Rurng Wu
;
Yingru Zhang
;
Arvind Mathur
;
Ronald White
;
Anne Rose
;
Haiqing Wang
;
Zheng Yang
;
Asoka Ranasinghe
;
Celia D鈥橝rienzo
;
Victor Guarino
;
Lan Xiao
;
Ching Su
;
Gerry Everlof
;
Vinod Arora
;
Ding Ren Shen
;
Mary Ellen Cvi
j
ic
;
Krista Menard
;
Mei-Li Wen
;
J
ere Meredith
;
George Trainor
;
Louis
J
.
Lombardo
;
Richard Olson
;
Phil S. Baran
;
J
ohn T. Hunt
;
Gregory D. Vite
;
Bruce S. Fischer
;
Richard A. Westhouse
;
Francis Y. Lee
刊名:ACS Medicinal Chemistry Letters
出版年:2015
4.
Benzazepinones and Benzoxazepinones as Antagonists of Inhibitor of Apoptosis Proteins (IAPs) Selective for the Second Baculovirus IAP Repeat (BIR2) Domain
作者:
Andrew F. Donnell
;
Christophe Michoud
;
Kenneth C. Rupert
;
Xiaochun Han
;
Douglas Aguilar
;
Karl B. Frank
;
Adrian
J
. Fretland
;
Lin Gao
;
Barry Goggin
;
J
. Heather Hogg
;
Kyoung
j
a Hong
;
Cheryl A.
J
anson
;
Robert F. Kester
;
Norman Kong
;
Kang Le
;
Shirley Li
;
Weiling Liang
;
Louis
J
.
Lombardo
;
Yan Lou
;
Christine M. Lukacs
;
Steven Mischke
;
J
ohn A. Moliterni
;
Ann Polonskaia
;
Andrew D. Schutt
;
Dave S. Solis
;
Anthony Specian
;
Robert T. Taylor
;
Martin Weisel
;
Stacy W. Remiszewski
刊名:
J
ournal of Medicinal Chemistry
出版年:2013
5.
Optimization of Benzodiazepinones as Selective Inhibitors of the X-Linked Inhibitor of Apoptosis Protein (XIAP) Second Baculovirus IAP Repeat (BIR2) Domain
作者:
Robert F. Kester
;
Andrew F. Donnell
;
Yan Lou
;
Stacy W. Remiszewski
;
Louis
J
.
Lombardo
;
Shaoqing Chen
;
Nam T. Le
;
J
ennifer Lo
;
J
ohn A. Moliterni
;
Xiaochun Han
;
J
. Heather Hogg
;
Weiling Liang
;
Christophe Michoud
;
Kenneth C. Rupert
;
Steven Mischke
;
Kang Le
;
Martin Weisel
;
Cheryl A.
J
anson
;
Christine M. Lukacs
;
Adrian
J
. Fretland
;
Kyoung
j
a Hong
;
Ann Polonskaia
;
Lin Gao
;
Shirley Li
;
Dave S. Solis
;
Doug Aguilar
;
Christine Tardell
;
Mark Dvorozniak
;
Shahid Tannu
;
Edmund C. Lee
;
Andy D. Schutt
;
Barry Goggin
刊名:
J
ournal of Medicinal Chemistry
出版年:2013
6.
Discovery of Pyrrolopyridine−Pyridone Based Inhibitors of Met Kinase: Synthesis, X-ray Crystallographic Analysis, and Biological Activities
作者:
Kyoung Soon Kim
;
Liping Zhang
;
Robert Schmidt
;
Zhen-Wei Cai
;
Donna Wei
;
David K. Williams
;
Louis
J
.
Lombardo
;
George L. Trainor
;
Dianlin Xie
;
Yaquan Zhang
;
Yongmi An
;
J
ohn S. Sack
;
J
ohn S. Tokarski
;
C
刊名:
J
ournal of Medicinal Chemistry
出版年:2008
7.
Second Generation Tetrahydroquinoline-Based Protein Farnesyltransferase Inhibitors as Antimalarials
作者:
Pravin Bendale
;
Srinivas Olepu
;
Praveen Kumar Suryadevara
;
Vivek Bulbule
;
Kasey Rivas
;
Laxman Nallan
;
Brian Smart
;
Kohei Yokoyama
;
Sudha Ankala
;
Prakash Rao Pendyala
;
David Floyd
;
Louis
J
.
Lombardo
;
D
刊名:
J
ournal of Medicinal Chemistry
出版年:2007
1
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