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Wiley电子期刊(2)
NATURE电子期刊(4)
ACS电子期刊(4)
SpringerLink电子期刊(1)
Elsevier电子期刊(7)
在“
ACS电子期刊
”中,
命中:
4
条,耗时:小于0.01 秒
在所有数据库中总计命中:
18
条
1.
Discovery of (S)-1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development
作者:
James F. Blake
;
Michael Burkard
;
Jocelyn Chan
;
Huifen Chen
;
Kang-Jye Chou
;
Dolores Diaz
;
Danette A. Dudley
;
John J. Gaudino
;
Stephen E. Gould
;
Jonas Grina
;
Thomas Hunsaker
;
Lichuan Liu
;
Matthew Martinson
;
David Moreno
;
Lars Mueller
;
Christine Orr
;
Patricia Pacheco
;
Ann Qin
;
Kevin Rasor
;
Li Ren
;
Kirk Robarge
;
Sheerin Shahidi-Latham
;
Jeffrey Stults
;
Francis Sullivan
;
Weiru Wang
;
Jianping Yin
;
Aihe Zhou
;
Marcia
Belvin
;
Mark Merchant
;
John Moffat
;
Jacob B. Schwarz
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Back Pocket Flexibility Provides Group II p21-Activated Kinase (PAK) Selectivity for Type I 1/2 Kinase Inhibitors
作者:
Steven T. Staben
;
Jianwen A. Feng
;
Karen Lyle
;
Marcia
Belvin
;
Jason Boggs
;
Jason D. Burch
;
Ching-ching Chua
;
Haifeng Cui
;
Antonio G. DiPasquale
;
Lori S. Friedman
;
Christopher Heise
;
Hartmut Koeppen
;
Adrian Kotey
;
Robert Mintzer
;
Angela Oh
;
David Allen Roberts
;
Lionel Rouge
;
Joachim Rudolph
;
Christine Tam
;
Weiru Wang
;
Yisong Xiao
;
Amy Young
;
Yamin Zhang
;
Klaus P. Hoeflich
刊名:Journal of Medicinal Chemistry
出版年:2014
3.
Discovery and Biological Profiling of Potent and Selective mTOR Inhibitor GDC-0349
作者:
Zhonghua Pei
;
Elizabeth Blackwood
;
Lichuan Liu
;
Shiva Malek
;
Marcia
Belvin
;
Michael F. T. Koehler
;
Daniel F. Ortwine
;
Huifen Chen
;
Frederick Cohen
;
Jane R. Kenny
;
Philippe Bergeron
;
Kevin Lau
;
Cuong Ly
;
Xianrui Zhao
;
Anthony A. Estrada
;
Tom Truong
;
Jennifer A. Epler
;
Jim Nonomiya
;
Lan Trinh
;
Steve Sideris
;
John Lesnick
;
Linda Bao
;
Ulka Vijapurkar
;
Sophie Mukadam
;
Suzanne Tay
;
Gauri Deshmukh
;
Yung-Hsiang Chen
;
Xiao Ding
;
Lori S. Friedman
;
Joseph P. Lyssikatos
刊名:ACS Medicinal Chemistry Letters
出版年:2013
4.
Discovery of Novel Allosteric Mitogen-Activated Protein Kinase Kinase (MEK) 1,2 Inhibitors Possessing Bidentate Ser212 Interactions
作者:
Robert A. Heald
;
Philip Jackson
;
Pascal Savy
;
Mark Jones
;
Emanuela Gancia
;
Brenda Burton
;
Richard Newman
;
Jason Boggs
;
Emily Chan
;
Jocelyn Chan
;
Edna Choo
;
Mark Merchant
;
Patrick Rudewicz
;
Mark Ultsch
;
Christian Wiesmann
;
Qin Yue
;
Marcia
Belvin
;
Steve Price
刊名:Journal of Medicinal Chemistry
出版年:2012
1
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