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ACS电子期刊(16)
在“
ACS电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
141
条
1.
Recent Progress in Histone Demethylase Inhibitors
作者:
Tom E. McAllister
;
Katherine S. England
;
Richard J. Hopkinson
;
Paul
E. Brennan
;
Akane Kawamura
;
Christopher J.
Schofield
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors
作者:
Vassilios Bavetsias
;
Rachel M. Lanigan
;
Gian Filippo Ruda
;
Butrus Atrash
;
Mark G. McLaughlin
;
Anthony Tumber
;
N. Yi Mok
;
Yann-Vaï Le Bihan
;
Sally Dempster
;
Katherine J. Boxall
;
Fiona Jeganathan
;
Stephanie B. Hatch
;
Pavel Savitsky
;
Srikannathasan Velupillai
;
Tobias Krojer
;
Katherine S. England
;
Jimmy Sejberg
;
Ching Thai
;
Adam Donovan
;
Akos Pal
;
Giuseppe Scozzafava
;
James M. Bennett
;
Akane Kawamura
;
Catrine Johansson
;
Aleksandra Szykowska
;
Carina Gileadi
;
Nicola A. Burgess-Brown
;
Frank von Delft
;
Udo Oppermann
;
Zoe Walters
;
Janet Shipley
;
Florence I. Raynaud
;
Susan M. Westaway
;
Rab K. Prinjha
;
Oleg Fedorov
;
Rosemary Burke
;
Christopher J.
Schofield
;
Isaac M. Westwood
;
Chas Bountra
;
Susanne Müller
;
Rob L. M. van Montfort
;
Paul
E. Brennan
;
Julian Blagg
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Circumventing Seizure Activity in a Series of G Protein Coupled Receptor 119 (GPR119) Agonists
作者:
James S. Scott
;
Suzanne S. Bowker
;
Katy J. Brocklehurst
;
Hayley S. Brown
;
David S. Clarke
;
Alison Easter
;
Anne Ertan
;
Kristin Goldberg
;
Julian A. Hudson
;
Stefan Kavanagh
;
David Laber
;
Andrew G. Leach
;
Philip A. MacFaul
;
Elizabeth A. Martin
;
Darren McKerrecher
;
Paul
Schofield
;
Per H. Svensson
;
Joanne Teague
刊名:Journal of Medicinal Chemistry
出版年:2014
4.
Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains
作者:
Duncan A. Hay
;
Oleg Fedorov
;
Sarah Martin
;
Dean C. Singleton
;
Cynthia Tallant
;
Christopher Wells
;
Sarah Picaud
;
Martin Philpott
;
Octovia P. Monteiro
;
Catherine M. Rogers
;
Stuart J. Conway
;
Timothy P. C. Rooney
;
Anthony Tumber
;
Clarence Yapp
;
Panagis Filippakopoulos
;
Mark E. Bunnage
;
Susanne M眉ller
;
Stefan Knapp
;
Christopher J.
Schofield
;
Paul
E. Brennan
刊名:Journal of the American Chemical Society
出版年:2014
5.
Quantum Mechanics/Molecular Mechanics Restrained Electrostatic Potential Fitting
作者:
Steven K. Burger
;
Jeremy
Schofield
;
Paul
W. Ayers
刊名:Journal of Physical Chemistry B
出版年:2013
6.
Assay Platform for Clinically Relevant Metallo-尾-lactamases
作者:
Sander S. van Berkel
;
J眉rgen Brem
;
Anna M. Rydzik
;
Ramya Salimraj
;
Ricky Cain
;
Anil Verma
;
Raymond J. Owens
;
Colin W. G. Fishwick
;
James Spencer
;
Christopher J.
Schofield
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Discovery of a Potent, Selective, and Orally Bioavailable Acidic 11尾-Hydroxysteroid Dehydrogenase Type 1 (11尾-HSD1) Inhibitor: Discovery of 2-[(3S)-1-[5-(Cyclohexylcarbamoyl)-6-propylsulfanylpy
作者:
James S. Scott
;
Suzanne S. Bowker
;
Joanne deSchoolmeester
;
Stefan Gerhardt
;
David Hargreaves
;
Elaine Kilgour
;
Adele Lloyd
;
Rachel M. Mayers
;
William McCoull
;
Nicholas J. Newcombe
;
Derek Ogg
;
Martin J. Packer
;
Amanda Rees
;
John Revill
;
Paul
Schofield
;
Nidhal Selmi
;
John G. Swales
;
Paul
R. O. Whittamore
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain鈥揂cetyl-lysine Interactions
作者:
David S. Hewings
;
Timothy P. C. Rooney
;
Laura E. Jennings
;
Duncan A. Hay
;
Christopher J.
Schofield
;
Paul
E. Brennan
;
Stefan Knapp
;
Stuart J. Conway
刊名:Journal of Medicinal Chemistry
出版年:2012
9.
Use of Small-Molecule Crystal Structures To Address Solubility in a Novel Series of G Protein Coupled Receptor 119 Agonists: Optimization of a Lead and in Vivo Evaluation
作者:
James S. Scott
;
Alan M. Birch
;
Katy J. Brocklehurst
;
Anders Broo
;
Hayley S. Brown
;
Roger J. Butlin
;
David S. Clarke
;
脰jvind Davidsson
;
Anne Ertan
;
Kristin Goldberg
;
Sam D. Groombridge
;
Julian A. Hudson
;
David Laber
;
Andrew G. Leach
;
Philip A. MacFaul
;
Darren McKerrecher
;
Adrian Pickup
;
Paul
Schofield
;
Per H. Svensson
;
Pernilla S枚rme
;
Joanne Teague
刊名:Journal of Medicinal Chemistry
出版年:2012
10.
Plant Growth Regulator Daminozide Is a Selective Inhibitor of Human KDM2/7 Histone Demethylases
作者:
Nathan R. Rose
;
Esther C. Y. Woon
;
Anthony Tumber
;
Louise J. Walport
;
Rasheduzzaman Chowdhury
;
Xuan Shirley Li
;
Oliver N. F. King
;
Clarisse Lejeune
;
Stanley S. Ng
;
Tobias Krojer
;
Mun Chiang Chan
;
Anna M. Rydzik
;
Richard J. Hopkinson
;
Ka Hing Che
;
Michelle Daniel
;
Claire Strain-Damerell
;
Carina Gileadi
;
Grazyna Kochan
;
Ivanhoe K. H. Leung
;
James Dunford
;
Kar Kheng Yeoh
;
Peter J. Ratcliffe
;
Nicola Burgess-Brown
;
Frank von Delft
;
Susanne Muller
;
Brian Marsden
;
Paul
E. Brennan
;
Michael A. McDonough
;
Udo Oppermann
;
Robert J. Klose
;
Christopher J.
Schofield
;
Akane Kawamura
刊名:Journal of Medicinal Chemistry
出版年:2012
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