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ACS电子期刊(11)
在“
ACS电子期刊
”中,
命中:
11
条,耗时:小于0.01 秒
在所有数据库中总计命中:
103
条
1.
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials
作者:
T. G. Murali Dhar
;
Hai-Yun Xiao
;
Jenny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurng Wu
;
Marta Dabros
;
Xiaoxia Yang
;
Tracy
L.
Taylor
;
Xia D. Zhou
;
Elizabeth M. Heimrich
;
Rochelle Thomas
;
Kim W. McIntyre
;
Bethanne Warrack
;
Hong Shi
;
Paul C. Levesque
;
Jia L. Zhu
;
James Hennan
;
Praveen Balimane
;
Zheng Yang
;
Anthony M. Marino
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Arvind Mathur
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery and Structure–Activity Relationship (SAR) of a Series of Ethanolamine-Based Direct-Acting Agonists of Sphingosine-1-phosphate (S1P1)
作者:
John L. Gilmore
;
James E. Sheppeck II
;
Scott H. Watterson
;
Lauren Haque
;
Parag Mukhopadhyay
;
Andrew J. Tebben
;
Michael A. Galella
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Virna Borowski
;
Kathleen Gillooly
;
Tracy
Taylor
;
Kim W. McIntyre
;
Bethanne Warrack
;
Paul C. Levesque
;
Julia P. Li
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Luisa Salter-Cid
;
Joel C. Barrish
;
William J. Pitts
;
Percy H. Carter
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 2. Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives
作者:
Susan M. Westaway
;
Alex G. S. Preston
;
Michael D. Barker
;
Fiona Brown
;
Jack A. Brown
;
Matthew Campbell
;
Chun-wa Chung
;
Gerard Drewes
;
Robert Eagle
;
Neil Garton
;
Laurie Gordon
;
Carl Haslam
;
Thomas G. Hayhow
;
Philip G. Humphreys
;
Gerard Joberty
;
Roy Katso
;
Laurens Kruidenier
;
Melanie Leveridge
;
Michelle Pemberton
;
Inma Rioja
;
Gail A. Seal
;
Tracy
Shipley
;
Onkar Singh
;
Colin J. Suckling
;
Joanna
Taylor
;
Pamela Thomas
;
David M. Wilson
;
Kevin Lee
;
Rab K. Prinjha
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Potent and Selective Agonists of Sphingosine 1-Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series
作者:
Scott H. Watterson
;
Junqing Guo
;
Steve H. Spergel
;
Charles M. Langevine
;
Robert V. Moquin
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Dana Banas
;
Richard Liu
;
Suzanne J. Suchard
;
Kathleen Gillooly
;
Tracy
Taylor
;
Sandra Rex-Rabe
;
David J. Shuster
;
Kim W. McIntyre
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Bethanne Warrack
;
Luisa Salter-Cid
;
Murray McKinnon
;
Joel C. Barrish
;
Percy H. Carter
;
William J. Pitts
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator
作者:
Michael G. YangZili Xiao
;
T. G. Murali Dhar
;
Hai-Yun Xiao
;
John L. Gilmore
;
David Marcoux
;
Jenny H. Xie
;
Kim W. McIntyre
;
Tracy
L.
Taylor
;
Virna Borowski
;
Elizabeth Heimrich
;
Yu-Wen Li
;
Jianlin Feng
;
Alda Fernandes
;
Zheng Yang
;
Praveen Balimane
;
Anthony M. Marino
;
Georgia Cornelius
;
Bethanne M. Warrack
;
Arvind Mathur
;
Dauh-Rurng Wu
;
Peng Li
;
Anuradha Gupta
;
Bala Pragalathan
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Lois D. Lehman-McKeeman
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Discovery of a Potent and Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300
作者:
Terry D. Crawford
;
F. Anthony Romero
;
Kwong Wah Lai
;
Vickie Tsui
;
Alexander M.
Taylor
;
Gladys de Leon Boenig
;
Cameron L. Noland
;
Jeremy Murray
;
Justin Ly
;
Edna F. Choo
;
Thomas L. Hunsaker
;
Emily W. Chan
;
Mark Merchant
;
Samir Kharbanda
;
Karen E. Gascoigne
;
Susan Kaufman
;
Maureen H. Beresini
;
Jiangpeng Liao
;
Wenfeng Liu
;
Kevin X. Chen
;
Zhongguo Chen
;
Andrew R. Conery
;
Alexandre Côté
;
Hariharan Jayaram
;
Ying Jiang
;
James R. Kiefer
;
Tracy
Kleinheinz
;
Yingjie Li
;
Jonathan Maher
;
Eneida Pardo
;
Florence Poy
;
Kerry L. Spillane
;
Fei Wang
;
Jian Wang
;
Xiaocang Wei
;
Zhaowu Xu
;
Zhongya Xu
;
Ivana Yen
;
Laura Zawadzke
;
Xiaoyu Zhu
;
Steven Bellon
;
Richard Cummings
;
Andrea G. Cochran
;
Brian K. Albrecht
;
Steven Magnuson
刊名:Journal of Medicinal Chemistry
出版年:2016
7.
Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked
作者:
Scott H. Watterson
;
George V. De Lucca
;
Qing Shi
;
Charles M. Langevine
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Hua Gong
;
Jun Dai
;
Shiuhang Yip
;
Peng Li
;
Dawn Sun
;
Dauh-Rurng Wu
;
Chunlei Wang
;
Yingru Zhang
;
Sarah C. Traeger
;
Mark A. Pattoli
;
Stacey Skala
;
Lihong Cheng
;
Mary T. Obermeier
;
Rodney Vickery
;
Lorell N. Discenza
;
Celia J. D’Arienzo
;
Yifan Zhang
;
Elizabeth Heimrich
;
Kathleen M. Gillooly
;
Tracy
L.
Taylor
;
Claudine Pulicicchio
;
Kim W. McIntyre
;
Michael A. Galella
;
Andy J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing Chang
;
Richard Rampulla
;
Arvind Mathur
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Aberra Fura
;
James R. Burke
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
8.
Small Molecule Reversible Inhibitors of Bruton’s Tyrosine Kinase (BTK): Structure–Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177)
作者:
George V. De Lucca
;
Qing Shi
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Rick Rampulla
;
Arvind Mathur
;
Lorell Discenza
;
Celia D’Arienzo
;
Jun Dai
;
Mary Obermeier
;
Rodney Vickery
;
Yingru Zhang
;
Zheng Yang
;
Punit Marathe
;
Andrew J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing J. Chang
;
Huiping Zhang
;
Kathleen Gillooly
;
Tracy
Taylor
;
Mark A. Pattoli
;
Stacey Skala
;
Daniel W. Kukral
;
Kim W. McIntyre
;
Luisa Salter-Cid
;
Aberra Fura
;
James R. Burke
;
Joel C. Barrish
;
Percy H. Carter
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
9.
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
作者:
Hai-Yun Xiao
;
Scott H. Watterson
;
Charles M. Langevine
;
Anurag S. Srivastava
;
Soo S. Ko
;
Yanlei Zhang
;
Robert J. Cherney
;
Wei-Wei Guo
;
John L. Gilmore
;
James E. Sheppeck II
;
Dauh-Rurng Wu
;
Peng Li
;
Duraisamy Ramasamy
;
Piramanayagam Arunachalam
;
Arvind Mathur
;
Tracy
L.
Taylor
;
David J. Shuster
;
Kim W. McIntyre
;
Ding-Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Anthony M. Marino
;
Praveen V. Balimane
;
Zheng Yang
;
Dana M. Banas
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Bethanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Salter-Cid
;
Jenny Xie
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
;
T. G. Murali Dhar
刊名:Journal of Medicinal Chemistry
出版年:2016
10.
Discovery of ((4-(5-(Cyclopropylcarbamoyl)-2-methylphenylamino)-5-methylpyrrolo[1,2-f][1,2,4]triazine-6-carbonyl)(propyl)carbamoyloxy)methyl-2-(4-(phosphonooxy)phenyl)acetate聽(BMS-751324), a Cl
作者:
Chunjian Liu
;
James Lin
;
John Hynes
;
Hong Wu
;
Stephen T. Wrobleski
;
Shuqun Lin
;
T. G. Murali Dhar
;
Vivekananda M. Vrudhula
;
Jung-Hui Sun
;
Sam Chao
;
Rulin Zhao
;
Bei Wang
;
Bang-Chi Chen
;
Gerry Everlof
;
Christoph Gesenberg
;
Hongjian Zhang
;
Punit H. Marathe
;
Kim W. McIntyre
;
Tracy
L.
Taylor
;
Kathleen Gillooly
;
David J. Shuster
;
Murray McKinnon
;
John H. Dodd
;
Joel C. Barrish
;
Gary L. Schieven
;
Katerina Leftheris
刊名:Journal of Medicinal Chemistry
出版年:2015
1
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